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CAS No.: 1032568-63-0
Synonyms: 库潘尼西;BAY 80-6946
Copanlisib is a potent and highly selective reversible PI3K inhibitor for PI3Kα/β with IC50 of 0.469 nM/3.72 nM.
生物活性
靶点 | PI3Kα IC50:0.469nM | PI3Kβ IC50:3.72nM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01660451 | Lymphoma, Non-Hodgkin | Phase 2 | Active, not recruiting | March 8, 2019 | - |
NCT00962611 | Neoplasms | Phase 1 | Completed | - | United States, Arizona ... more >> Scottsdale, Arizona, United States, 85258 United States, Pennsylvania Pittsburgh, Pennsylvania, United States, 15213 United States, Texas San Antonio, Texas, United States, 78229-3307 Collapse << |
NCT01460537 | Neoplasms | Phase 1 | Completed | - | United States, Florida ... more >> Tampa, Florida, United States, 33612 United States, Minnesota Rochester, Minnesota, United States, 55905 United States, North Carolina Chapel Hill, North Carolina, United States, 27599-7305 Collapse << |
实验方案
技术信息
CAS号 | 1032568-63-0 | 储存条件 |
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分子式 | C23H28N8O4 | 运输 | 蓝冰 | |||||||||||||
分子量 | 480.52 | 别名 | 库潘尼西;BAY 80-6946 | |||||||||||||
溶解度 |
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动物实验配方 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01660451 | Lymphoma, Non-Hodgkin | Phase 2 | Active, not recruiting | March 8, 2019 | - |
NCT00962611 | Neoplasms | Phase 1 | Completed | - | United States, Arizona ... more >> Scottsdale, Arizona, United States, 85258 United States, Pennsylvania Pittsburgh, Pennsylvania, United States, 15213 United States, Texas San Antonio, Texas, United States, 78229-3307 Collapse << |
NCT01460537 | Neoplasms | Phase 1 | Completed | - | United States, Florida ... more >> Tampa, Florida, United States, 33612 United States, Minnesota Rochester, Minnesota, United States, 55905 United States, North Carolina Chapel Hill, North Carolina, United States, 27599-7305 Collapse << |
NCT01392521 | Neoplasms | Phase 1 | Completed | - | United States, Arizona ... more >> Scottsdale, Arizona, United States, 85260 United States, Nevada Las Vegas, Nevada, United States, 89169 United States, South Carolina Greenville, South Carolina, United States, 29605 United States, Texas Houston, Texas, United States, 77030 Tyler, Texas, United States, 75702 United States, Washington Vancouver, Washington, United States, 98684 Germany Freiburg, Baden-Württemberg, Germany, 79106 Netherlands Rotterdam, Netherlands, 3015 CE Collapse << |
NCT01411410 | Neoplasms | Phase 1 | Completed | - | United States, Missouri ... more >> Saint Louis, Missouri, United States, 63110 United States, New York New York, New York, United States, 10065 United States, Texas Houston, Texas, United States, 77030 Collapse << |
NCT01660451 | - | - | Active, not recruiting | - | - |
NCT03458728 | Mixed Tumor, Malignant | Phase 1 Phase 2 | Recruiting | August 24, 2021 | United States, Alabama ... more >> Children's Hospital of Alabama Not yet recruiting Birmingham, Alabama, United States, 35233 United States, California Children's Hospital of Los Angeles Not yet recruiting Los Angeles, California, United States, 90027-6089 Children's Hospital of Orange County Not yet recruiting Orange, California, United States, 92868-3974 United States, Colorado The Children's Hospital Recruiting Aurora, Colorado, United States, 80045 United States, District of Columbia