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CAS No.: 223132-37-4
Synonyms: Efatutazone;CS-7017;RS5444
Inolitazone is a high-affinity PPARγ agonist, which activates PPARγ with an EC50 about 1/50 that of rosiglitazone and has no effect on RIE cells that do not express PPARγ.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00408434 | Neoplasm | Phase 1 | Completed | - | United States, District of Col... more >>umbia Washington, District of Columbia, United States United States, Massachusetts Boston, Massachusetts, United States Collapse << |
NCT00806286 | Metastatic Non-small Cell Lung... more >> Cancer Collapse << | Phase 2 | Completed | - | - |
NCT00967616 | Colorectal Cancer ... more >> Neoplasms, Colorectal Collapse << | Phase 2 | Completed | - | United States, California ... more >> Beverly Hills Cancer Center Beverly Hills, California, United States, 90211 St. Jude Heritage Medical Group Fullerton, California, United States, 92835 United States, District of Columbia John Marshall Washington, District of Columbia, United States, 20007 United States, Georgia Georgia Cancer Specialists Atlanta, Georgia, United States, 30341 United States, Maryland Victor Priego Bethesda, Maryland, United States, 20817 United States, Ohio Gabrail Cancer Center Canton, Ohio, United States, 44718 Argentina Instituto FIDES Oncologia y Especialidades Medicas Buenos Aires, Argentina, B1900BAJ CAIPO Centro para la Atencion Integral del Paciente Oncologico Tucuman, Argentina, T4000GTB Brazil Hospital Sao Lucas da Pontificia Universidade Catolica do Rio Grande do Sul - PUC-RS Porto Alegre, Brazil, 90610-000 Instituto Nacional de Cancer INCA Rio de Janeiro, Brazil, 20231-050 ICAVC Sao Paulo, Brazil, 01209-000 Chile Fundacion Arturo Lopez Perez Santiago, Chile, 8320000 Instituto Nacional del Cancer Santiago, Chile, 8380455 Instituto Oncologico Clinica Renaca Vina del Mar, Chile, 2540364 Peru Hospital Nacional Alberto Sabogai Sologuren Callao, Peru Hospital Nacional Dos de Mayo Lima, Peru, 01 Oncosalud SAC Lima, Peru, 41 Hospital Nacional Dos de Mayo Lima, Peru Collapse << |
实验方案
技术信息
CAS号 | 223132-37-4 | 储存条件 |
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分子式 | C27H26N4O4S | 运输 | 蓝冰 | |
分子量 | 502.58 | 别名 | Efatutazone;CS-7017;RS5444;Efatutazone Free Base |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00408434 | Neoplasm | Phase 1 | Completed | - | United States, District of Col... more >>umbia Washington, District of Columbia, United States United States, Massachusetts Boston, Massachusetts, United States Collapse << |
NCT00806286 | Metastatic Non-small Cell Lung... more >> Cancer Collapse << | Phase 2 | Completed | - | - |
NCT00967616 | Colorectal Cancer ... more >> Neoplasms, Colorectal Collapse << | Phase 2 | Completed | - | United States, California ... more >> Beverly Hills Cancer Center Beverly Hills, California, United States, 90211 St. Jude Heritage Medical Group Fullerton, California, United States, 92835 United States, District of Columbia John Marshall Washington, District of Columbia, United States, 20007 United States, Georgia Georgia Cancer Specialists Atlanta, Georgia, United States, 30341 United States, Maryland Victor Priego Bethesda, Maryland, United States, 20817 United States, Ohio Gabrail Cancer Center Canton, Ohio, United States, 44718 Argentina Instituto FIDES Oncologia y Especialidades Medicas Buenos Aires, Argentina, B1900BAJ CAIPO Centro para la Atencion Integral del Paciente Oncologico Tucuman, Argentina, T4000GTB Brazil Hospital Sao Lucas da Pontificia Universidade Catolica do Rio Grande do Sul - PUC-RS Porto Alegre, Brazil, 90610-000 Instituto Nacional de Cancer INCA Rio de Janeiro, Brazil, 20231-050 ICAVC Sao Paulo, Brazil, 01209-000 Chile Fundacion Arturo Lopez Perez Santiago, Chile, 8320000 Instituto Nacional del Cancer Santiago, Chile, 8380455 Instituto Oncologico Clinica Renaca Vina del Mar, Chile, 2540364 Peru Hospital Nacional Alberto Sabogai Sologuren Callao, Peru Hospital Nacional Dos de Mayo Lima, Peru, 01 Oncosalud SAC Lima, Peru, 41 Hospital Nacional Dos de Mayo Lima, Peru Collapse << |
