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CAS No.: 747412-49-3
Synonyms: VER-52296;AUY922;NVP-AUY922
AUY922 is a highly potent HSP90 inhibitor for HSP90α/β with IC50 of 13 nM /21 nM, weaker potency against the HSP90 family members GRP94 and TRAP-1.
生物活性
实验方案
技术信息
CAS号 | 747412-49-3 | 储存条件 |
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分子式 | C26H31N3O5 | 运输 | 蓝冰 | |||||||
分子量 | 465.54 | 别名 | VER-52296;AUY922;NVP-AUY922 | |||||||
溶解度 |
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动物实验配方 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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22RV1 | - | Growth Inhibition Assay | - | IC50=0.03507 μM | SANGER |
23132-87 | - | Growth Inhibition Assay | - | IC50=0.10488 μM | SANGER |
5637 | - | Growth Inhibition Assay | - | IC50=0.02822 μM | SANGER |
639-V | - | Growth Inhibition Assay | - | IC50=0.00485 μM | SANGER |
647-V | - | Growth Inhibition Assay | - | IC50=0.14942 μM | SANGER |
697 | - | Growth Inhibition Assay | - | IC50=0.02031 μM | SANGER |
769-P | - | Growth Inhibition Assay | - | IC50=0.01073 μM | SANGER |
786-0 | - | Growth Inhibition Assay | - | IC50=0.00663 μM | SANGER |
8305C | - | Growth Inhibition Assay | - | IC50=0.03072 μM | SANGER |
8505C | - | Growth Inhibition Assay | - | IC50=0.00821 μM | SANGER |
8-MG-BA | - | Growth Inhibition Assay | - | IC50=0.01884 μM | SANGER |
A101D | - | Growth Inhibition Assay | - | IC50=0.01987 μM | SANGER |
A172 | - | Growth Inhibition Assay | - | IC50=0.0395 μM | SANGER |
A204 | - | Growth Inhibition Assay | - | IC50=0.02115 μM | SANGER |
A2058 | - | Growth Inhibition Assay | - | IC50=0.02929 μM | SANGER |
A253 | - | Growth Inhibition Assay | - | IC50=0.05052 μM | SANGER |
A2780 | - | Growth Inhibition Assay | - | IC50=0.01715 μM | SANGER |
A375 | - | Growth Inhibition Assay | - | IC50=0.02171 μM | SANGER |
A388 | - | Growth Inhibition Assay | - | IC50=0.02115 μM | SANGER |
A3-KAW | - | Growth Inhibition Assay | - | IC50=0.22708 μM | SANGER |
A427 | - | Growth Inhibition Assay | - | IC50=0.01299 μM | SANGER |
A431 | - | Growth Inhibition Assay | - | IC50=0.00607 μM | SANGER |
A498 | - | Growth Inhibition Assay | - | IC50=5.21251 μM | SANGER |
A4-Fuk | - | Growth Inhibition Assay | - | IC50=0.01702 μM | SANGER |
A673 | - | Growth Inhibition Assay | - | IC50=0.10431 μM | SANGER |
A704 | - | Growth Inhibition Assay | - | IC50=0.34923 μM | SANGER |
ABC-1 | - | Growth Inhibition Assay | - | IC50=0.08759 μM | SANGER |
ACHN | - | Growth Inhibition Assay | - | IC50=0.02345 μM | SANGER |
ACN | - | Growth Inhibition Assay | - | IC50=0.01657 μM | SANGER |
AGS | - | Growth Inhibition Assay | - | IC50=0.01061 μM | SANGER |
ALL-PO | - | Growth Inhibition Assay | - | IC50=0.01735 μM | SANGER |
AM-38 | - | Growth Inhibition Assay | - | IC50=0.01302 μM | SANGER |
AN3-CA | - | Growth Inhibition Assay | - | IC50=0.01017 μM | SANGER |
ARH-77 | - | Growth Inhibition Assay | - | IC50=0.05395 μM | SANGER |
AsPC-1 | - | Growth Inhibition Assay | - | IC50=2.53929 μM | SANGER |
ATN-1 | - | Growth Inhibition Assay | - | IC50=0.85115 μM | SANGER |
AU565 | - | Growth Inhibition Assay | - | IC50=0.11831 μM | SANGER |
BB30-HNC | - | Growth Inhibition Assay | - | IC50=0.00952 μM | SANGER |
BB49-HNC | - | Growth Inhibition Assay | - | IC50=0.01077 μM | SANGER |
BB65-RCC | - | Growth Inhibition Assay | - | IC50=0.01204 μM | SANGER |
BC-1 | - | Growth Inhibition Assay | - | IC50=0.03367 μM | SANGER |
BC-3 | - | Growth Inhibition Assay | - | IC50=0.03018 μM | SANGER |
BCPAP | - | Growth Inhibition Assay | - | IC50=0.02646 μM | SANGER |
BE-13 | - | Growth Inhibition Assay | - | IC50=0.27249 μM | SANGER |
Becker | - | Growth Inhibition Assay | - | IC50=0.01514 μM | SANGER |
BEN | - | Growth Inhibition Assay | - | IC50=0.11607 μM | SANGER |
BFTC-905 | - | Growth Inhibition Assay | - | IC50=0.00938 μM | SANGER |
BFTC-909 | - | Growth Inhibition Assay | - | IC50=0.03125 μM | SANGER |
BHT-101 | - | Growth Inhibition Assay | - | IC50=0.05876 μM | SANGER |
BHY | - | Growth Inhibition Assay | - | IC50=0.01912 μM | SANGER |
BL-41 | - | Growth Inhibition Assay | - | IC50=0.05596 μM | SANGER |
BL-70 | - | Growth Inhibition Assay | - | IC50=0.03389 μM | SANGER |
BOKU | - | Growth Inhibition Assay | - | IC50=0.06674 μM | SANGER |
BPH-1 | - | Growth Inhibition Assay | - | IC50=0.0103 μM | SANGER |
BT-20 | - | Growth Inhibition Assay | - | IC50=0.31099 μM | SANGER |
BT-474 | - | Growth Inhibition Assay | - | IC50=0.07061 μM | SANGER |
BV-173 | - | Growth Inhibition Assay | - | IC50=0.03426 μM | SANGER |
BxPC-3 | - | Growth Inhibition Assay | - | IC50=0.04341 μM | SANGER |
C2BBe1 | - | Growth Inhibition Assay | - | IC50=0.19893 μM | SANGER |
C32 | - | Growth Inhibition Assay | - | IC50=0.57313 μM | SANGER |
C-33-A | - | Growth Inhibition Assay | - | IC50=0.01509 μM | SANGER |
C3A | - | Growth Inhibition Assay | - | IC50=0.02475 μM | SANGER |
C-4-II | - | Growth Inhibition Assay | - | IC50=0.1217 μM | SANGER |
C8166 | - | Growth Inhibition Assay | - | IC50=0.01129 μM | SANGER |
CA46 | - | Growth Inhibition Assay | - | IC50=0.0543 μM | SANGER |
Ca9-22 | - | Growth Inhibition Assay | - | IC50=0.02796 μM | SANGER |
CAKI-1 | - | Growth Inhibition Assay | - | IC50=0.25086 μM | SANGER |
CAL-120 | - | Growth Inhibition Assay | - | IC50=0.04241 μM | SANGER |
CAL-12T | - | Growth Inhibition Assay | - | IC50=0.00922 μM | SANGER |
CAL-148 | - | Growth Inhibition Assay | - | IC50=0.24282 μM | SANGER |
CAL-27 | - | Growth Inhibition Assay | - | IC50=0.08156 μM | SANGER |
CAL-33 | - | Growth Inhibition Assay | - | IC50=0.04375 μM | SANGER |
CAL-39 | - | Growth Inhibition Assay | - | IC50=0.0142 μM | SANGER |
CAL-51 | - | Growth Inhibition Assay | - | IC50=0.00325 μM | SANGER |
CAL-54 | - | Growth Inhibition Assay | - | IC50=2.26795 μM | SANGER |
CAL-62 | - | Growth Inhibition Assay | - | IC50=0.0257 μM | SANGER |