Children's National Medical Center Not yet recruiting Washington, District of Columbia, United States, 20010-2970 United States, Georgia Children's Healthcare of Atlanta Not yet recruiting Atlanta, Georgia, United States, 30322 United States, Illinois Ann & Robert H. Lurie Children's Hospital of Chicago Withdrawn Chicago, Illinois, United States, 60611 United States, Indiana Riley Hospital For Children Not yet recruiting Indianapolis, Indiana, United States, 46202 United States, Massachusetts Dana-Farber Cancer Institute Recruiting Boston, Massachusetts, United States, 02215 United States, Michigan C.S. Mott Children's Hospital Not yet recruiting Ann Arbor, Michigan, United States, 48109 United States, Minnesota University of Minnesota Medical Center Not yet recruiting Minneapolis, Minnesota, United States, 55455 United States, New York Columbia University Medical Center Not yet recruiting New York, New York, United States, 10032 United States, Ohio Cincinnati Children's Hospital and Medical Center Not yet recruiting Cincinnati, Ohio, United States, 45229 United States, Pennsylvania Children's Hospital of Philadelphia Not yet recruiting Philadelphia, Pennsylvania, United States, 19104 Children's Hospital of Pittsburgh of UPMC Recruiting Pittsburgh, Pennsylvania, United States, 15224 United States, Tennessee St. Jude Children's Research Hospital Not yet recruiting Memphis, Tennessee, United States, 38105 United States, Texas Texas Children's Hospital Not yet recruiting Houston, Texas, United States, 77030 United States, Washington Seattle Children's Hospital Recruiting Seattle, Washington, United States, 98105 Collapse << |
NCT03128619 | Estrogen Receptor Positive ... more >> HER2/Neu Negative Invasive Breast Carcinoma Multifocal Breast Carcinoma Postmenopausal Progesterone Receptor Positive Stage I Breast Cancer Stage IA Breast Cancer Stage IB Breast Cancer Stage II Breast Cancer Stage IIA Breast Cancer Stage IIB Breast Cancer Stage III Breast Cancer Stage IIIA Breast Cancer Stage IIIB Breast Cancer Stage IIIC Breast Cancer Stage IV Breast Cancer Collapse << | Phase 1 Phase 2 | Recruiting | August 2, 2021 | United States, California ... more >> UCLA / Jonsson Comprehensive Cancer Center Recruiting Los Angeles, California, United States, 90095 Contact: Sara A. Hurvitz 310-829-5471 shurvitz@mednet.ucla.edu Principal Investigator: Sara A. Hurvitz Collapse << |
NCT03377101 | Estrogen Receptor Positive ... more >> HER2/Neu Negative Progesterone Receptor Positive Stage IV Breast Cancer AJCC v6 and v7 Collapse << | Phase 2 | Withdrawn(change in study desi... more >>gn.) Collapse << | - | - |
NCT02253420 | Medical Oncology | Phase 1 | Active, not recruiting | December 19, 2018 | United States, Texas ... more >> Dallas, Texas, United States, 75230 Canada, Alberta Edmonton, Alberta, Canada, T6G 1Z2 Canada, British Columbia Vancouver, British Columbia, Canada, V5Z 4E6 Canada, Ontario Hamilton, Ontario, Canada, L8V 5C2 Toronto, Ontario, Canada, M5G 2M9 Collapse << |
NCT02455297 | Lymphoma, Mantle-Cell | Phase 2 | Terminated | - | United States, Maryland ... more >> Baltimore, Maryland, United States, 21287 United States, New Jersey Hackensack, New Jersey, United States, 07601 United States, New York New York, New York, United States, 10021 New York, New York, United States, 10029 United States, Vermont Burlington, Vermont, United States, 05401 Collapse << |
