CAS No.: 439288-66-1
GW627368 Catalog No. CSN18274
Synonyms: GW 627368X
GW627368 is a potent and selective competitive antagonist of prostanoid EP4 receptor (Ki= 100 nM) with additional human TP receptor affinity (Ki= 150 nM).
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Parida S, Parekh A, et al. Molecular inhibition of prostaglandin E2 with GW627368X: Therapeutic potential and preclinical safety assessment in mouse sarcoma model. Cancer Biol Ther. 2015;16(6):922-32.
- [2] Wilson RJ, Giblin GM, et al. GW627368X((N-{2-[4-(4,9-diethoxy-1-oxo-1,3-dihydro-2H-benzo[f] isoindol-2-yl)phenyl] acetyl} benzene sulphonamide): a novel, potent and selective prostanoid EP4 receptor antagonist. Br J Pharmacol. 2006 Jun;148(3):326-39.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 439288-66-1 | 储存条件 |
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| 分子式 | C30H28N2O6S | 运输 | 蓝冰 | |||||
| 分子量 | 544.62 | 别名 | GW 627368X | |||||
| 溶解度 |
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动物实验配方 |