CAL-72 | - | Growth Inhibition Assay | - | IC50=0.1659 μM | SANGER |
CAL-85-1 | - | Growth Inhibition Assay | - | IC50=0.01192 μM | SANGER |
Calu-1 | - | Growth Inhibition Assay | - | IC50=0.07332 μM | SANGER |
Calu-3 | - | Growth Inhibition Assay | - | IC50=0.03789 μM | SANGER |
Calu-6 | - | Growth Inhibition Assay | - | IC50=0.07965 μM | SANGER |
CAMA-1 | - | Growth Inhibition Assay | - | IC50=0.06303 μM | SANGER |
Caov-3 | - | Growth Inhibition Assay | - | IC50=2.00625 μM | SANGER |
CAPAN-1 | - | Growth Inhibition Assay | - | IC50=0.07143 μM | SANGER |
Capan-2 | - | Growth Inhibition Assay | - | IC50=0.00638 μM | SANGER |
CaR-1 | - | Growth Inhibition Assay | - | IC50=0.50367 μM | SANGER |
CAS-1 | - | Growth Inhibition Assay | - | IC50=0.11964 μM | SANGER |
Ca-Ski | - | Growth Inhibition Assay | - | IC50=0.03784 μM | SANGER |
CCF-STTG1 | - | Growth Inhibition Assay | - | IC50=0.00297 μM | SANGER |
CCRF-CEM | - | Growth Inhibition Assay | - | IC50=0.02329 μM | SANGER |
CESS | - | Growth Inhibition Assay | - | IC50=0.0312 μM | SANGER |
CGTH-W-1 | - | Growth Inhibition Assay | - | IC50=0.02328 μM | SANGER |
ChaGo-K-1 | - | Growth Inhibition Assay | - | IC50=0.12699 μM | SANGER |
CHL-1 | - | Growth Inhibition Assay | - | IC50=0.04169 μM | SANGER |
CHP-126 | - | Growth Inhibition Assay | - | IC50=0.07565 μM | SANGER |
CHP-212 | - | Growth Inhibition Assay | - | IC50=0.02212 μM | SANGER |
CMK | - | Growth Inhibition Assay | - | IC50=0.000125 μM | SANGER |
COLO-205 | - | Growth Inhibition Assay | - | IC50=0.04919 μM | SANGER |
COLO-320-HSR | - | Growth Inhibition Assay | - | IC50=0.18493 μM | SANGER |
COLO-668 | - | Growth Inhibition Assay | - | IC50=0.07984 μM | SANGER |
COLO-678 | - | Growth Inhibition Assay | - | IC50=0.33389 μM | SANGER |
COLO-679 | - | Growth Inhibition Assay | - | IC50=0.03107 μM | SANGER |
COLO-680N | - | Growth Inhibition Assay | - | IC50=0.04407 μM | SANGER |
COLO-684 | - | Growth Inhibition Assay | - | IC50=0.08158 μM | SANGER |
COLO-741 | - | Growth Inhibition Assay | - | IC50=0.05531 μM | SANGER |
COLO-792 | - | Growth Inhibition Assay | - | IC50=0.08855 μM | SANGER |
COLO-800 | - | Growth Inhibition Assay | - | IC50=3.33897 μM | SANGER |
COLO-824 | - | Growth Inhibition Assay | - | IC50=0.1102 μM | SANGER |
COLO-829 | - | Growth Inhibition Assay | - | IC50=0.34452 μM | SANGER |
COR-L105 | - | Growth Inhibition Assay | - | IC50=0.01911 μM | SANGER |
COR-L23 | - | Growth Inhibition Assay | - | IC50=0.02713 μM | SANGER |
COR-L279 | - | Growth Inhibition Assay | - | IC50=0.15836 μM | SANGER |
COR-L88 | - | Growth Inhibition Assay | - | IC50=0.17114 μM | SANGER |
CP50-MEL-B | - | Growth Inhibition Assay | - | IC50=0.08368 μM | SANGER |
CP66-MEL | - | Growth Inhibition Assay | - | IC50=0.07887 μM | SANGER |
CPC-N | - | Growth Inhibition Assay | - | IC50=11.007 μM | SANGER |
CTB-1 | - | Growth Inhibition Assay | - | IC50=0.13469 μM | SANGER |
CTV-1 | - | Growth Inhibition Assay | - | IC50=0.04116 μM | SANGER |
D-263MG | - | Growth Inhibition Assay | - | IC50=0.05683 μM | SANGER |
D-283MED | - | Growth Inhibition Assay | - | IC50=3.18937 μM | SANGER |
D-392MG | - | Growth Inhibition Assay | - | IC50=0.03842 μM | SANGER |
D-502MG | - | Growth Inhibition Assay | - | IC50=0.4803 μM | SANGER |
D-542MG | - | Growth Inhibition Assay | - | IC50=0.13965 μM | SANGER |
Daoy | - | Growth Inhibition Assay | - | IC50=0.00695 μM | SANGER |
Daudi | - | Growth Inhibition Assay | - | IC50=0.03376 μM | SANGER |
DB | - | Growth Inhibition Assay | - | IC50=0.22865 μM | SANGER |
DBTRG-05MG | - | Growth Inhibition Assay | - | IC50=0.02955 μM | SANGER |
DEL | - | Growth Inhibition Assay | - | IC50=0.11192 μM | SANGER |
Detroit562 | - | Growth Inhibition Assay | - | IC50=0.03872 μM | SANGER |
DG-75 | - | Growth Inhibition Assay | - | IC50=2.48576 μM | SANGER |
DJM-1 | - | Growth Inhibition Assay | - | IC50=0.04272 μM | SANGER |
DK-MG | - | Growth Inhibition Assay | - | IC50=0.07526 μM | SANGER |
DMS-114 | - | Growth Inhibition Assay | - | IC50=0.3612 μM | SANGER |
DMS-153 | - | Growth Inhibition Assay | - | IC50=0.07735 μM | SANGER |
DMS-273 | - | Growth Inhibition Assay | - | IC50=0.03479 μM | SANGER |
DMS-53 | - | Growth Inhibition Assay | - | IC50=0.12276 μM | SANGER |
DMS-79 | - | Growth Inhibition Assay | - | IC50=0.77845 μM | SANGER |
DOHH-2 | - | Growth Inhibition Assay | - | IC50=0.18569 μM | SANGER |
DOK | - | Growth Inhibition Assay | - | IC50=0.2593 μM | SANGER |
DoTc2-4510 | - | Growth Inhibition Assay | - | IC50=0.02122 μM | SANGER |
DSH1 | - | Growth Inhibition Assay | - | IC50=0.0627 μM | SANGER |
DU-145 | - | Growth Inhibition Assay | - | IC50=0.0129 μM | SANGER |
DU-4475 | - | Growth Inhibition Assay | - | IC50=0.0215 μM | SANGER |
DV-90 | - | Growth Inhibition Assay | - | IC50=18.9945 μM | SANGER |
EB2 | - | Growth Inhibition Assay | - | IC50=0.07285 μM | SANGER |
EB-3 | - | Growth Inhibition Assay | - | IC50=0.22376 μM | SANGER |
ECC4 | - | Growth Inhibition Assay | - | IC50=0.19863 μM | SANGER |
EC-GI-10 | - | Growth Inhibition Assay | - | IC50=0.77975 μM | SANGER |
EFE-184 | - | Growth Inhibition Assay | - | IC50=0.24597 μM | SANGER |
EFM-19 | - | Growth Inhibition Assay | - | IC50=0.33132 μM | SANGER |
EFO-21 | - | Growth Inhibition Assay | - | IC50=0.08991 μM | SANGER |
EFO-27 | - | Growth Inhibition Assay | - | IC50=0.01017 μM | SANGER |
EGI-1 | - | Growth Inhibition Assay | - | IC50=0.1797 μM | SANGER |
EHEB | - | Growth Inhibition Assay | - | IC50=0.02555 μM | SANGER |
EKVX | - | Growth Inhibition Assay | - | IC50=0.10483 μM | SANGER |
EM-2 | - | Growth Inhibition Assay | - | IC50=2.20293 μM | SANGER |
EoL-1-cell | - | Growth Inhibition Assay | - | IC50=1.58889 μM | SANGER |
ES1 | - | Growth Inhibition Assay | - | IC50=0.00266 μM | SANGER |
ES3 | - | Growth Inhibition Assay | - | IC50=0.08763 μM | SANGER |
ES4 | - | Growth Inhibition Assay | - | IC50=0.01502 μM | SANGER |