NCT02626455 | Lymphoma, Non-Hodgkin | Phase 3 | Recruiting | December 31, 2024 | - |
NCT03172884 | Hepatic Insufficiency | Phase 1 | Recruiting | July 17, 2019 | Germany ... more >> CRS Clinical-Research-Services Mönchengladbach GmbH Withdrawn Mönchengladbach, Nordrhein-Westfalen, Germany, 41061 CRS Clinical-Research-Services Kiel GmbH Recruiting Kiel, Schleswig-Holstein, Germany, 24105 Romania Institutul National de Boli Infectioase Prof.Dr.Matei Bals Not yet recruiting Bucuresti, Romania, 021105 Collapse << |
NCT02342665 | Lymphoma Non-Hodgkin | Phase 1 Phase 2 | Active, not recruiting | October 31, 2021 | Japan ... more >> Nagoya, Aichi, Japan, 460-0001 Nagoya, Aichi, Japan, 464-8681 Nagoya, Aichi, Japan, 466-8560 Nagoya, Aichi, Japan, 466-8650 Nagoya, Aichi, Japan, 467-8602 Maebashi, Gunma, Japan, 371-8511 Kobe, Hyogo, Japan, 650-0017 Sendai, Miyagi, Japan, 980-8574 Chuo-ku, Tokyo, Japan, 104-0045 Koto-ku, Tokyo, Japan, 135-8550 Fukuoka, Japan, 811-1395 Fukuoka, Japan, 812-8582 Kyoto, Japan, 602-8566 Collapse << |
NCT02369016 | Lymphoma, Non-Hodgkin | Phase 3 | Active, not recruiting | December 20, 2019 | Brazil ... more >> Jaú, Sao Paulo, Brazil, 17210-120 São Paulo, Sao Paulo, Brazil, 08270-070 Sao Paulo, Brazil Bulgaria Plovdiv, Bulgaria, 4002 China, Heilongjiang Harbin, Heilongjiang, China France France, France Greece Athens, Greece, 11526 Italy Bologna, Emilia-Romagna, Italy, 40138 Genova, Liguria, Italy, 16132 Korea, Republic of Jeollabuk-do, Korea, Republic of, 561-712 Jeollanam-do, Korea, Republic of, 519-763 Seoul, Korea, Republic of, 03080 Seoul, Korea, Republic of, 03722 Seoul, Korea, Republic of, 05505 Poland Gdynia, Poland, 81-519 Portugal Almada, Portugal, 2801-951 Russian Federation Kazan, Russian Federation, 420029 Kemerovo, Russian Federation, 650066 Moscow, Russian Federation, 123182 Omsk, Russian Federation, 644013 Penza, Russian Federation, 440071 South Africa Johannesburg, Gauteng, South Africa, 2013 Taiwan Taipei, Taiwan, 10002 Turkey Istanbul, Turkey, 34093 Collapse << |
NCT03517956 | Advanced or Metastatic Solid T... more >>umor Collapse << | Phase 1 | Recruiting | March 10, 2021 | - |
NCT02367040 | Lymphoma,Non-Hodgkin | Phase 3 | Recruiting | August 28, 2020 | - |
NCT02119221 | Healthy Volunteers | Phase 1 | Completed | - | Netherlands ... more >> Zuidlaren, Netherlands, 9471 GP Collapse << |
NCT03484819 | Recurrent Diffuse Large B-Cell... more >> Lymphoma Recurrent Primary Mediastinal (Thymic) Large B-Cell Cell Lymphoma Refractory Diffuse Large B-Cell Lymphoma Refractory Primary Mediastinal (Thymic) Large B-Cell Cell Lymphoma Collapse << | Phase 2 | Not yet recruiting | August 31, 2020 | - |
NCT02705859 | HER2 Positive Breast Cancer | Phase 1 | Recruiting | October 2020 | Ireland ... more >> St Vincent's University Hospital Recruiting Elm Park, Dublin 4, Ireland Contact: Jo Ballott +353 1 221 4000 Principal Investigator: Prof John Crown Beaumont University Hospital Recruiting Beaumont Road, Dublin 9, Ireland Contact: Derval Kehily +353 1 809 3000 Principal Investigator: Prof Bryan Hennessy University Hospital Galway Not yet recruiting Galway, Ireland Contact: Mary Byrne Contact +353 91 524 222 Principal Investigator: Dr Maccon Keane Collapse << |
NCT03655301 | Healthy Volunteers | Phase 1 | Active, not recruiting | January 18, 2019 | United States, Texas ... more >> Pharmaceutical Product Development, LLC Austin, Texas, United States, 78744 Collapse << |
