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CAS No.: 1802148-05-5
Synonyms: AZD7986;INS 1007
AZD7986 is a second generation reversible covalent, potent and selective DPP1 inhibitor potentially for the treatment of chronic obstructive pulmonary disease (COPD) with predicted human PK properties suitable for once daily human dosing.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02653872 | Healthy Subjects | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
NCT02653872 | - | - | Completed | - | - |
NCT02303574 | - | - | Completed | - | - |
实验方案
技术信息
CAS号 | 1802148-05-5 | 储存条件 |
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分子式 | C23H24N4O4 | 运输 | 蓝冰 | |||||
分子量 | 420.46 | 别名 | AZD7986;INS 1007 | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02653872 | Healthy Subjects | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
NCT02653872 | - | - | Completed | - | - |
NCT02303574 | - | - | Completed | - | - |
NCT02303574 | Safety, Pharmacokinetics, Phar... more >>macodynamics, Food Effect Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site Harrow, United Kingdom, HA1 3UJ Collapse << |
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