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CAS No.: 96206-92-7
MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors.
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01024491 | Premature Ejaculation | Phase 3 | Completed | - | Mexico ... more >> Asociacion Mexicana para la Salud Sexual, A.C. Mexico City, Mexico D.F., Mexico, 14000 Centro Especializado en Urología y Andrología del Hospital Star Médica Mexico City, Mexico D.F, Mexico, 06700 Collapse << |
NCT03506945 | Depressive Symptoms ... more >> Stress, Psychological Collapse << | Not Applicable | Not yet recruiting | July 2023 | United States, California ... more >> University of California San Diego La Jolla, California, United States, 92093 Collapse << |
实验方案
技术信息
CAS号 | 96206-92-7 | 储存条件 |
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分子式 | C14H11N | 运输 | 蓝冰 | |||||
分子量 | 193.24 | 别名 | ||||||
溶解度 |
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动物实验配方 |