CAS No.: 57477-39-1
BRL 54443 Catalog No. CSN13853
Synonyms: BRL 54443
BRL 54443 is a selective agonist for 5-HT1E and 5-HT1F receptor with pEC50 values of 8.5 and 8.6.
| 规格 | 价格 | 促销价格 | 库存 | 数量 |
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纯度 & 质量文件
批次:
靶点选择性
生物活性
靶点 5-HT Receptor 1E
pKi:8.75-HT Receptor 1F
pKi:8.9- 描述
- 参考文献
- [1] Janssen P, Tack J, et al. Influence of 5-HT1 receptor agonists on feline stomach relaxation. Eur J Pharmacol. 2004 May 25;492(2-3):259-67.
- [2] McKune CM, Watts SW. Characterization of the serotonin receptor mediating contraction in the mouse thoracic aorta and signal pathway coupling. J Pharmacol Exp Ther. 2001 Apr;297(1):88-95.
- [3] Klein MT, Teitler M. Guinea pig hippocampal 5-HT(1E) receptors: a tool for selective drug development. J Neurochem. 2009 Apr;109(1):268-74.
- [4] Hisadome K, Smith MA, Choudhury AI, Claret M, Withers DJ, Ashford ML. 5-HT inhibition of rat insulin 2 promoter Cre recombinase transgene and proopiomelanocortin neuron excitability in the mouse arcuate nucleus. Neuroscience. 2009 Mar 3;159(1):83-93.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 57477-39-1 | 储存条件 |
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| 分子式 | C14H18N2O | 运输 | 蓝冰 | |||||||
| 分子量 | 230.31 | 别名 | BRL 54443 | |||||||
| 溶解度 |
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动物实验配方 |
