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CAS No.: 1373215-15-6
Synonyms: Z-FL-COCHO;Cathepsin S Inhibitor
LY 3000328 is a highly selective and potent Cathepsin S inhibitor with IC50 of 7.7±5.85 nM and 1.67±1.17 nM for hCat S and mCat S respectively, can be used in treatment for abdominal aortic aneurysm.
生物活性
动物研究 | |
剂量 | Mice: 1 mg/kg - 10 mg/kg[1] (p.o.,BID) |
给药途径 | p.o. |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01515358 | Healthy Volunteers | Phase 1 | Completed | - | Singapore ... more >> For additional information regarding investigative sites for this trial, contact 1-877-CTLILLY (1-877-285-4559, 1-317-615-4559) Mon - Fri from 9 AM to 5 PM Eastern Time (UTC/GMT - 5 hours, EST), or speak with your personal physician. Singapore, Singapore, 117597 Collapse << |
实验方案
技术信息
CAS号 | 1373215-15-6 | 储存条件 |
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分子式 | C25H29FN4O5 | 运输 | 蓝冰 | |||||
分子量 | 484.52 | 别名 | Z-FL-COCHO;Cathepsin S Inhibitor | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01515358 | Healthy Volunteers | Phase 1 | Completed | - | Singapore ... more >> For additional information regarding investigative sites for this trial, contact 1-877-CTLILLY (1-877-285-4559, 1-317-615-4559) Mon - Fri from 9 AM to 5 PM Eastern Time (UTC/GMT - 5 hours, EST), or speak with your personal physician. Singapore, Singapore, 117597 Collapse << |
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