CAS No.: 1346133-08-1
LY2795050 Catalog No. CSN17719
LY2795050 is a selective κ-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 临床研究
NCT号 适应症或疾病 临床期 招募状态 预计完成时间 地点 NCT02236702 - - Terminated(The original PI, Al... more >>exander Neumeister, left NYULMC. No data was analyzed.) Collapse << - United States, New York ... more >> NYU School of Medicine New York, New York, United States, 10016 Collapse << NCT02237703 - - Terminated(The original PI, Al... more >>exander Neumeister, left NYULMC. No data was analyzed.) Collapse << - United States, New York ... more >> NYU School of Medicine New York, New York, United States, 10016 Collapse << - 参考文献
- [1] Zheng MQ, Nabulsi N, et al. Synthesis and evaluation of 11C-LY2795050 as a κ-opioid receptor antagonist radiotracer for PET imaging. J Nucl Med. 2013 Mar;54(3):455-63.
- [2] Mitch CH, Quimby SJ, et al. Discovery of aminobenzyloxyarylamides as κ opioid receptor selective antagonists: application to preclinical development of a κ opioid receptor antagonist receptor occupancy tracer. J Med Chem. 2011 Dec 8;54(23):8000-12.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 1346133-08-1 | 储存条件 |
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| 分子式 | C23H22ClN3O2 | 运输 | 蓝冰 | |
| 分子量 | 407.89 | 别名 |