NCT02249949 | Liposarcoma | Phase 2 | Active, not recruiting | - | - |
NCT01101334 | Advanced Non-small Cell Lung C... more >>ancer Collapse << | Phase 2 | Completed | - | United States, Colorado ... more >> DHHA Denver, Colorado, United States, 80204 United States, Ohio Gabrail Cancer Center Canton, Ohio, United States, 44718 United States, Washington Providence Regional Medical Center Everett Everett, Washington, United States, 98201 Germany Zentrum fur Pneumologie und Thoraxchirurgie Gauting, Germany, D-82131 India King George Hospital Visakhapatnam, Andhra Pradesh, India, 530002 Vedanta Institute of Medical Sciences Ahmedabad, Gujarat, India, 380009 Kodlikeri Memorial Hospital Aurangabad, Maharashtra, India, 431001 Tata Memorial Hospital Mumbai, Maharashtra, India, 400012 Noble Hospital Pune, Maharastra, India, 411 013 Apollo Speciality Hospital Chennai, Tamil Nadu, India, 600 035 Meenakshi Mission Hospital Madurai, Tamil Nadu, India, 625107 Orchid Nursing Home Kolkata, West Bengal, India, 700 054 Korea, Republic of St. Vincent's Hospital Gyeonggi-Do, Korea, Republic of, 442-723 Hwasun Hospital Jeonnam, Korea, Republic of, 519-763 Severance Hospital Seoul, Korea, Republic of, 120-752 Samsung Medical Center Seoul, Korea, Republic of, 135-710 Asan Medical Center Seoul, Korea, Republic of, 138-736 Collapse << |
NCT01199055 | Carcinoma, Non-Small-Cell Lung | Phase 1 | Completed | - | Korea, Republic of ... more >> Samsung Medical Center Seoul, Gangnam-gu, Korea, Republic of, 135-710 Collapse << |
NCT00881569 | Cancer | Phase 1 | Completed | - | United States, District of Col... more >>umbia Washington, District of Columbia, United States Collapse << |
NCT01504490 | Solid Tumors ... more >>Lymphoma Multiple Myeloma Collapse << | Phase 1 | Terminated(Drug no longer avai... more >>lable) Collapse << | - | United States, District of Col... more >>umbia Georgetown Lombardi Comprehensive Cancer Center Washington, District of Columbia, United States, 20007 Collapse << |
NCT02152137 | Anaplastic Thyroid Cancer ... more >> Recurrent Thyroid Cancer Collapse << | Phase 2 | Active, not recruiting | - | - |
NCT01199068 | Carcinoma, Non-Small-Cell Lung | Phase 1 | Completed | - | Korea, Republic of ... more >> Asan Medical Center Seoul, Songpa-Gu, Korea, Republic of, 138-736 Collapse << |
NCT00603941 | Anaplastic Thyroid Cancer | Phase 1 Phase 2 | Completed | - | United States, Colorado ... more >> Univ of Colorado Cancer Center Aurora, Colorado, United States, 80045 United States, Florida Mayo Clinic Jacksonville, Florida, United States, 32224 United States, Massachusetts Massachusetts General Hospital Boston, Massachusetts, United States, 02115 United States, Minnesota Mayo Clinic Rochester, Minnesota, United States, 55905 United States, Missouri Washington University, Siteman Cancer Center St. Louis, Missouri, United States, 63110 United States, Ohio Ohio State Univ Columbus, Ohio, United States, 43210 United States, Oregon Oregon Health Science Univ Portland, Oregon, United States, 97239 United States, Pennsylvania University of Pennsylvania Maloney Hospital Philadelphia, Pennsylvania, United States, 19104 United States, Tennessee Vanderbilt Ingram Cancer Center Nashville, Tennessee, United States, 37232 United States, Virginia Eastern Virginia Medical School Norfolk, Virginia, United States, 23507 Collapse << |
NCT00986440 | Colorectal Cancer | Phase 2 | Completed | - | - |
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