ES5 | - | Growth Inhibition Assay | - | IC50=5.61178 μM | SANGER |
ES6 | - | Growth Inhibition Assay | - | IC50=0.01261 μM | SANGER |
ES7 | - | Growth Inhibition Assay | - | IC50=0.03374 μM | SANGER |
ES8 | - | Growth Inhibition Assay | - | IC50=0.03538 μM | SANGER |
ESS-1 | - | Growth Inhibition Assay | - | IC50=0.07868 μM | SANGER |
ETK-1 | - | Growth Inhibition Assay | - | IC50=0.02806 μM | SANGER |
EVSA-T | - | Growth Inhibition Assay | - | IC50=0.09265 μM | SANGER |
EW-1 | - | Growth Inhibition Assay | - | IC50=0.02822 μM | SANGER |
EW-11 | - | Growth Inhibition Assay | - | IC50=0.07535 μM | SANGER |
EW-13 | - | Growth Inhibition Assay | - | IC50=0.00518 μM | SANGER |
EW-16 | - | Growth Inhibition Assay | - | IC50=0.00749 μM | SANGER |
EW-18 | - | Growth Inhibition Assay | - | IC50=0.10604 μM | SANGER |
EW-24 | - | Growth Inhibition Assay | - | IC50=0.2881 μM | SANGER |
EW-3 | - | Growth Inhibition Assay | - | IC50=0.17486 μM | SANGER |
EW-7 | - | Growth Inhibition Assay | - | IC50=0.00754 μM | SANGER |
FADU | - | Growth Inhibition Assay | - | IC50=0.06745 μM | SANGER |
FTC-133 | - | Growth Inhibition Assay | - | IC50=2.53689 μM | SANGER |
G-361 | - | Growth Inhibition Assay | - | IC50=0.02677 μM | SANGER |
G-401 | - | Growth Inhibition Assay | - | IC50=0.01025 μM | SANGER |
G-402 | - | Growth Inhibition Assay | - | IC50=0.03614 μM | SANGER |
GAK | - | Growth Inhibition Assay | - | IC50=0.05734 μM | SANGER |
GAMG | - | Growth Inhibition Assay | - | IC50=0.01371 μM | SANGER |
GB-1 | - | Growth Inhibition Assay | - | IC50=0.02188 μM | SANGER |
GCIY | - | Growth Inhibition Assay | - | IC50=0.02055 μM | SANGER |
GCT | - | Growth Inhibition Assay | - | IC50=0.04161 μM | SANGER |
GDM-1 | - | Growth Inhibition Assay | - | IC50=0.0084 μM | SANGER |
GI-1 | - | Growth Inhibition Assay | - | IC50=0.14772 μM | SANGER |
GI-ME-N | - | Growth Inhibition Assay | - | IC50=0.07426 μM | SANGER |
GMS-10 | - | Growth Inhibition Assay | - | IC50=0.13444 μM | SANGER |
GOTO | - | Growth Inhibition Assay | - | IC50=0.17246 μM | SANGER |
GP5d | - | Growth Inhibition Assay | - | IC50=0.02723 μM | SANGER |
GR-ST | - | Growth Inhibition Assay | - | IC50=0.1021 μM | SANGER |
GT3TKB | - | Growth Inhibition Assay | - | IC50=0.01202 μM | SANGER |
H4 | - | Growth Inhibition Assay | - | IC50=0.01366 μM | SANGER |
HAL-01 | - | Growth Inhibition Assay | - | IC50=0.99379 μM | SANGER |
HC-1 | - | Growth Inhibition Assay | - | IC50=0.04069 μM | SANGER |
HCC1143 | - | Growth Inhibition Assay | - | IC50=2.50658 μM | SANGER |
HCC1187 | - | Growth Inhibition Assay | - | IC50=1.55522 μM | SANGER |
HCC1395 | - | Growth Inhibition Assay | - | IC50=2.98602 μM | SANGER |
HCC1419 | - | Growth Inhibition Assay | - | IC50=0.09541 μM | SANGER |
HCC1569 | - | Growth Inhibition Assay | - | IC50=0.03608 μM | SANGER |
HCC1599 | - | Growth Inhibition Assay | - | IC50=0.09601 μM | SANGER |
HCC1806 | - | Growth Inhibition Assay | - | IC50=0.11108 μM | SANGER |
HCC1937 | - | Growth Inhibition Assay | - | IC50=0.04456 μM | SANGER |
HCC1954 | - | Growth Inhibition Assay | - | IC50=0.64726 μM | SANGER |
HCC2157 | - | Growth Inhibition Assay | - | IC50=0.05733 μM | SANGER |
HCC2218 | - | Growth Inhibition Assay | - | IC50=0.09999 μM | SANGER |
HCC2998 | - | Growth Inhibition Assay | - | IC50=0.02945 μM | SANGER |
HCC38 | - | Growth Inhibition Assay | - | IC50=0.03771 μM | SANGER |
HCC70 | - | Growth Inhibition Assay | - | IC50=0.05452 μM | SANGER |
HCE-4 | - | Growth Inhibition Assay | - | IC50=0.02145 μM | SANGER |
HCE-T | - | Growth Inhibition Assay | - | IC50=0.0286 μM | SANGER |
HCT-116 | - | Growth Inhibition Assay | - | IC50=0.15169 μM | SANGER |
HCT-15 | - | Growth Inhibition Assay | - | IC50=0.06597 μM | SANGER |
HDLM-2 | - | Growth Inhibition Assay | - | IC50=0.04114 μM | SANGER |
HD-MY-Z | - | Growth Inhibition Assay | - | IC50=0.14429 μM | SANGER |
HEC-1 | - | Growth Inhibition Assay | - | IC50=0.07161 μM | SANGER |
HEL | - | Growth Inhibition Assay | - | IC50=0.03891 μM | SANGER |
HGC-27 | - | Growth Inhibition Assay | - | IC50=0.01758 μM | SANGER |
HH | - | Growth Inhibition Assay | - | IC50=0.14201 μM | SANGER |
HL-60 | - | Growth Inhibition Assay | - | IC50=0.01807 μM | SANGER |
HLE | - | Growth Inhibition Assay | - | IC50=0.06082 μM | SANGER |
HMV-II | - | Growth Inhibition Assay | - | IC50=0.00449 μM | SANGER |
HN | - | Growth Inhibition Assay | - | IC50=0.02593 μM | SANGER |
HO-1-N-1 | - | Growth Inhibition Assay | - | IC50=0.02549 μM | SANGER |
HOP-62 | - | Growth Inhibition Assay | - | IC50=0.01542 μM | SANGER |
HOP-92 | - | Growth Inhibition Assay | - | IC50=0.07711 μM | SANGER |
HOS | - | Growth Inhibition Assay | - | IC50=0.00138 μM | SANGER |
HPAF-II | - | Growth Inhibition Assay | - | IC50=0.41117 μM | SANGER |
Hs-578-T | - | Growth Inhibition Assay | - | IC50=18.5759 μM | SANGER |
HSC-2 | - | Growth Inhibition Assay | - | IC50=0.00518 μM | SANGER |
HSC-3 | - | Growth Inhibition Assay | - | IC50=0.00641 μM | SANGER |
HSC-4 | - | Growth Inhibition Assay | - | IC50=0.1716 μM | SANGER |
HT | - | Growth Inhibition Assay | - | IC50=0.22566 μM | SANGER |
HT-1080 | - | Growth Inhibition Assay | - | IC50=0.02214 μM | SANGER |
HT-1197 | - | Growth Inhibition Assay | - | IC50=0.01685 μM | SANGER |
HT-1376 | - | Growth Inhibition Assay | - | IC50=0.09861 μM | SANGER |
HT-144 | - | Growth Inhibition Assay | - | IC50=0.00155 μM | SANGER |
HT-29 | - | Growth Inhibition Assay | - | IC50=0.04357 μM | SANGER |
HT-3 | - | Growth Inhibition Assay | - | IC50=0.8942 μM | SANGER |
HT55 | - | Growth Inhibition Assay | - | IC50=2.62019 μM | SANGER |
HTC-C3 | - | Growth Inhibition Assay | - | IC50=0.02607 μM | SANGER |
HuCCT1 | - | Growth Inhibition Assay | - | IC50=0.02961 μM | SANGER |
HuH-7 | - | Growth Inhibition Assay | - | IC50=0.07035 μM | SANGER |
HuO-3N1 | - | Growth Inhibition Assay | - | IC50=1.83412 μM | SANGER |
