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CAS No.: 754240-09-0
Synonyms: EHT 1864
EHT 1864 2HCl is an inhibitor of Rac1 (Kd = 40 nM), Rac1b (Kd = 50 nM), Rac2 (Kd = 60 nM) and Rac3 (Kd = 250 nM).
生物活性
实验方案
技术信息
CAS号 | 754240-09-0 | 储存条件 |
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分子式 | C25H29Cl2F3N2O4S | 运输 | 蓝冰 | |||||
分子量 | 581.48 | 别名 | EHT 1864 | |||||
溶解度 |
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动物实验配方 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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293T cells | - | Function assay | - | Effect on Rac1 binding to RhoGDI2 expressed in 293T cells by Western blot analysis | 17932039 |
mouse NIH3T3 cells | - | Function assay | - | Effect on Rac1 binding to RhoGDI2 in mouse NIH3T3 cells by Western blot analysis | 17932039 |
mouse NIH3T3 cells | - | Function assay | - | Effect on Rac1 binding to RhoGDI1 in mouse NIH3T3 cells by Western blot analysis | 17932039 |
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