CAS No.: 3717-88-2
Flavoxate HCl/盐酸黄酮哌酯 Catalog No. CSN11016
Synonyms: Rec-7-0040;DW61;NSC 114649
Flavoxate HCl is a competitive AChR antagonist with IC50 of 12.2 μM, used as a muscle relaxant.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 临床研究
NCT号 适应症或疾病 临床期 招募状态 预计完成时间 地点 NCT00440739 Pain Phase 4 Completed - Thailand ... more >> Faculty of Medicine Siriraj Hospital, Mahidol University Bangkok, Thailand, 10700 Collapse << NCT00992238 Healthy Phase 1 Completed - United States, North Dakota ... more >> PRACS Institute, Ltd Fargo, North Dakota, United States, 58104 Collapse << NCT00992238 Healthy Phase 1 Completed - United States, North Dakota ... more >> PRACS Institute, Ltd Fargo, North Dakota, United States, 58104 Collapse << - 更多
- 参考文献
- [1] Dansette PM, Jaoen M, et al. HMG-CoA reductase activity in human liver microsomes: comparative inhibition by statins. Exp Toxicol Pathol. 2000 May;52(2):145-8.
- [2] Kimura Y, Sasaki Y, et al. Mechanisms of the suppression of the bladder activity by flavoxate. Int J Urol. 1996 May;3(3):218-27.
- [3] Tomoda T, Aishima M, Takano N, Nakano T, Seki N, Yonemitsu Y, Sueishi K, Naito S, Ito Y, Teramoto N. The effects of flavoxate hydrochloride on voltage-dependent L-type Ca2+ currents in human urinary bladder. Br J Pharmacol. 2005 Sep;146(1):25-32.
- [4] Oka M, Kimura Y, Itoh Y, Sasaki Y, Taniguchi N, Ukai Y, Yoshikuni Y, Kimura K. Brain pertussis toxin-sensitive G proteins are involved in the flavoxate hydrochloride-induced suppression of the micturition reflex in rats. Brain Res. 1996 Jul 15;727(1-2):91-8.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 3717-88-2 | 储存条件 |
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| 分子式 | C24H26ClNO4 | 运输 | 蓝冰 | |||||
| 分子量 | 427.92 | 别名 | Rec-7-0040;DW61;NSC 114649;Flavoxate (hydrochloride);Rec 7/0040;Flavoxate HCl;黄酮盐酸盐 | |||||
| 溶解度 |
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动物实验配方 |