HuP-T3 | - | Growth Inhibition Assay | - | IC50=0.01653 μM | SANGER |
HuP-T4 | - | Growth Inhibition Assay | - | IC50=0.06586 μM | SANGER |
HUTU-80 | - | Growth Inhibition Assay | - | IC50=0.02004 μM | SANGER |
IA-LM | - | Growth Inhibition Assay | - | IC50=0.01086 μM | SANGER |
IGR-1 | - | Growth Inhibition Assay | - | IC50=0.0205 μM | SANGER |
IGROV-1 | - | Growth Inhibition Assay | - | IC50=0.00814 μM | SANGER |
IM-9 | - | Growth Inhibition Assay | - | IC50=0.23476 μM | SANGER |
IMR-5 | - | Growth Inhibition Assay | - | IC50=0.0449 μM | SANGER |
IPC-298 | - | Growth Inhibition Assay | - | IC50=0.09644 μM | SANGER |
IST-MEL1 | - | Growth Inhibition Assay | - | IC50=0.00852 μM | SANGER |
IST-MES1 | - | Growth Inhibition Assay | - | IC50=0.411 μM | SANGER |
IST-SL1 | - | Growth Inhibition Assay | - | IC50=0.60435 μM | SANGER |
IST-SL2 | - | Growth Inhibition Assay | - | IC50=0.05743 μM | SANGER |
J82 | - | Growth Inhibition Assay | - | IC50=0.03007 μM | SANGER |
JAR | - | Growth Inhibition Assay | - | IC50=2.0792 μM | SANGER |
JEG-3 | - | Growth Inhibition Assay | - | IC50=0.09505 μM | SANGER |
JiyoyeP-2003 | - | Growth Inhibition Assay | - | IC50=0.03388 μM | SANGER |
J-RT3-T3-5 | - | Growth Inhibition Assay | - | IC50=0.08968 μM | SANGER |
JVM-2 | - | Growth Inhibition Assay | - | IC50=0.44401 μM | SANGER |
JVM-3 | - | Growth Inhibition Assay | - | IC50=0.54117 μM | SANGER |
K052 | - | Growth Inhibition Assay | - | IC50=0.17061 μM | SANGER |
K5 | - | Growth Inhibition Assay | - | IC50=0.01308 μM | SANGER |
K-562 | - | Growth Inhibition Assay | - | IC50=0.05387 μM | SANGER |
KALS-1 | - | Growth Inhibition Assay | - | IC50=0.01466 μM | SANGER |
KARPAS-299 | - | Growth Inhibition Assay | - | IC50=0.22994 μM | SANGER |
KARPAS-422 | - | Growth Inhibition Assay | - | IC50=0.14037 μM | SANGER |
KARPAS-45 | - | Growth Inhibition Assay | - | IC50=0.09345 μM | SANGER |
KE-37 | - | Growth Inhibition Assay | - | IC50=0.05683 μM | SANGER |
KG-1 | - | Growth Inhibition Assay | - | IC50=0.55984 μM | SANGER |
KGN | - | Growth Inhibition Assay | - | IC50=0.00703 μM | SANGER |
KINGS-1 | - | Growth Inhibition Assay | - | IC50=0.02433 μM | SANGER |
KLE | - | Growth Inhibition Assay | - | IC50=0.16169 μM | SANGER |
KM12 | - | Growth Inhibition Assay | - | IC50=0.01399 μM | SANGER |
KM-H2 | - | Growth Inhibition Assay | - | IC50=0.07241 μM | SANGER |
KMOE-2 | - | Growth Inhibition Assay | - | IC50=0.05749 μM | SANGER |
KMS-12-PE | - | Growth Inhibition Assay | - | IC50=0.12869 μM | SANGER |
KNS-42 | - | Growth Inhibition Assay | - | IC50=0.78831 μM | SANGER |
KNS-81-FD | - | Growth Inhibition Assay | - | IC50=0.06918 μM | SANGER |
KOSC-2 | - | Growth Inhibition Assay | - | IC50=0.0411 μM | SANGER |
KP-4 | - | Growth Inhibition Assay | - | IC50=0.03663 μM | SANGER |
KP-N-YN | - | Growth Inhibition Assay | - | IC50=0.31118 μM | SANGER |
KP-N-YS | - | Growth Inhibition Assay | - | IC50=0.08345 μM | SANGER |
KS-1 | - | Growth Inhibition Assay | - | IC50=0.00859 μM | SANGER |
KU-19-19 | - | Growth Inhibition Assay | - | IC50=0.10817 μM | SANGER |
KU812 | - | Growth Inhibition Assay | - | IC50=0.03684 μM | SANGER |
KURAMOCHI | - | Growth Inhibition Assay | - | IC50=0.06189 μM | SANGER |
KY821 | - | Growth Inhibition Assay | - | IC50=0.70229 μM | SANGER |
KYSE-140 | - | Growth Inhibition Assay | - | IC50=0.02024 μM | SANGER |
KYSE-150 | - | Growth Inhibition Assay | - | IC50=0.03608 μM | SANGER |
KYSE-180 | - | Growth Inhibition Assay | - | IC50=0.00586 μM | SANGER |
KYSE-270 | - | Growth Inhibition Assay | - | IC50=0.01059 μM | SANGER |
KYSE-410 | - | Growth Inhibition Assay | - | IC50=0.01586 μM | SANGER |
KYSE-450 | - | Growth Inhibition Assay | - | IC50=0.01349 μM | SANGER |
KYSE-510 | - | Growth Inhibition Assay | - | IC50=0.01442 μM | SANGER |
KYSE-520 | - | Growth Inhibition Assay | - | IC50=0.02613 μM | SANGER |
KYSE-70 | - | Growth Inhibition Assay | - | IC50=0.03812 μM | SANGER |
L-363 | - | Growth Inhibition Assay | - | IC50=0.06901 μM | SANGER |
L-428 | - | Growth Inhibition Assay | - | IC50=0.07704 μM | SANGER |
L-540 | - | Growth Inhibition Assay | - | IC50=0.30089 μM | SANGER |
LAMA-84 | - | Growth Inhibition Assay | - | IC50=0.04171 μM | SANGER |
LAN-6 | - | Growth Inhibition Assay | - | IC50=0.08498 μM | SANGER |
LB1047-RCC | - | Growth Inhibition Assay | - | IC50=0.05031 μM | SANGER |
LB2241-RCC | - | Growth Inhibition Assay | - | IC50=0.03642 μM | SANGER |
LB2518-MEL | - | Growth Inhibition Assay | - | IC50=0.40872 μM | SANGER |
LB373-MEL-D | - | Growth Inhibition Assay | - | IC50=0.29431 μM | SANGER |
LB647-SCLC | - | Growth Inhibition Assay | - | IC50=0.24014 μM | SANGER |
LB771-HNC | - | Growth Inhibition Assay | - | IC50=22.4813 μM | SANGER |
LB831-BLC | - | Growth Inhibition Assay | - | IC50=0.03219 μM | SANGER |
LB996-RCC | - | Growth Inhibition Assay | - | IC50=0.0271 μM | SANGER |
LC-1F | - | Growth Inhibition Assay | - | IC50=6.09291 μM | SANGER |
LC-2-ad | - | Growth Inhibition Assay | - | IC50=0.0137 μM | SANGER |
LC4-1 | - | Growth Inhibition Assay | - | IC50=0.11466 μM | SANGER |
LCLC-103H | - | Growth Inhibition Assay | - | IC50=0.0043 μM | SANGER |
LCLC-97TM1 | - | Growth Inhibition Assay | - | IC50=0.013 μM | SANGER |
LK-2 | - | Growth Inhibition Assay | - | IC50=0.10176 μM | SANGER |
LN-405 | - | Growth Inhibition Assay | - | IC50=0.7436 μM | SANGER |
LNCaP-Clone-FGC | - | Growth Inhibition Assay | - | IC50=0.08165 μM | SANGER |
LOUCY | - | Growth Inhibition Assay | - | IC50=0.00505 μM | SANGER |
LoVo | - | Growth Inhibition Assay | - | IC50=0.03933 μM | SANGER |
LOXIMVI | - | Growth Inhibition Assay | - | IC50=0.02323 μM | SANGER |
LP-1 | - | Growth Inhibition Assay | - | IC50=1.0693 μM | SANGER |
LS-1034 | - | Growth Inhibition Assay | - | IC50=0.04191 μM | SANGER |
LS-123 | - | Growth Inhibition Assay | - | IC50=0.02435 μM | SANGER |
