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CAS No.: 743420-02-2
Synonyms: Chidamide impurity
HDAC-IN-7 is an analogue of Chidamide. Chidamide is a class I HDAC inhibitor with IC50s of 95/160/67/733 nM for HDAC1/2/3/8, also inhibiting HDAC10/11 (IC50=78/432 nM) and showing no inhibition on HDAC4/5/7/9/6 (IC50> 30 μM).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT03574402 | Carcinoma, Non-Small-Cell Lung | Phase 2 | Not yet recruiting | December 30, 2024 | - |
NCT03453255 | Chemotherapy | Phase 1 Phase 2 | Recruiting | December 31, 2020 | China ... more >> Chinese PLA General Hospital Recruiting Beijing, China, 100853 Contact: Li Yu, M.D. Ph.D. 86-010-55499003 chunhuiliyu@yahoo.com Principal Investigator: Li Yu, M.D. Ph.D. Collapse << |
NCT02697552 | Non-Hodgkin's Lymphoma | Phase 1 | Completed | - | Japan ... more >> Nagoya City University Hospital Aichi, Japan Fukuoka University Hospital Fukuoka, Japan NHO Kyushu Cancer Center Fukuoka, Japan Kagoshima University Medical and Dental Hospital Kagoshima, Japan Tokai University Hospital Kanagawa, Japan NHO Kumamoto Medical Center Kumamoto, Japan NHO Nagasaki Medical Center Nagasaki, Japan National Cancer Center Hospital Tokyo, Japan Collapse << |
实验方案
技术信息
CAS号 | 743420-02-2 | 储存条件 |
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分子式 | C22H19FN4O2 | 运输 | 蓝冰 | |||||
分子量 | 390.41 | 别名 | Chidamide impurity | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03574402 | Carcinoma, Non-Small-Cell Lung | Phase 2 | Not yet recruiting | December 30, 2024 | - |
NCT03453255 | Chemotherapy | Phase 1 Phase 2 | Recruiting | December 31, 2020 | China ... more >> Chinese PLA General Hospital Recruiting Beijing, China, 100853 Contact: Li Yu, M.D. Ph.D. 86-010-55499003 chunhuiliyu@yahoo.com Principal Investigator: Li Yu, M.D. Ph.D. Collapse << |
NCT02697552 | Non-Hodgkin's Lymphoma | Phase 1 | Completed | - | Japan ... more >> Nagoya City University Hospital Aichi, Japan Fukuoka University Hospital Fukuoka, Japan NHO Kyushu Cancer Center Fukuoka, Japan Kagoshima University Medical and Dental Hospital Kagoshima, Japan Tokai University Hospital Kanagawa, Japan NHO Kumamoto Medical Center Kumamoto, Japan NHO Nagasaki Medical Center Nagasaki, Japan National Cancer Center Hospital Tokyo, Japan Collapse << |
NCT02718066 | Melanoma Rena... more >>l Cell Carcinoma Non-Small Cell Lung Cancer Collapse << | Phase 1 Phase 2 | Recruiting | January 2020 | United States, Arizona ... more >> [Site 02] Mayo Clinic Arizona Recruiting Phoenix, Arizona, United States, 85054 Contact: Thai Ho United States, California [Site 11] University of California, San Diego Medical Center Recruiting La Jolla, California, United States, 92037 Contact: Lyudmila Bazhenova United States, Florida [Site 01] Hematology - Oncology Associates of the Treasure Coast Recruiting Port Saint Lucie, Florida, United States, 34952 Contact: Heather Yeckes-Rodin [Site 09] H. Lee Moffitt Cancer Center and Research Institute, Inc. Recruiting Tampa, Florida, United States, 33612 Contact: Nikhil Khushalani United States, Maryland [Site 13] Frederick Memorial Hospital d/b/a James M Stockman Cancer Institute Recruiting Frederick, Maryland, United States, 21702 Contact: Elhamy Eskander United States, Texas [Site 12] University of Texas M.D. Anderson Cancer Center - Investigational Cancer Therapeutics Recruiting Houston, Texas, United States, 77030 Contact: Siqing Fu Collapse << |