NCT02631590 | Biliary Carcinoma ... more >> Gall Bladder Carcinoma Cholangiocarcinoma Gastrointestinal Tumor Collapse << | Phase 2 | Recruiting | December 2020 | United States, Florida ... more >> H. Lee Moffitt Cancer Center and Research Institute Recruiting Tampa, Florida, United States, 33612 Contact: Maria Martinez Jimenez 813-745-1946 maria.martinez@moffitt.org Contact: Richard D. Kim 813-745-1277 richard.kim@moffitt.org Principal Investigator: Richard D. Kim, M.D. Sub-Investigator: Rutika Mehta, M.D. Sub-Investigator: Dae Won Kim, M.D. Collapse << |
NCT02155582 | Non Hodgkin Lymphoma | Phase 1 | Completed | - | Belgium ... more >> Bruxelles - Brussel, Belgium, 1000 Bruxelles - Brussel, Belgium, 1200 Gent, Belgium, 9000 France Caen Cedex 5, France, 14076 Lille, France, 59037 Nice Cedex 2, France, 06102 Pierre Benite, France, 69495 United Kingdom Sutton, Surrey, United Kingdom, SM2 5PT London, United Kingdom, W1G 6AD Collapse << |
NCT03474744 | Marginal Zone Lymphoma | Phase 2 | Not yet recruiting | December 1, 2026 | - |
NCT03735628 | Non-small Cell Lung Cancer (NS... more >>CLC), Head and Neck Squamous Cell Carcinoma (HNSCC), Colorectal Cancer (CRC), Hepatocellular Carcinoma (HCC) Collapse << | Phase 1 Phase 2 | Recruiting | April 30, 2021 | United States, California ... more >> Sarcoma Oncology Center Not yet recruiting Santa Monica, California, United States, 90403 United States, Ohio Gabrail Cancer Center Recruiting Canton, Ohio, United States, 44718 United States, Rhode Island Rhode Island Hospital Not yet recruiting Providence, Rhode Island, United States, 02903-4900 Canada, Ontario Princess Margaret Cancer Centre Not yet recruiting Toronto, Ontario, Canada, M5G 1Z5 Collapse << |
NCT03502733 | Ann Arbor Stage III Lymphoma ... more >> Ann Arbor Stage IV Lymphoma Metastatic Malignant Solid Neoplasm Collapse << | Phase 1 | Recruiting | February 1, 2020 | United States, Maryland ... more >> National Cancer Institute Developmental Therapeutics Clinic Recruiting Bethesda, Maryland, United States, 20892 Contact: Site Public Contact 800-411-1222 Principal Investigator: Geraldine O'Sullivan Coyne National Institutes of Health Clinical Center Recruiting Bethesda, Maryland, United States, 20892 Contact: Site Public Contact 800-411-1222 Principal Investigator: Geraldine O'Sullivan Coyne United States, Texas M D Anderson Cancer Center Recruiting Houston, Texas, United States, 77030 Contact: Site Public Contact 877-312-3961 Principal Investigator: Timothy A. Yap Collapse << |
NCT02728258 | Endometrial Endometrioid Adeno... more >>carcinoma Endometrial Mixed Adenocarcinoma Endometrial Serous Adenocarcinoma Endometrial Undifferentiated Carcinoma Metastatic Endometrioid Adenocarcinoma PIK3CA Gene Mutation Recurrent Uterine Corpus Carcinoma Collapse << | Phase 2 | Suspended(Scheduled Interim Mo... more >>nitoring) Collapse << | - | - |
NCT02391116 | Diffuse, Large B-Cell, Lymphom... more >>a Collapse << | Phase 2 | Completed | - | - |
NCT02391116 | - | - | Completed | - | - |
