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CAS No.: 1032823-75-8
GSK1292263 is an agonist of GPR119 receptor that is used to treat type 2 diabetes.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00783549 | Dyslipidaemias | Phase 1 | Completed | - | United States, Minnesota ... more >> GSK Investigational Site Minneapolis, Minnesota, United States, 55404 Collapse << |
NCT01218204 | Dyslipidaemias | Phase 2 | Completed | - | - |
NCT01128621 | Diabetes Mellitus, Type 2 | Phase 2 | Completed | - | United States, California ... more >> GSK Investigational Site Chula Vista, California, United States, 91910 United States, Florida GSK Investigational Site Miami, Florida, United States, 33169 Collapse << |
实验方案
技术信息
CAS号 | 1032823-75-8 | 储存条件 |
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分子式 | C23H28N4O4S | 运输 | 蓝冰 | |||||||
分子量 | 456.56 | 别名 | ||||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00783549 | Dyslipidaemias | Phase 1 | Completed | - | United States, Minnesota ... more >> GSK Investigational Site Minneapolis, Minnesota, United States, 55404 Collapse << |
NCT01218204 | Dyslipidaemias | Phase 2 | Completed | - | - |
NCT01128621 | Diabetes Mellitus, Type 2 | Phase 2 | Completed | - | United States, California ... more >> GSK Investigational Site Chula Vista, California, United States, 91910 United States, Florida GSK Investigational Site Miami, Florida, United States, 33169 Collapse << |
NCT01128621 | - | - | Completed | - | - |
NCT01218204 | - | - | Completed | - | - |
NCT01101568 | Diabetes Mellitus, Type 2 | Phase 1 | Completed | - | United States, Texas ... more >> GSK Investigational Site Austin, Texas, United States, 78744 Collapse << |
NCT01119846 | Diabetes Mellitus, Type 2 | Phase 2 | Completed | - | United States, Arizona ... more >> GSK Investigational Site Phoenix, Arizona, United States, 85013 United States, California GSK Investigational Site Chula Vista, California, United States, 91910 United States, Florida GSK Investigational Site Miami, Florida, United States, 33169 United States, North Carolina GSK Investigational Site Durham, North Carolina, United States, 27705 United States, Ohio GSK Investigational Site Columbus, Ohio, United States, 43212 United States, Texas GSK Investigational Site San Antonio, Texas, United States, 78209 United States, Washington GSK Investigational Site Tacoma, Washington, United States, 98418 Collapse << |
NCT01119846 | - | - | Completed | - | - |
靶点 | Description | IC50 |
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