NCT03564470 | Leukemia Leuk... more >>emia, Acute Leukemia, Lymphoblastic Leukemia, B-cell Collapse << | Phase 2 Phase 3 | Recruiting | August 30, 2020 | China, Guangdong ... more >> Department of Hematology, Nanfang Hospital Recruiting Guangzhou, Guangdong, China, 510515 Contact: Hongsheng Zhou, PhD, MD 86-20-62787349 zhs1@i.smu.edu.cn Collapse << |
NCT03617432 | Experimental Tumor | Phase 2 | Recruiting | September 30, 2022 | China ... more >> Beijing Cancer Hospital Recruiting Beijing, China, 100142 Contact: Jun Zhu, MD +86-10-88196596 zj@bjcancer.org Contact: Weiping Liu, MD +86-10-88196109 dreaming2217@126.com Principal Investigator: Jun Zhu, MD Collapse << |
NCT03605056 | Multiple Myeloma | Phase 2 | Not yet recruiting | July 31, 2022 | China, Shanghai ... more >> 180 Fenglin Road Active, not recruiting Shanghai, Shanghai, China, 200032 Collapse << |
NCT03321890 | Peripheral T-cell Lymphoma | Phase 2 | Recruiting | December 31, 2020 | China, Guangdong ... more >> Department of Medical Oncology,Sun Yat-Sen University Cancer Center Recruiting Guangzhou, Guangdong, China, 510060 Contact: Zhiming Li, DM +86-13719189172 Lizhm@sysucc.org.cn Contact: Yu Wang, DM 86-20-87343765 Wangyu@sysucc.org.cn Collapse << |
NCT03602131 | Hodgkin Lymphoma ... more >> Non-hodgkin Lymphoma Collapse << | Phase 2 | Not yet recruiting | March 30, 2021 | - |
NCT03564704 | Leukemia Leuk... more >>emia, Acute Adult Lymphoblastic Lymphoma Leukemia, Lymphoblastic Leukemia, T Cell Adult Acute Lymphoblastic Leukemia Lymphoblastic Lymphoma Lymphoblastic Leukemia Collapse << | Phase 2 Phase 3 | Recruiting | May 30, 2021 | China, Guangdong ... more >> Department of Hematology, Nanfang Hospital Recruiting Guangzhou, Guangdong, China, 510515 Contact: Hongsheng Zhou +862062787349 zhs1@i.smu.edu.cn Collapse << |
NCT03023358 | Peripheral T Cell Lymphoma | Phase 3 | Not yet recruiting | March 2019 | China, Guangdong ... more >> Ru Feng Not yet recruiting Guangzhou, Guangdong, China, 510515 Contact: Ru Feng, M.D. +86 13725119762 ruth1626@hotmail.com Contact: Qi Wei, M.D. +86 13427564102 sinbad37@126.com Principal Investigator: Ru Feng, M.D. Collapse << |
NCT03151876 | Lymphoma | Phase 2 | Recruiting | December 2021 | China, Beijing ... more >> Beijing cancer hospital Not yet recruiting Beijing, Beijing, China, 100142 Contact: Yan Xie, MD Peking university third hospital Not yet recruiting Beijing, Beijing, China, 100191 Contact: Xiaoyan Ke, MD China, Chongqing The first affiliated hospital of Chongqing medical university Not yet recruiting Chongqing, Chongqing, China, 400016 Contact: Lin Liu, MD Southwest Hospital Recruiting Chongqing, Chongqing, China, 400038 Contact: Dabing Qin, MD China, Gansu General Hospital of Lanzhou military command Not yet recruiting Lanzhou, Gansu, China, 730070 Contact: Hai Bai, MD China, Henan Henan cancer hospital Not yet recruiting Zhengzhou, Henan, China, 450008 Contact: Jian Zhou, MD The first affiliated hospital of Zhengzhou university Not yet recruiting Zhengzhou, Henan, China, 450052 Contact: Xinhua Wang, MD China, Hubei Tongji Hospital Not yet recruiting Wuhan, Hubei, China, 430030 Contact: Yang Cao, MD China, Jiangsu Jiangsu province hospital Not yet recruiting Nanjing, Jiangsu, China, 210029 Contact: Wei Xu, MD China, Shanghai Rui jin hospital Shanghai jiao tong University Not yet recruiting Shanghai, Shanghai, China, 200025 Contact: Jiong Hu, MD Tong Ren Hospital Not yet recruiting Shanghai, Shanghai, China Contact: Ligen L i u, MD China, Shanxi Shan Xi Da Yi Hospital Not yet recruiting