CAS No.: 257639-98-8
CP-154526 Hydrochloride Catalog No. CSN20174
CP-154526 HCl is a selective, non-peptide CRF1 receptor antagonist (Ki values are 2.7 and > 10000 nM for CRF1 and CRF2 receptors respectively). CP-154526 HCl blocks CRF-induced adenylate cyclase activation (Ki = 3.7 nM) and attenuates activation of the HPA axis by CRF.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Kobayashi T, Kiyokawa Y, et al. Pretreatment with CP-154526 blocks the modifying effects of alarm pheromone on components of sexual behavior in male, but not in female, rats. Chem Senses. 2011 Sep;36(7):623-32.
- [2] Nalivaiko E, Blessing WW. CRF1-receptor antagonist CP-154526 reduces alerting-related cutaneous vasoconstriction in conscious rabbits. Neuroscience. 2003;117(1):129-38.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 257639-98-8 | 储存条件 |
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| 分子式 | C23H33ClN4 | 运输 | 蓝冰 | |
| 分子量 | 400.99 | 别名 |
