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CAS No.: 1243244-14-5
Synonyms: WNT974;NVP-LGK974;PORCN Inhibitor IV
LGK974 is a potent and specific small molecule inhibitor of PORCN (IC50 = 0.4 nM).
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
靶点 | PORCN IC50:0.4nM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01351103 | Pancreatic Cancer ... more >> BRAF Mutant Colorectal Cancer Melanoma Triple Negative Breast Cancer Head and Neck Squamous Cell Cancer Cervical Squamous Cell Cancer Esophageal Squamous Cell Cancer Lung Squamous Cell Cancer Collapse << | Phase 1 | Recruiting | August 20, 2020 | United States, California ... more >> Novartis Investigative Site Recruiting Los Angeles, California, United States, 90024 United States, Maryland Novartis Investigative Site Recruiting Baltimore, Maryland, United States, 21287-0013 Contact: Ashley Elza O'Connor +1 410 502 2377 aoconnor@jhmi.edu Principal Investigator: Roisin Connolly United States, Massachusetts Dana Farber Cancer Institute SC Withdrawn Boston, Massachusetts, United States, 02115 Dana Farber Cancer Institute SC-7 Recruiting Boston, Massachusetts, United States, 02215 Contact: Marios Giannakis, M.D., Ph.D. 617-632-6805 Marios_Giannakis@dfci.harvard.edu Principal Investigator: Marios Giannakis, M.D., Ph.D. United States, Michigan University of Michigan Comprehensive Cancer Center Onc Dept. Not yet recruiting Ann Arbor, Michigan, United States, 48109-0944 Contact: Cancer AnswerLine 800-865-1125 Principal Investigator: David Smith Karmanos Cancer Institute Wayne St Recruiting Detroit, Michigan, United States, 48201 Contact: DeQuindalyn Moore 313-576-9371 moored@karmanos.org Principal Investigator: Ulka A. Vaishampayan United States, Texas University of Texas/MD Anderson Cancer Center MD Anderson 2 Recruiting Houston, Texas, United States, 77030-4009 Contact: Stepanek M. Vanda 713-792-2921 vstepane@mdanderson.org Principal Investigator: Filip P. Janku Netherlands Novartis Investigative Site Recruiting Rotterdam, Netherlands, 3075 EA Novartis Investigative Site Recruiting Utrecht, Netherlands, 3584CX Spain Novartis Investigative Site Recruiting Barcelona, Catalunya, Spain, 08035 Novartis Investigative Site Recruiting Barcelona, Catalunya, Spain, 08036 Novartis Investigative Site Recruiting Madrid, Spain, 28007 Novartis Investigative Site Recruiting Madrid, Spain, 28050 Collapse << |
实验方案
技术信息
CAS号 | 1243244-14-5 | 储存条件 |
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分子式 | C23H20N6O | 运输 | 蓝冰 | |||||||||||||
分子量 | 396.44 | 别名 | WNT974;NVP-LGK974;PORCN Inhibitor IV | |||||||||||||
溶解度 |
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动物实验配方 |
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