LS-411N | - | Growth Inhibition Assay | - | IC50=0.03731 μM | SANGER |
LS-513 | - | Growth Inhibition Assay | - | IC50=0.07456 μM | SANGER |
LU-134-A | - | Growth Inhibition Assay | - | IC50=0.05715 μM | SANGER |
LU-139 | - | Growth Inhibition Assay | - | IC50=0.51457 μM | SANGER |
LU-165 | - | Growth Inhibition Assay | - | IC50=0.15413 μM | SANGER |
LU-65 | - | Growth Inhibition Assay | - | IC50=0.20211 μM | SANGER |
LU-99A | - | Growth Inhibition Assay | - | IC50=0.07287 μM | SANGER |
LXF-289 | - | Growth Inhibition Assay | - | IC50=0.02668 μM | SANGER |
M059J | - | Growth Inhibition Assay | - | IC50=0.02241 μM | SANGER |
M14 | - | Growth Inhibition Assay | - | IC50=0.21803 μM | SANGER |
MC116 | - | Growth Inhibition Assay | - | IC50=2.36397 μM | SANGER |
MC-CAR | - | Growth Inhibition Assay | - | IC50=0.04569 μM | SANGER |
MCF7 | - | Growth Inhibition Assay | - | IC50=0.00335 μM | SANGER |
MC-IXC | - | Growth Inhibition Assay | - | IC50=0.01736 μM | SANGER |
MDA-MB-134-VI | - | Growth Inhibition Assay | - | IC50=0.17367 μM | SANGER |
MDA-MB-157 | - | Growth Inhibition Assay | - | IC50=5.66443 μM | SANGER |
MDA-MB-175-VII | - | Growth Inhibition Assay | - | IC50=0.32348 μM | SANGER |
MDA-MB-231 | - | Growth Inhibition Assay | - | IC50=0.09082 μM | SANGER |
MDA-MB-361 | - | Growth Inhibition Assay | - | IC50=0.05872 μM | SANGER |
MDA-MB-415 | - | Growth Inhibition Assay | - | IC50=0.19748 μM | SANGER |
MDA-MB-453 | - | Growth Inhibition Assay | - | IC50=0.90304 μM | SANGER |
MDA-MB-468 | - | Growth Inhibition Assay | - | IC50=0.09985 μM | SANGER |
ME-180 | - | Growth Inhibition Assay | - | IC50=0.04782 μM | SANGER |
MEG-01 | - | Growth Inhibition Assay | - | IC50=0.17257 μM | SANGER |
MEL-HO | - | Growth Inhibition Assay | - | IC50=0.01643 μM | SANGER |
MEL-JUSO | - | Growth Inhibition Assay | - | IC50=0.01681 μM | SANGER |
MES-SA | - | Growth Inhibition Assay | - | IC50=0.00452 μM | SANGER |
Mewo | - | Growth Inhibition Assay | - | IC50=2.22265 μM | SANGER |
MFE-280 | - | Growth Inhibition Assay | - | IC50=0.35715 μM | SANGER |
MFE-296 | - | Growth Inhibition Assay | - | IC50=0.02322 μM | SANGER |
MFH-ino | - | Growth Inhibition Assay | - | IC50=0.01293 μM | SANGER |
MFM-223 | - | Growth Inhibition Assay | - | IC50=3.36097 μM | SANGER |
MG-63 | - | Growth Inhibition Assay | - | IC50=0.01874 μM | SANGER |
MHH-CALL-2 | - | Growth Inhibition Assay | - | IC50=0.4483 μM | SANGER |
MHH-ES-1 | - | Growth Inhibition Assay | - | IC50=0.01263 μM | SANGER |
MHH-NB-11 | - | Growth Inhibition Assay | - | IC50=0.2535 μM | SANGER |
MHH-PREB-1 | - | Growth Inhibition Assay | - | IC50=0.0931 μM | SANGER |
MIA-PaCa-2 | - | Growth Inhibition Assay | - | IC50=0.01509 μM | SANGER |
MKN1 | - | Growth Inhibition Assay | - | IC50=0.0493 μM | SANGER |
MKN28 | - | Growth Inhibition Assay | - | IC50=0.03012 μM | SANGER |
MKN45 | - | Growth Inhibition Assay | - | IC50=0.2064 μM | SANGER |
MKN7 | - | Growth Inhibition Assay | - | IC50=0.30639 μM | SANGER |
ML-2 | - | Growth Inhibition Assay | - | IC50=0.03671 μM | SANGER |
MLMA | - | Growth Inhibition Assay | - | IC50=0.04609 μM | SANGER |
MMAC-SF | - | Growth Inhibition Assay | - | IC50=0.04297 μM | SANGER |
MN-60 | - | Growth Inhibition Assay | - | IC50=0.24239 μM | SANGER |
MOLT-16 | - | Growth Inhibition Assay | - | IC50=0.01788 μM | SANGER |
MOLT-4 | - | Growth Inhibition Assay | - | IC50=0.04803 μM | SANGER |
MONO-MAC-6 | - | Growth Inhibition Assay | - | IC50=0.03893 μM | SANGER |
Mo-T | - | Growth Inhibition Assay | - | IC50=0.29331 μM | SANGER |
MPP-89 | - | Growth Inhibition Assay | - | IC50=0.09721 μM | SANGER |
MRK-nu-1 | - | Growth Inhibition Assay | - | IC50=0.023 μM | SANGER |
MS-1 | - | Growth Inhibition Assay | - | IC50=0.186 μM | SANGER |
MV-4-11 | - | Growth Inhibition Assay | - | IC50=0.000558 μM | SANGER |
MZ1-PC | - | Growth Inhibition Assay | - | IC50=0.02639 μM | SANGER |
MZ2-MEL | - | Growth Inhibition Assay | - | IC50=0.03177 μM | SANGER |
MZ7-mel | - | Growth Inhibition Assay | - | IC50=0.0433 μM | SANGER |
NALM-6 | - | Growth Inhibition Assay | - | IC50=0.000842 μM | SANGER |
NB1 | - | Growth Inhibition Assay | - | IC50=0.14426 μM | SANGER |
NB10 | - | Growth Inhibition Assay | - | IC50=0.23731 μM | SANGER |
NB12 | - | Growth Inhibition Assay | - | IC50=0.09518 μM | SANGER |
NB13 | - | Growth Inhibition Assay | - | IC50=0.04227 μM | SANGER |
NB5 | - | Growth Inhibition Assay | - | IC50=0.03613 μM | SANGER |
NB6 | - | Growth Inhibition Assay | - | IC50=0.67335 μM | SANGER |
NB69 | - | Growth Inhibition Assay | - | IC50=0.01102 μM | SANGER |
NCCIT | - | Growth Inhibition Assay | - | IC50=0.06604 μM | SANGER |
NCI-H1092 | - | Growth Inhibition Assay | - | IC50=0.14101 μM | SANGER |
NCI-H1155 | - | Growth Inhibition Assay | - | IC50=0.74868 μM | SANGER |
NCI-H1299 | - | Growth Inhibition Assay | - | IC50=0.01154 μM | SANGER |
NCI-H1304 | - | Growth Inhibition Assay | - | IC50=0.08271 μM | SANGER |
NCI-H1355 | - | Growth Inhibition Assay | - | IC50=0.02401 μM | SANGER |
NCI-H1395 | - | Growth Inhibition Assay | - | IC50=5.10633 μM | SANGER |
NCI-H1417 | - | Growth Inhibition Assay | - | IC50=0.0489 μM | SANGER |
NCI-H1436 | - | Growth Inhibition Assay | - | IC50=0.21826 μM | SANGER |
NCI-H1437 | - | Growth Inhibition Assay | - | IC50=0.06328 μM | SANGER |
NCI-H1522 | - | Growth Inhibition Assay | - | IC50=0.14787 μM | SANGER |
NCI-H1563 | - | Growth Inhibition Assay | - | IC50=19.7888 μM | SANGER |
NCI-H1573 | - | Growth Inhibition Assay | - | IC50=0.17678 μM | SANGER |
NCI-H1581 | - | Growth Inhibition Assay | - | IC50=1.35687 μM | SANGER |
NCI-H1618 | - | Growth Inhibition Assay | - | IC50=0.2751 μM | SANGER |
NCI-H1623 | - | Growth Inhibition Assay | - | IC50=5.83556 μM | SANGER |
NCI-H1648 | - | Growth Inhibition Assay | - | IC50=0.01499 μM | SANGER |
NCI-H1650 | - | Growth Inhibition Assay | - | IC50=0.01646 μM | SANGER |
