400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / Cell Cycle / HSP / CH5138303
CAS No.: 959763-06-5
CH5138303 is an orally available Hsp90 inhibitor with Kd of 0.48 nM.
生物活性
实验方案
技术信息
| CAS号 | 959763-06-5 | 储存条件 |
|
|
| 分子式 | C19H18ClN5O2S | 运输 | 蓝冰 | |
| 分子量 | 415.90 | 别名 |
| Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
|---|
| HCT116 cells | - | Cytotoxicity assay | 4 days | Cytotoxicity against human HCT116 cells after 4 days by CCk-8 assay, IC50=0.098 μM | 24369839 |
| NCI-N87 cells | - | Cytotoxicity assay | 4 days | Cytotoxicity against human NCI-N87 cells after 4 days by CCk-8 assay, IC50=0.066 μM | 24369839 |
| NCI-N87 cells | 0.04 to 5 uM | Function assay | 24 h | Inhibition of Hsp90 in human NCI-N87 cells assessed as reduction in EGFR protein level at 0.04 to 5 uM after 24 hrs by Western blotting analysis | 24369839 |
联系我们
官方电话：400-920-2911
二维码
微信公众号 CSN官网
400-920-2911
sales@csnpharm.cn
tech@csnpharm.cn