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CAS No.: 1391076-61-1

GLPG0974 Catalog No. CSN22413

GLPG0974 is a free fatty acid receptor-2 (FFA2/GPR43) antagonist with an IC50 of 9 nM.

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靶点选择性

生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT01496937HealthyPhase 1Completed-Belgium ... more >> SGS Stuivenberg Antwerp, Belgium Collapse <<
    NCT01829321Ulcerative ColitisPhase 2Completed-Belgium ... more >> Imelda Bonheiden, Belgium UZ Gent Gent, Belgium AZ Groeninge Kortrijk, Belgium UZ Leuven Leuven, Belgium Czech Republic Hepato-Gastroenterologie HK, s.r.o. Hradec Kralove, Czech Republic Fakulní nemocnice Olomouc Olomouc, Czech Republic Homolka Hospitál Prague, Czech Republic Nemocnice Slaný Slany, Czech Republic Krajská zdravotní a.s., Masarykova nemocnice v Ústí nad Labem T. Bati a.s. Usti nad Labem, Czech Republic Krajská nemocnice Tomáše Bati - Zlin Zlin, Czech Republic Nemocnice Znojmo Znojmo, Czech Republic Latvia Latvijas Jūras Medicīnas Centrs Riga, Latvia Rīgas slimnīca Bikor Holim Riga, Latvia SIA Gremošanas slimību centrs "Gastro" Riga, Latvia Slovakia Univerzitná nemocnica Bratislava Bratislava, Slovakia Fakultná Nemocnica Nitra Nitra, Slovakia Collapse <<
    NCT01721980HealthyPhase 1Completed-Belgium ... more >> SGS LSS Clinical Pharmacology Unit Antwerp Antwerp, Belgium Collapse <<

实验方案

技术信息

CAS号 1391076-61-1 储存条件
分子式 C25H25ClN2O4S 运输 蓝冰
分子量 485.00 别名

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