NCI-H1651 | - | Growth Inhibition Assay | - | IC50=0.02431 μM | SANGER |
NCI-H1693 | - | Growth Inhibition Assay | - | IC50=0.03617 μM | SANGER |
NCI-H1694 | - | Growth Inhibition Assay | - | IC50=0.27733 μM | SANGER |
NCI-H1703 | - | Growth Inhibition Assay | - | IC50=0.06178 μM | SANGER |
NCI-H1734 | - | Growth Inhibition Assay | - | IC50=0.0323 μM | SANGER |
NCI-H1755 | - | Growth Inhibition Assay | - | IC50=0.13827 μM | SANGER |
NCI-H1770 | - | Growth Inhibition Assay | - | IC50=0.05879 μM | SANGER |
NCI-H1792 | - | Growth Inhibition Assay | - | IC50=0.04581 μM | SANGER |
NCI-H1793 | - | Growth Inhibition Assay | - | IC50=1.87593 μM | SANGER |
NCI-H1838 | - | Growth Inhibition Assay | - | IC50=8.51731 μM | SANGER |
NCI-H187 | - | Growth Inhibition Assay | - | IC50=9.51835 μM | SANGER |
NCI-H1882 | - | Growth Inhibition Assay | - | IC50=0.41784 μM | SANGER |
NCI-H1963 | - | Growth Inhibition Assay | - | IC50=0.05176 μM | SANGER |
NCI-H1993 | - | Growth Inhibition Assay | - | IC50=1.04657 μM | SANGER |
NCI-H2009 | - | Growth Inhibition Assay | - | IC50=0.0276 μM | SANGER |
NCI-H2030 | - | Growth Inhibition Assay | - | IC50=0.01697 μM | SANGER |
NCI-H2052 | - | Growth Inhibition Assay | - | IC50=0.10407 μM | SANGER |
NCI-H2081 | - | Growth Inhibition Assay | - | IC50=0.15218 μM | SANGER |
NCI-H2087 | - | Growth Inhibition Assay | - | IC50=0.03289 μM | SANGER |
NCI-H209 | - | Growth Inhibition Assay | - | IC50=4.78572 μM | SANGER |
NCI-H2122 | - | Growth Inhibition Assay | - | IC50=0.01384 μM | SANGER |
NCI-H2126 | - | Growth Inhibition Assay | - | IC50=0.63152 μM | SANGER |
NCI-H2141 | - | Growth Inhibition Assay | - | IC50=0.23841 μM | SANGER |
NCI-H2170 | - | Growth Inhibition Assay | - | IC50=0.16304 μM | SANGER |
NCI-H2171 | - | Growth Inhibition Assay | - | IC50=0.18649 μM | SANGER |
NCI-H2196 | - | Growth Inhibition Assay | - | IC50=0.21747 μM | SANGER |
NCI-H2227 | - | Growth Inhibition Assay | - | IC50=1.04981 μM | SANGER |
NCI-H2228 | - | Growth Inhibition Assay | - | IC50=0.01064 μM | SANGER |
NCI-H226 | - | Growth Inhibition Assay | - | IC50=0.05988 μM | SANGER |
NCI-H23 | - | Growth Inhibition Assay | - | IC50=0.24059 μM | SANGER |
NCI-H2342 | - | Growth Inhibition Assay | - | IC50=0.01758 μM | SANGER |
NCI-H2347 | - | Growth Inhibition Assay | - | IC50=0.08028 μM | SANGER |
NCI-H2405 | - | Growth Inhibition Assay | - | IC50=0.02887 μM | SANGER |
NCI-H2452 | - | Growth Inhibition Assay | - | IC50=14.73 μM | SANGER |
NCI-H28 | - | Growth Inhibition Assay | - | IC50=0.29837 μM | SANGER |
NCI-H292 | - | Growth Inhibition Assay | - | IC50=0.01709 μM | SANGER |
NCI-H322M | - | Growth Inhibition Assay | - | IC50=9.16281 μM | SANGER |
NCI-H345 | - | Growth Inhibition Assay | - | IC50=21.8779 μM | SANGER |
NCI-H358 | - | Growth Inhibition Assay | - | IC50=0.04212 μM | SANGER |
NCI-H441 | - | Growth Inhibition Assay | - | IC50=0.10899 μM | SANGER |
NCI-H446 | - | Growth Inhibition Assay | - | IC50=0.29921 μM | SANGER |
NCI-H460 | - | Growth Inhibition Assay | - | IC50=0.01336 μM | SANGER |
NCI-H510A | - | Growth Inhibition Assay | - | IC50=0.29304 μM | SANGER |
NCI-H520 | - | Growth Inhibition Assay | - | IC50=0.02664 μM | SANGER |
NCI-H522 | - | Growth Inhibition Assay | - | IC50=0.01939 μM | SANGER |
NCI-H524 | - | Growth Inhibition Assay | - | IC50=24.3812 μM | SANGER |
NCI-H526 | - | Growth Inhibition Assay | - | IC50=0.18696 μM | SANGER |
NCI-H596 | - | Growth Inhibition Assay | - | IC50=0.1738 μM | SANGER |
NCI-H64 | - | Growth Inhibition Assay | - | IC50=1.1542 μM | SANGER |
NCI-H650 | - | Growth Inhibition Assay | - | IC50=0.02117 μM | SANGER |
NCI-H661 | - | Growth Inhibition Assay | - | IC50=0.11195 μM | SANGER |
NCI-H69 | - | Growth Inhibition Assay | - | IC50=0.27201 μM | SANGER |
NCI-H716 | - | Growth Inhibition Assay | - | IC50=0.44848 μM | SANGER |
NCI-H719 | - | Growth Inhibition Assay | - | IC50=0.35124 μM | SANGER |
NCI-H720 | - | Growth Inhibition Assay | - | IC50=2.26585 μM | SANGER |
NCI-H727 | - | Growth Inhibition Assay | - | IC50=0.0103 μM | SANGER |
NCI-H747 | - | Growth Inhibition Assay | - | IC50=0.0457 μM | SANGER |
NCI-H748 | - | Growth Inhibition Assay | - | IC50=1.35738 μM | SANGER |
NCI-H810 | - | Growth Inhibition Assay | - | IC50=0.01724 μM | SANGER |
NCI-H82 | - | Growth Inhibition Assay | - | IC50=23.5526 μM | SANGER |
NCI-H838 | - | Growth Inhibition Assay | - | IC50=0.23714 μM | SANGER |
NCI-H889 | - | Growth Inhibition Assay | - | IC50=2.56706 μM | SANGER |
NCI-N87 | - | Growth Inhibition Assay | - | IC50=0.07799 μM | SANGER |
NCI-SNU-1 | - | Growth Inhibition Assay | - | IC50=0.07888 μM | SANGER |
NCI-SNU-16 | - | Growth Inhibition Assay | - | IC50=48.3142 μM | SANGER |
NCI-SNU-5 | - | Growth Inhibition Assay | - | IC50=0.27613 μM | SANGER |
NEC8 | - | Growth Inhibition Assay | - | IC50=0.45145 μM | SANGER |
NH-12 | - | Growth Inhibition Assay | - | IC50=0.0444 μM | SANGER |
NKM-1 | - | Growth Inhibition Assay | - | IC50=0.00547 μM | SANGER |
NMC-G1 | - | Growth Inhibition Assay | - | IC50=0.0228 μM | SANGER |
no-10 | - | Growth Inhibition Assay | - | IC50=0.03016 μM | SANGER |
no-11 | - | Growth Inhibition Assay | - | IC50=0.03048 μM | SANGER |
NOMO-1 | - | Growth Inhibition Assay | - | IC50=0.07172 μM | SANGER |
NOS-1 | - | Growth Inhibition Assay | - | IC50=0.01593 μM | SANGER |
NTERA-S-cl-D1 | - | Growth Inhibition Assay | - | IC50=0.01339 μM | SANGER |
NUGC-3 | - | Growth Inhibition Assay | - | IC50=0.04827 μM | SANGER |
NY | - | Growth Inhibition Assay | - | IC50=0.0174 μM | SANGER |
OAW-28 | - | Growth Inhibition Assay | - | IC50=0.26677 μM | SANGER |
OAW-42 | - | Growth Inhibition Assay | - | IC50=0.03747 μM | SANGER |
OCI-AML2 | - | Growth Inhibition Assay | - | IC50=0.01281 μM | SANGER |
OCUB-M | - | Growth Inhibition Assay | - | IC50=0.03961 μM | SANGER |
OE19 | - | Growth Inhibition Assay | - | IC50=0.0195 μM | SANGER |
