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CAS No.: 1197420-05-5
BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM. BMS-819881 also is selective and potent for CYP3A4 activity with an EC50 of 13 μM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00909766 | Obesity | Phase 1 Phase 2 | Completed | - | United States, Louisiana ... more >> Pennington Biomedical Research Center Baton Rouge, Louisiana, United States, 70808 Collapse << |
NCT00878020 | Obesity | Phase 1 | Completed | - | United States, Texas ... more >> Ppd Development, Lp Austin, Texas, United States, 78744 Collapse << |
实验方案
技术信息
CAS号 | 1197420-05-5 | 储存条件 |
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分子式 | C24H21ClN2O4S | 运输 | 蓝冰 | |
分子量 | 468.95 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00909766 | Obesity | Phase 1 Phase 2 | Completed | - | United States, Louisiana ... more >> Pennington Biomedical Research Center Baton Rouge, Louisiana, United States, 70808 Collapse << |
NCT00878020 | Obesity | Phase 1 | Completed | - | United States, Texas ... more >> Ppd Development, Lp Austin, Texas, United States, 78744 Collapse << |
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