Taiyuan, Shanxi, China, 030032 Contact: Rong Gong, MD Tangdu Hospital Not yet recruiting Xi'an, Shanxi, China, 710038 Contact: Qiang Liu, MD China, Sichuan West China Hospital of Sichuan University Recruiting Chengdu, Sichuan, China, 610044 Contact: Jie Ji, MD 86-28-85422370 jieji@scu.edu.cn Affiliated Hospital of Southwest Medical University Recruiting Nanchong, Sichuan, China, 646000 Contact: Xiaoming Li, MD China, Tianjing Blood diseases hospital, Chinese academy of medica Not yet recruiting Tianjin, Tianjing, China, 300020 Contact: Lvgui Qiu, MD China, Xinjiang The first affiliated hospital of Xinjiang medical Universtiy Not yet recruiting Ürümqi, Xinjiang, China, 830054 Contact: Ming Jiang, MD China, Yunnan Kunming General Hospital of Chengdu Military Area Not yet recruiting Kunming, Yunnan, China, 650032 Contact: Sanbin Wang, MD Collapse << |
NCT03629873 | Lymphoma, Large B-Cell, Diffus... more >>e Mantle Cell Lymphoma Peripheral T Cell Lymphoma Double-hit Lymphoma Collapse << | Phase 2 | Recruiting | August 1, 2020 | China, Jiangsu ... more >> Hematological Department, People's Hospital of Jiangsu Province Recruiting Nanjing, Jiangsu, China, 210029 Contact: Wei Xu, Ph.D. +86-2568302182 xuwei10000@hotmail.com Collapse << |
NCT02809573 | Peripheral T-cell Lymphoma | Phase 1 | Recruiting | December 2019 | China, Beijing ... more >> Cancer Hospital, Chinese Academy of Medical Sciences Recruiting Beijing, Beijing, China, 100000 Contact: Yuankai Shi, MD +86-10-8778-8293 syuankai@cicams.ac.cn Collapse << |
NCT02879526 | Relapse/Refratory Peripheral T... more >> Cell Lymphoma Collapse << | Phase 2 | Recruiting | August 2019 | China, Jiangsu ... more >> HuaiAn First People's Hospital Recruiting HuaiAn, Jiangsu, China, 223300 Contact: Liang Yu, M.D., Ph.D. WuXi People's Hospital Recruiting WuXi, Jiangsu, China, 214023 Contact: Yun Zhuang, M.D. Contact: YunFeng Shen, M.D., Ph.D Collapse << |
NCT01836679 | Non-small-cell Lung Cancer | Phase 2 | Completed | - | China, Beijing ... more >> Cancer Hospital, Chinese Academy of Medical Sciences Beijing, Beijing, China, 100021 Beijing Chest Hospital, Capital Medical University Beijing, Beijing, China, 101149 China, Hebei Hebei Provincial Tumor Hospital Shijiazhuang, Hebei, China, 050011 China, Jiangsu Jiangsu Cancer Hospital Nanjing, Jiangsu, China, 210009 China, Liaoning The first Hospital of China Medical University Shenyang, Liaoning, China, 110001 China, Shanghai Shanghai Chest Hospital Affiliated to Shanghai Jiaotong University Shanghai, Shanghai, China, 200030 China, Sichuan The Second People's Hospital of Sichuan Chengdu, Sichuan, China, 82816 China, Tianjin Tianjin Medical University Cancer Institute & Hospital Tianjin, Tianjin, China, 300060 Collapse << |
NCT02753647 | Diffuse Large B-cell Lymphoma | Phase 2 | Recruiting | April 2019 | China, Shanghai ... more >> Shanghai Ruijin Hospital Recruiting Shanghai, Shanghai, China, 200023 Contact: Weili Zhao, MD,PhD 64370045 ext 610707 zhao.weili@yahoo.com Contact: Pengpeng Xu, MD 64370045 ext 610707 xpproc@msn.com Collapse << |
NCT02733380 | Diffuse Large B-cell Lymphoma | Phase 2 | Recruiting | May 2020 | China, Henan ... more >> Henan Cancer Hospital/The affiliated Cancer Hospital of ZhengZhou university Recruiting ZhengZhou, Henan, China, 450008 Contact: Yanyan Liu, M.D. +8613838176375 yyliu@zzu.edu.cn Contact: Jiuyang Zhang, Master +8615003810435 zhangjiuyang9103@163.com Principal Investigator: Yanyan Liu, M.D. Collapse << |