OE33 | - | Growth Inhibition Assay | - | IC50=0.04241 μM | SANGER |
OMC-1 | - | Growth Inhibition Assay | - | IC50=0.01751 μM | SANGER |
ONS-76 | - | Growth Inhibition Assay | - | IC50=0.02954 μM | SANGER |
OPM-2 | - | Growth Inhibition Assay | - | IC50=0.31064 μM | SANGER |
OS-RC-2 | - | Growth Inhibition Assay | - | IC50=0.03396 μM | SANGER |
OVCAR-3 | - | Growth Inhibition Assay | - | IC50=0.14078 μM | SANGER |
OVCAR-4 | - | Growth Inhibition Assay | - | IC50=0.03858 μM | SANGER |
OVCAR-5 | - | Growth Inhibition Assay | - | IC50=0.01812 μM | SANGER |
OVCAR-8 | - | Growth Inhibition Assay | - | IC50=0.03281 μM | SANGER |
P12-ICHIKAWA | - | Growth Inhibition Assay | - | IC50=2.82046 μM | SANGER |
P30-OHK | - | Growth Inhibition Assay | - | IC50=0.26905 μM | SANGER |
P31-FUJ | - | Growth Inhibition Assay | - | IC50=1.10766 μM | SANGER |
PA-1 | - | Growth Inhibition Assay | - | IC50=0.02755 μM | SANGER |
PANC-03-27 | - | Growth Inhibition Assay | - | IC50=0.01162 μM | SANGER |
PANC-08-13 | - | Growth Inhibition Assay | - | IC50=0.07716 μM | SANGER |
PANC-10-05 | - | Growth Inhibition Assay | - | IC50=0.01755 μM | SANGER |
PC-14 | - | Growth Inhibition Assay | - | IC50=0.01934 μM | SANGER |
PC-3 | - | Growth Inhibition Assay | - | IC50=0.13177 μM | SANGER |
PF-382 | - | Growth Inhibition Assay | - | IC50=0.04826 μM | SANGER |
PFSK-1 | - | Growth Inhibition Assay | - | IC50=0.10267 μM | SANGER |
PLC-PRF-5 | - | Growth Inhibition Assay | - | IC50=0.88475 μM | SANGER |
PSN1 | - | Growth Inhibition Assay | - | IC50=0.00318 μM | SANGER |
QIMR-WIL | - | Growth Inhibition Assay | - | IC50=0.01269 μM | SANGER |
Raji | - | Growth Inhibition Assay | - | IC50=0.26603 μM | SANGER |
Ramos-2G6-4C10 | - | Growth Inhibition Assay | - | IC50=0.07648 μM | SANGER |
RCC10RGB | - | Growth Inhibition Assay | - | IC50=0.71918 μM | SANGER |
RCM-1 | - | Growth Inhibition Assay | - | IC50=0.1568 μM | SANGER |
RD | - | Growth Inhibition Assay | - | IC50=0.02658 μM | SANGER |
REH | - | Growth Inhibition Assay | - | IC50=0.02059 μM | SANGER |
RERF-LC-MS | - | Growth Inhibition Assay | - | IC50=0.1343 μM | SANGER |
RH-1 | - | Growth Inhibition Assay | - | IC50=0.0623 μM | SANGER |
RKO | - | Growth Inhibition Assay | - | IC50=0.00826 μM | SANGER |
RL | - | Growth Inhibition Assay | - | IC50=0.28174 μM | SANGER |
RMG-I | - | Growth Inhibition Assay | - | IC50=0.36691 μM | SANGER |
RO82-W-1 | - | Growth Inhibition Assay | - | IC50=1.33339 μM | SANGER |
RPMI-2650 | - | Growth Inhibition Assay | - | IC50=0.01432 μM | SANGER |
RPMI-6666 | - | Growth Inhibition Assay | - | IC50=0.00852 μM | SANGER |
RPMI-7951 | - | Growth Inhibition Assay | - | IC50=0.00631 μM | SANGER |
RPMI-8226 | - | Growth Inhibition Assay | - | IC50=0.11719 μM | SANGER |
RPMI-8402 | - | Growth Inhibition Assay | - | IC50=0.52207 μM | SANGER |
RPMI-8866 | - | Growth Inhibition Assay | - | IC50=5.84792 μM | SANGER |
RS4-11 | - | Growth Inhibition Assay | - | IC50=0.03383 μM | SANGER |
RT-112 | - | Growth Inhibition Assay | - | IC50=0.00535 μM | SANGER |
RT4 | - | Growth Inhibition Assay | - | IC50=23.3282 μM | SANGER |
RVH-421 | - | Growth Inhibition Assay | - | IC50=0.01957 μM | SANGER |
RXF393 | - | Growth Inhibition Assay | - | IC50=0.0086 μM | SANGER |
S-117 | - | Growth Inhibition Assay | - | IC50=0.12674 μM | SANGER |
Saos-2 | - | Growth Inhibition Assay | - | IC50=0.07597 μM | SANGER |
SAS | - | Growth Inhibition Assay | - | IC50=0.09215 μM | SANGER |
SBC-1 | - | Growth Inhibition Assay | - | IC50=9.93656 μM | SANGER |
SBC-5 | - | Growth Inhibition Assay | - | IC50=0.09193 μM | SANGER |
SCC-15 | - | Growth Inhibition Assay | - | IC50=0.02801 μM | SANGER |
SCC-25 | - | Growth Inhibition Assay | - | IC50=0.13588 μM | SANGER |
SCC-3 | - | Growth Inhibition Assay | - | IC50=10.5679 μM | SANGER |
SCC-4 | - | Growth Inhibition Assay | - | IC50=0.02809 μM | SANGER |
SCC-9 | - | Growth Inhibition Assay | - | IC50=0.0587 μM | SANGER |
SCLC-21H | - | Growth Inhibition Assay | - | IC50=0.76903 μM | SANGER |
SF126 | - | Growth Inhibition Assay | - | IC50=0.0501 μM | SANGER |
SF268 | - | Growth Inhibition Assay | - | IC50=0.03401 μM | SANGER |
SF295 | - | Growth Inhibition Assay | - | IC50=0.01721 μM | SANGER |
SF539 | - | Growth Inhibition Assay | - | IC50=0.79925 μM | SANGER |
SH-4 | - | Growth Inhibition Assay | - | IC50=0.04141 μM | SANGER |
SHP-77 | - | Growth Inhibition Assay | - | IC50=0.14472 μM | SANGER |
SIG-M5 | - | Growth Inhibition Assay | - | IC50=0.00489 μM | SANGER |
SiHa | - | Growth Inhibition Assay | - | IC50=4.95203 μM | SANGER |
SIMA | - | Growth Inhibition Assay | - | IC50=0.71719 μM | SANGER |
SJRH30 | - | Growth Inhibition Assay | - | IC50=0.09444 μM | SANGER |
SJSA-1 | - | Growth Inhibition Assay | - | IC50=0.02037 μM | SANGER |
SK-CO-1 | - | Growth Inhibition Assay | - | IC50=0.07992 μM | SANGER |
SKG-IIIa | - | Growth Inhibition Assay | - | IC50=0.17807 μM | SANGER |
SK-HEP-1 | - | Growth Inhibition Assay | - | IC50=0.00336 μM | SANGER |
SK-LMS-1 | - | Growth Inhibition Assay | - | IC50=0.00458 μM | SANGER |
SK-LU-1 | - | Growth Inhibition Assay | - | IC50=0.01846 μM | SANGER |
SK-MEL-1 | - | Growth Inhibition Assay | - | IC50=1.20595 μM | SANGER |
SK-MEL-2 | - | Growth Inhibition Assay | - | IC50=0.1246 μM | SANGER |
SK-MEL-24 | - | Growth Inhibition Assay | - | IC50=0.04283 μM | SANGER |
SK-MEL-28 | - | Growth Inhibition Assay | - | IC50=2.18098 μM | SANGER |
SK-MEL-3 | - | Growth Inhibition Assay | - | IC50=0.04802 μM | SANGER |
SK-MEL-30 | - | Growth Inhibition Assay | - | IC50=0.04362 μM | SANGER |
SK-MES-1 | - | Growth Inhibition Assay | - | IC50=0.00945 μM | SANGER |
SK-MM-2 | - | Growth Inhibition Assay | - | IC50=0.11145 μM | SANGER |
SK-N-AS | - | Growth Inhibition Assay | - | IC50=0.2722 μM | SANGER |
SK-N-DZ | - | Growth Inhibition Assay | - | IC50=0.17883 μM | SANGER |
