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CAS No.: 1391712-60-9
Synonyms: CEP-37440
CEP-37440 is a potent and selective Dual FAK/ALK inhibitor with IC50 s of 2.3 nM (FAK) and 120 nM (ALK cellular IC50 in 75% human plasma).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01922752 | Solid Tumors | Phase 1 | Completed | - | United States, Illinois ... more >> Teva Investigational Site 10689 Chicago, Illinois, United States United States, Pennsylvania Teva Investigational Site 10687 Philadelphia, Pennsylvania, United States United States, Texas Teva Investigational Site 10686 San Antonio, Texas, United States Collapse << |
实验方案
技术信息
CAS号 | 1391712-60-9 | 储存条件 |
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分子式 | C30H38ClN7O3 | 运输 | 蓝冰 | |||
分子量 | 580.12 | 别名 | CEP-37440 | |||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01922752 | Solid Tumors | Phase 1 | Completed | - | United States, Illinois ... more >> Teva Investigational Site 10689 Chicago, Illinois, United States United States, Pennsylvania Teva Investigational Site 10687 Philadelphia, Pennsylvania, United States United States, Texas Teva Investigational Site 10686 San Antonio, Texas, United States Collapse << |
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