NCT03031262 | AML | Phase 1 Phase 2 | Recruiting | December 2022 | China, Tianjin ... more >> Institute of Hematology & Blood Diseases Hospital Recruiting Tianjin, Tianjin, China Contact: lijun Liu 86-22-23909237 bloodgcp@126.com Collapse << |
NCT02886559 | AML Relapse | Phase 1 Phase 2 | Recruiting | June 2019 | China ... more >> China PLA General Hospital Recruiting Beijing, China, 100039 Contact: Li Yu, M.D Ph.D 010-66937644 chunhuiliyu@yahoo.com Principal Investigator: Li-Xin Yu Collapse << |
NCT03553238 | Leukemia, Acute ... more >> Leukemia, T Cell Leukemia, Lymphoblastic Collapse << | Phase 2 Phase 3 | Recruiting | August 30, 2020 | China, Guangdong ... more >> Nanfang Hospital, Southern Medical University Recruiting Guangzhou, Guangdong, China, 510515 Contact: Hongsheng Zhou, MD, PhD +862062787349 zhs1@i.smu.edu.cn Collapse << |
NCT03630731 | Natural Killer/T-Cell Lymphoma... more >>, Nasal and Nasal-Type Collapse << | Phase 2 | Recruiting | March 2020 | China, Beijing ... more >> Cancer Hospital and Institute, Chinese Academy of Medical Sciences (CAMS) and Peking Union Medical College (PUMC) Recruiting Beijing, Beijing, China, 100021 Contact: Mei Dong (86)13811929322 dongmei030224@163.com Collapse << |
NCT02987244 | T Cell Non-Hodgkin's Lymphoma | Phase 1 Phase 2 | Recruiting | March 2023 | China, Beijing ... more >> Peking Union medical college hospital Recruiting Beijing, Beijing, China, 100730 Contact: Wei Zhang China, Tianjin Tianjin medical universty cancer institute & hospital Recruiting Tianjin, Tianjin, China, 300060 Collapse << |
NCT02753543 | Peripheral T Cell Lymphoma | Phase 2 | Recruiting | November 2019 | China, Shanghai ... more >> Ruijin Hospital Recruiting Shanghai, Shanghai, China, 200023 Contact: Weili Zhao, MD, PhD 64370045 ext 610707 zhao.weili@yahoo.com Contact: Pengpeng Xu, MD 64370045 ext 610707 xpproc@msn.com Collapse << |
NCT03336632 | Leukemia, Acute ... more >> MDS Collapse << | Phase 2 | Not yet recruiting | March 30, 2021 | China, Sichuan ... more >> West China Hospital of Sichuan University Chengdu, Sichuan, China, 610044 West China Hospital of Sichuan University Not yet recruiting Chengdu, Sichuan, China, 610044 Contact: Jie Ji, MD 86-28-85422370 jieji@scu.edu.cn Collapse << |
NCT02482753 | Breast Cancer | Phase 3 | Active, not recruiting | March 2019 | China, Beijing ... more >> The 307th Hospital of Chinese people's Liberation Army Beijing, Beijing, China, 100021 Collapse << |
NCT03273452 | Angioimmunoblastic T-cell Lymp... more >>homa Collapse << | Phase 2 | Recruiting | May 2019 | China, Shandong ... more >> The Affiliated Hospital of Qingdao University Recruiting Qingdao, Shandong, China, 266000 Contact: Hongwei Xue, MD. PhD (+86)13475875599 Xuehongwei1867@163.com Collapse << |
NCT03245905 | Relapsed or Refractory B-cell ... more >>Non-Hodgkin's Lymphoma (NHL) Collapse << | Phase 2 | Not yet recruiting | September 30, 2019 | China, Guangdong ... more >> Department of Medical Oncology, Sun Yat-sen University Cancer Center, Guangzhou, Guangdong, China, 510060 Collapse << |
NCT03598959 | Extranodal NK/T-cell Lymphoma | Phase 2 | Not yet recruiting | December 31, 2021 | China, Sichuan ... more >> West China Hospital of Sichuan University Chengdu, Sichuan, China, 610044 Collapse << |
NCT03494634 | Experimental Tumor | Phase 2 | Not yet recruiting | September 30, 2020 | China, Guangdong ... more >> Cancer Center of Sun Yat-Sen University (CCSU) Guangzhou, Guangdong, China Collapse << |
