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CAS No.: 544417-40-5
Synonyms: BAY 68-4986
Capadenoson is an oral active, potent and selective adenosine A1 receptor agonist.
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生物活性
动物研究 | |||||||||||||||||||||||||||||
剂量 | Rat: 0.03 mg/kg - 0.3 mg/kg[4] (i.v.); 1 mg/kg, 2 mg/kg[5] (i.p.) | ||||||||||||||||||||||||||||
给药途径 | i.v., i.p. | ||||||||||||||||||||||||||||
动物药代数据 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00568945 | Atrial Fibrillation | Phase 2 | Completed | - | Germany ... more >> Erfurt, Thüringen, Germany, 99084 Collapse << |
NCT00518921 | Chronic Stable Angina | Phase 2 | Withdrawn | November 2008 | Czech Republic ... more >> Brno, Czech Republic, 656 91 Hodonin, Czech Republic, 695 26 Kromeriz, Czech Republic, 767 55 Olomouc, Czech Republic, 775 20 Ostrava, Czech Republic, 708 52 Plzen, Czech Republic, 30599 Praha 13, Czech Republic, 158 00 Praha 6, Czech Republic, 169 02 Hungary Balatonfured, Hungary, 8230 Kecskemet, Hungary, 6000 Miskolc, Hungary, 3526 Pecs, Hungary, 7624 Zalaegerszeg, Hungary, 8900 Israel Hadera, Israel, 38100 Rehovot, Israel, 76100 Safed, Israel, 13100 Italy Mestre, Venezia, Italy, 30174 Genova, Italy, 16132 Pavia, Italy, 27100 Trieste, Italy, 34100 Poland Bialystok, Poland, 15-276 Gdansk, Poland, 80-952 Gdynia, Poland, 81-519 Katowice, Poland, 40-635 Krakow, Poland, 30-501 Legnica, Poland, 59-220 Lodz, Poland, 91-347 Starogard Gdanski, Poland, 83-200 Szczecin, Poland, 70-111 Warszawa, Poland, 03-401 Wroclaw, Poland, 50-420 Wroclaw, Poland, 50-981 Slovakia Bratislava, Slovakia, 811 04 Bratislava, Slovakia, 813 69 Nitra, Slovakia, 949 01 Nove Zamky, Slovakia, 940 34 Collapse << |
实验方案
技术信息
CAS号 | 544417-40-5 | 储存条件 |
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分子式 | C25H18ClN5O2S2 | 运输 | 蓝冰 | |||||
分子量 | 520.03 | 别名 | BAY 68-4986 | |||||
溶解度 |
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动物实验配方 |