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CAS No.: 1391076-61-1
GLPG0974 is a free fatty acid receptor-2 (FFA2/GPR43) antagonist with an IC50 of 9 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01496937 | Healthy | Phase 1 | Completed | - | Belgium ... more >> SGS Stuivenberg Antwerp, Belgium Collapse << |
NCT01829321 | Ulcerative Colitis | Phase 2 | Completed | - | Belgium ... more >> Imelda Bonheiden, Belgium UZ Gent Gent, Belgium AZ Groeninge Kortrijk, Belgium UZ Leuven Leuven, Belgium Czech Republic Hepato-Gastroenterologie HK, s.r.o. Hradec Kralove, Czech Republic Fakulní nemocnice Olomouc Olomouc, Czech Republic Homolka Hospitál Prague, Czech Republic Nemocnice Slaný Slany, Czech Republic Krajská zdravotní a.s., Masarykova nemocnice v Ústí nad Labem T. Bati a.s. Usti nad Labem, Czech Republic Krajská nemocnice Tomáše Bati - Zlin Zlin, Czech Republic Nemocnice Znojmo Znojmo, Czech Republic Latvia Latvijas Jūras Medicīnas Centrs Riga, Latvia Rīgas slimnīca Bikor Holim Riga, Latvia SIA Gremošanas slimību centrs "Gastro" Riga, Latvia Slovakia Univerzitná nemocnica Bratislava Bratislava, Slovakia Fakultná Nemocnica Nitra Nitra, Slovakia Collapse << |
NCT01721980 | Healthy | Phase 1 | Completed | - | Belgium ... more >> SGS LSS Clinical Pharmacology Unit Antwerp Antwerp, Belgium Collapse << |
实验方案
技术信息
CAS号 | 1391076-61-1 | 储存条件 |
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分子式 | C25H25ClN2O4S | 运输 | 蓝冰 | |
分子量 | 485.00 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01496937 | Healthy | Phase 1 | Completed | - | Belgium ... more >> SGS Stuivenberg Antwerp, Belgium Collapse << |
NCT01829321 | Ulcerative Colitis | Phase 2 | Completed | - | Belgium ... more >> Imelda Bonheiden, Belgium UZ Gent Gent, Belgium AZ Groeninge Kortrijk, Belgium UZ Leuven Leuven, Belgium Czech Republic Hepato-Gastroenterologie HK, s.r.o. Hradec Kralove, Czech Republic Fakulní nemocnice Olomouc Olomouc, Czech Republic Homolka Hospitál Prague, Czech Republic Nemocnice Slaný Slany, Czech Republic Krajská zdravotní a.s., Masarykova nemocnice v Ústí nad Labem T. Bati a.s. Usti nad Labem, Czech Republic Krajská nemocnice Tomáše Bati - Zlin Zlin, Czech Republic Nemocnice Znojmo Znojmo, Czech Republic Latvia Latvijas Jūras Medicīnas Centrs Riga, Latvia Rīgas slimnīca Bikor Holim Riga, Latvia SIA Gremošanas slimību centrs "Gastro" Riga, Latvia Slovakia Univerzitná nemocnica Bratislava Bratislava, Slovakia Fakultná Nemocnica Nitra Nitra, Slovakia Collapse << |
NCT01721980 | Healthy | Phase 1 | Completed | - | Belgium ... more >> SGS LSS Clinical Pharmacology Unit Antwerp Antwerp, Belgium Collapse << |
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