SK-NEP-1 | - | Growth Inhibition Assay | - | IC50=0.15899 μM | SANGER |
SK-N-FI | - | Growth Inhibition Assay | - | IC50=0.37637 μM | SANGER |
SK-OV-3 | - | Growth Inhibition Assay | - | IC50=0.0063 μM | SANGER |
SK-PN-DW | - | Growth Inhibition Assay | - | IC50=0.05588 μM | SANGER |
SK-UT-1 | - | Growth Inhibition Assay | - | IC50=0.03221 μM | SANGER |
SN12C | - | Growth Inhibition Assay | - | IC50=0.24694 μM | SANGER |
SNB75 | - | Growth Inhibition Assay | - | IC50=0.02466 μM | SANGER |
SNG-M | - | Growth Inhibition Assay | - | IC50=0.00856 μM | SANGER |
SNU-387 | - | Growth Inhibition Assay | - | IC50=0.09218 μM | SANGER |
SNU-423 | - | Growth Inhibition Assay | - | IC50=0.01053 μM | SANGER |
SNU-449 | - | Growth Inhibition Assay | - | IC50=0.02026 μM | SANGER |
SNU-475 | - | Growth Inhibition Assay | - | IC50=0.79202 μM | SANGER |
SNU-C1 | - | Growth Inhibition Assay | - | IC50=24.9105 μM | SANGER |
SNU-C2B | - | Growth Inhibition Assay | - | IC50=0.01272 μM | SANGER |
SR | - | Growth Inhibition Assay | - | IC50=0.02785 μM | SANGER |
ST486 | - | Growth Inhibition Assay | - | IC50=0.05525 μM | SANGER |
SU-DHL-1 | - | Growth Inhibition Assay | - | IC50=0.0692 μM | SANGER |
SUP-T1 | - | Growth Inhibition Assay | - | IC50=0.0676 μM | SANGER |
SW1088 | - | Growth Inhibition Assay | - | IC50=0.53869 μM | SANGER |
SW13 | - | Growth Inhibition Assay | - | IC50=0.0459 μM | SANGER |
SW1417 | - | Growth Inhibition Assay | - | IC50=0.81339 μM | SANGER |
SW1463 | - | Growth Inhibition Assay | - | IC50=1.18349 μM | SANGER |
SW1573 | - | Growth Inhibition Assay | - | IC50=0.05802 μM | SANGER |
SW1710 | - | Growth Inhibition Assay | - | IC50=0.00186 μM | SANGER |
SW1783 | - | Growth Inhibition Assay | - | IC50=0.00591 μM | SANGER |
SW1990 | - | Growth Inhibition Assay | - | IC50=0.02724 μM | SANGER |
SW48 | - | Growth Inhibition Assay | - | IC50=0.04031 μM | SANGER |
SW620 | - | Growth Inhibition Assay | - | IC50=0.01915 μM | SANGER |
SW626 | - | Growth Inhibition Assay | - | IC50=0.0212 μM | SANGER |
SW684 | - | Growth Inhibition Assay | - | IC50=0.28383 μM | SANGER |
SW756 | - | Growth Inhibition Assay | - | IC50=0.04157 μM | SANGER |
SW780 | - | Growth Inhibition Assay | - | IC50=21.1318 μM | SANGER |
SW837 | - | Growth Inhibition Assay | - | IC50=0.03014 μM | SANGER |
SW872 | - | Growth Inhibition Assay | - | IC50=0.03217 μM | SANGER |
SW948 | - | Growth Inhibition Assay | - | IC50=10.7511 μM | SANGER |
SW954 | - | Growth Inhibition Assay | - | IC50=0.01071 μM | SANGER |
SW962 | - | Growth Inhibition Assay | - | IC50=0.02852 μM | SANGER |
SW982 | - | Growth Inhibition Assay | - | IC50=0.01293 μM | SANGER |
T-24 | - | Growth Inhibition Assay | - | IC50=0.05384 μM | SANGER |
T47D | - | Growth Inhibition Assay | - | IC50=0.44528 μM | SANGER |
T84 | - | Growth Inhibition Assay | - | IC50=0.01331 μM | SANGER |
T98G | - | Growth Inhibition Assay | - | IC50=0.07421 μM | SANGER |
TALL-1 | - | Growth Inhibition Assay | - | IC50=1.25165 μM | SANGER |
TCCSUP | - | Growth Inhibition Assay | - | IC50=6.60349 μM | SANGER |
TE-1 | - | Growth Inhibition Assay | - | IC50=0.01581 μM | SANGER |
TE-10 | - | Growth Inhibition Assay | - | IC50=0.01977 μM | SANGER |
TE-11 | - | Growth Inhibition Assay | - | IC50=0.19975 μM | SANGER |
TE-12 | - | Growth Inhibition Assay | - | IC50=0.01775 μM | SANGER |
TE-15 | - | Growth Inhibition Assay | - | IC50=0.01336 μM | SANGER |
TE-441-T | - | Growth Inhibition Assay | - | IC50=0.0493 μM | SANGER |
TE-5 | - | Growth Inhibition Assay | - | IC50=4.56147 μM | SANGER |
TE-6 | - | Growth Inhibition Assay | - | IC50=0.24612 μM | SANGER |
TE-8 | - | Growth Inhibition Assay | - | IC50=0.00237 μM | SANGER |
TE-9 | - | Growth Inhibition Assay | - | IC50=0.04237 μM | SANGER |
TGBC1TKB | - | Growth Inhibition Assay | - | IC50=0.20997 μM | SANGER |
TGBC24TKB | - | Growth Inhibition Assay | - | IC50=13.529 μM | SANGER |
TGW | - | Growth Inhibition Assay | - | IC50=0.16471 μM | SANGER |
THP-1 | - | Growth Inhibition Assay | - | IC50=0.15333 μM | SANGER |
TK10 | - | Growth Inhibition Assay | - | IC50=0.01382 μM | SANGER |
TT | - | Growth Inhibition Assay | - | IC50=8.33009 μM | SANGER |
TUR | - | Growth Inhibition Assay | - | IC50=0.07733 μM | SANGER |
TYK-nu | - | Growth Inhibition Assay | - | IC50=0.67952 μM | SANGER |
U031 | - | Growth Inhibition Assay | - | IC50=0.04771 μM | SANGER |
U-118-MG | - | Growth Inhibition Assay | - | IC50=0.02576 μM | SANGER |
U251 | - | Growth Inhibition Assay | - | IC50=0.04763 μM | SANGER |
U-266 | - | Growth Inhibition Assay | - | IC50=0.1448 μM | SANGER |
U-2-OS | - | Growth Inhibition Assay | - | IC50=0.03935 μM | SANGER |
U-698-M | - | Growth Inhibition Assay | - | IC50=0.07382 μM | SANGER |
U-87-MG | - | Growth Inhibition Assay | - | IC50=0.0329 μM | SANGER |
UACC-257 | - | Growth Inhibition Assay | - | IC50=0.07505 μM | SANGER |
UACC-62 | - | Growth Inhibition Assay | - | IC50=0.1212 μM | SANGER |
UACC-812 | - | Growth Inhibition Assay | - | IC50=0.46776 μM | SANGER |
UACC-893 | - | Growth Inhibition Assay | - | IC50=0.05896 μM | SANGER |
UMC-11 | - | Growth Inhibition Assay | - | IC50=2.78715 μM | SANGER |
UM-UC-3 | - | Growth Inhibition Assay | - | IC50=0.0495 μM | SANGER |
VA-ES-BJ | - | Growth Inhibition Assay | - | IC50=0.04292 μM | SANGER |
VM-CUB-1 | - | Growth Inhibition Assay | - | IC50=0.05311 μM | SANGER |
VMRC-RCZ | - | Growth Inhibition Assay | - | IC50=0.01651 μM | SANGER |
WM-115 | - | Growth Inhibition Assay | - | IC50=0.65092 μM | SANGER |
WSU-NHL | - | Growth Inhibition Assay | - | IC50=0.07329 μM | SANGER |
YAPC | - | Growth Inhibition Assay | - | IC50=0.55211 μM | SANGER |
YKG-1 | - | Growth Inhibition Assay | - | IC50=0.0116 μM | SANGER |
YT | - | Growth Inhibition Assay | - | IC50=0.01179 μM | SANGER |
靶点 | Description | IC50 |
---|---|---|
HSP90α | IC50:13nM | |
HSP90β | IC50:21nM |
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