CAS No.: 172854-55-6
GR 55562 hydrochloride Catalog No. CSN13859
GR55562 is a selective competitive 5-HT1B(5-HT1Dβ) silent antagonist with pKB values of 7.3 and 6.3 for human cloned 5-HT1B and 5-HT1D receptors respectively and only weak binding at a number of other 5-HT subtypes.
| 规格 | 价格 | 促销价格 | 库存 | 数量 |
|---|
400-920-2911
sales@csnpharm.cn
tech@csnpharm.cn
纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Maassen VanDenBrink A, et al. Human isolated coronary artery contraction to sumatriptan characterised by the selective 5-HT1B/1D receptor antagonist GR55562. Pharmacol Toxicol. 2000 Jun;86(6):287-90.
- [2] MacLean MR, Clayton RA, et al. Evidence for 5-HT1-like receptor-mediated vasoconstriction in human pulmonary artery. Br J Pharmacol. 1996 Sep;119(2):277-82.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 172854-55-6 | 储存条件 |
|
|
| 分子式 | C23H26ClN3O2 | 运输 | 蓝冰 | |
| 分子量 | 411.92 | 别名 |