NCT03201471 | Diffuse Large B Cell Lymphoma | Phase 2 | Recruiting | February 5, 2020 | China, Zhejiang ... more >> The first affiliated hospital of Zhejiang University Recruiting Hangzhou, Zhejiang, China, 310000 Contact: Wenbin Qian, MD. PhD. (+86)13605801032 Collapse << |
NCT03611231 | Experimental Tumor | Phase 2 | Not yet recruiting | December 30, 2022 | China, Beijing ... more >> Beijing Not yet recruiting Beijing, Beijing, China, 100000 Contact: Yuqin Song, Dr. 0086 13683398726 songyuqin622@163.com Collapse << |
NCT02902185 | Chronic HIV Infections | Phase 2 Phase 3 | Active, not recruiting | December 2018 | China, Guangxi ... more >> The First Affiliated Hospital of Guangxi Medical University Nanning, Guangxi, China China, Shaanxi Department of Infectious Diseases, Tangdu Hospital, The Fourth Military Medical University Xi'an, Shaanxi, China, 710038 China, Zhejiang Zhejiang University Hangzhou, Zhejiang, China Collapse << |
NCT02856997 | Peripheral T Cell Lymphoma | Phase 2 | Not yet recruiting | - | - |
NCT02815007 | Advanced EGFR-TKI-resistant No... more >>n-Small Cell Lung Cancer Collapse << | Phase 2 | Unknown | June 2018 | - |
NCT02878278 | Lymphoma, Extranodal NK-T-Cell... more >> EBV Collapse << | Phase 2 | Not yet recruiting | September 2019 | - |
NCT03410004 | Experimental | Phase 2 | Not yet recruiting | September 30, 2020 | - |
NCT03373019 | Chidamide Lym... more >>phoma, B-Cell Lymphoma, Large B-Cell, Diffuse Neoplasm by Histology Neoplasms Lymphoproliferative Disorders Lymphatic Diseases Immunoproliferative Disorders Immune System Diseases Lymphoma, Non-Hodgkin Cyclophosphamide Rituximab Gemcitabine Cisplatin Dexamethasone HDAC Inhibitor Collapse << | Phase 2 | Recruiting | March 1, 2021 | China, Shanghai ... more >> Kai Xue Recruiting Shanghai, Shanghai, China, 200032 Contact: Kai Xue, MD 13818659448 xuekaishanghai@126.com China Kai Xue Recruiting Shanghai, China Contact: Kai Xue, MD 13818659448 xuekaishanghai@126.com Contact: Junning Cao, MD 13818659448 Collapse << |
NCT02513901 | Chronic HIV Infections | Phase 1 Phase 2 | Completed | - | China, Shaanxi ... more >> Department of Infectious Diseases, Tangdu Hospital, The Fourth Military Medical University Xi'an, Shaanxi, China, 710038 Collapse << |
NCT03268889 | Peripheral T Cell Lymphoma | Not Applicable | Recruiting | September 15, 2020 | China, Jiangsu ... more >> the First Affiliated Hospital of Soochow University Recruiting Suzhou, Jiangsu, China, 215006 Contact: Zhengming Jin, MD, PhD (+86)512-67781856 Collapse << |
NCT02883374 | Adenocystic Carcinoma | Phase 2 | Recruiting | June 2020 | China, Beijing ... more >> Cancer Hospital, Chinese Academy of Medical Science Recruiting Beijing, Beijing, China, 100021 Contact: Mei Dong, Doctor 13811929322 dongmei030224@163.com Principal Investigator: Mei Dong, Doctor Collapse << |
NCT03105596 | B-cell Non-Hodgkin's Lymphoma | Phase 2 | Not yet recruiting | September 30, 2019 | - |
NCT02944812 | Peripheral T Cell Lymphoma | Phase 2 | Recruiting | January 2019 | China, Guangdong ... more >> Guangdong general hospital Recruiting Guangzhou, Guangdong, China, 510080 Contact: Wenyu Li, MD PhD +86 20 81884713-80412 Collapse << |
NCT03639168 | Adenoid Cystic Carcinomas ... more >> Chidamide Cisplatin Collapse << | Phase 2 | Recruiting | June 1, 2020 | China, Shanghai ... more >> Kai Xue Recruiting Shanghai, Shanghai, China, 200032 Contact: Kai Xue, MD 13818659448 xuekaishanghai@126.com Collapse << |
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