NCT03581942 | Refractory/Recurrent Primary C... more >>entral Nervous System Lymphoma (PCNSL) Collapse << | Phase 1 Phase 2 | Recruiting | July 2021 | United States, New Jersey ... more >> Memoral Sloan Kettering Basking Ridge Recruiting Basking Ridge, New Jersey, United States, 07920 Contact: Christian Grommes, MD 212-639-4058 Memorial Sloan Kettering Monmouth Recruiting Middletown, New Jersey, United States, 07748 Contact: Christian Grommes, MD 212-639-4058 United States, New York Memorial Sloan Kettering Commack Recruiting Commack, New York, United States, 11725 Contact: Christian Grommes, MD 212-639-4058 Memorial Sloan Kettering Westchester Recruiting Harrison, New York, United States, 10604 Contact: Christian Grommes, MD 212-639-4058 Memorial Sloan Kettering Cancer Center Recruiting New York, New York, United States, 10065 Contact: Christian Grommes, MD 212-639-4058 Contact: Ingo Mellinghoff, MD 646-888-2766 Collapse << |
NCT03052933 | Mature T-Cell and NK-Cell Neop... more >>lasm Collapse << | Phase 1 Phase 2 | Recruiting | December 2021 | Korea, Republic of ... more >> Chonnam National University Hwasun Hospital Recruiting Hwasun-gun, Jeollanam-do, Korea, Republic of, 519-809 Contact: Deok-Hwan Yang, M.D. and Ph.D. 82-61-379-7636 drydh1685@gmail.com Contact: Kun-Hee Choi, Research Nurse 82-61-379-7717 iris9904@hanmail.net Collapse << |
NCT03711058 | Unresectable or Metastatic Mic... more >>rosatellite Stable (MSS) Solid Tumor Along With Microsatellite Stable (MSS) Colon Cancer Colon Cancer Collapse << | Phase 1 Phase 2 | Not yet recruiting | January 2022 | United States, Maryland ... more >> Sidney Kimmel Comprehensive Cancer Center Baltimore, Maryland, United States, 21231 Collapse << |
NCT02822482 | Carcinoma, Squamous Cell of He... more >>ad and Neck Collapse << | Phase 1 Phase 2 | Recruiting | June 2020 | France ... more >> Institut de Cancérologie de l'Ouest Recruiting Angers, France, 49933 Contact: Frédéric Rolland, MD frederic.rolland@ico.unicancer.fr Contact: Olivier Capitain, MD olivier.capitain@ico.unicancer.fr Centre Georges François Leclerc Not yet recruiting Dijon, France, 21079 Contact: Nicolas Isambert, MD nisambert@cgfl.fr Centre Oscar Lambret Not yet recruiting Lille, France, 59020 Contact: Nuria Kotecki, MD n-kotecki@o-lambret.fr Centre Léon Bérard Not yet recruiting Lyon, France, 69437 Contact: Jérôme Fayette, MD jerome.fayette@lyon.unicancer.fr Institut de Cancérologie de Lorraine Not yet recruiting Nancy, France, 54511 Contact: Marie-Christine Kaminsky, MD mc.kaminsky@nancy.unicancer.fr Centre Antoine Lacassagne Not yet recruiting Nice, France, 06189 Contact: Esma Saada-Bouzid, MD esma.saada-bouzid@nice.unicancer.fr Institut Curie Recruiting Paris, France, 75005 Contact: Christophe Le Tourneau, MD christophe.letourneau@curie.fr Contact: Marie Alt, MD marie.alt@curie.fr Collapse << |
NCT03498430 | Lymphoma, Non-Hodgkin | Phase 1 | Recruiting | September 3, 2019 | China ... more >> Beijing Cancer Hospital Recruiting Beijing, China, 100142 Collapse << |
NCT03586661 | Deleterious BRCA1 Gene Mutatio... more >>n Deleterious BRCA2 Gene Mutation Endometrial Adenocarcinoma High Grade Ovarian Serous Adenocarcinoma Primary Peritoneal High Grade Serous Adenocarcinoma Recurrent Endometrial Carcinoma Recurrent Fallopian Tube Carcinoma Recurrent Ovarian Carcinoma Recurrent Primary Peritoneal Carcinoma Collapse << | Phase 1 | Not yet recruiting | October 2020 | United States, Texas ... more >> M D Anderson Cancer Center Not yet recruiting Houston, Texas, United States, 77030 Contact: N. swestin@mdanderson.org Collapse << |
靶点 | Description | IC50 |
---|---|---|
PI3Kα | IC50:0.469nM | |
PI3Kβ | IC50:3.72nM |
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