CAS No.: 1456858-58-4
HG-9-91-01 Catalog No. CSN17882
Synonyms: SIK inhibitor 1
HG-9-91-01 is a potent and highly selective salt-inducible kinase (SIKs) inhibitor with IC50s of 0.92 nM, 6.6 nM and 9.6 nM for SIK1, SIK2 and SIK3 respectively.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Sundberg TB, Choi HG, et al. Small-molecule screening identifies inhibition of salt-inducible kinases as a therapeutic strategy to enhance immunoregulatory functions of dendritic cells. Proc Natl Acad Sci U S A. 2014 Aug 26;111(34):12468-73.
- [2] Clark K, MacKenzie KF, et al. Phosphorylation of CRTC3 by the salt-inducible kinases controls the interconversion of classically activated and regulatory macrophages. Proc Natl Acad Sci U S A. 2012 Oct 16;109(42):16986-91.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 1456858-58-4 | 储存条件 |
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| 分子式 | C32H37N7O3 | 运输 | 蓝冰 | |
| 分子量 | 567.68 | 别名 | SIK inhibitor 1 |
