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CAS No.: 2095432-75-8
Synonyms: Wnt Agonist 1;BML 284;CID 11210285
AMBMP HCl is a cell permeable Wnt signaling pathway activator, which induces β-catenin- and TCF-dependent transcriptional activity with EC50 of 0.7 μM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01358045 | Basal Cell Carcinoma | Phase 2 | Completed | - | Netherlands ... more >> Maastricht University Medical Center Maastricht, Limburg, Netherlands, 6202 AZ Collapse << |
NCT01878617 | Medulloblastoma | Phase 2 | Recruiting | December 2026 | - |
NCT00085202 | Brain and Central Nervous Syst... more >>em Tumors Collapse << | Phase 3 | Active, not recruiting | January 2023 | United States, North Carolina ... more >> Duke Comprehensive Cancer Center Durham, North Carolina, United States, 27710 United States, Pennsylvania Children's Hospital of Philadelphia Philadelphia, Pennsylvania, United States, 19104 United States, Tennessee St. Jude Children's Research Hospital Memphis, Tennessee, United States, 38105 United States, Texas Texas Children's Cancer Center and Hematology Service at Texas Children's Hospital Houston, Texas, United States, 77030-2399 Australia, New South Wales Sydney Children's Hospital Randwick, New South Wales, Australia, 2031 Children's Hospital at Westmead Westmead, New South Wales, Australia, 2145 Australia, Queensland Lady Cilento Children's Hospital, Brisbane Brisbane, Queensland, Australia, 4029 Australia, Victoria Royal Children's Hospital Parkville, Victoria, Australia, 3052 Canada, Ontario Hospital for Sick Children Toronto, Ontario, Canada, M5G 1X8 Collapse << |
实验方案
技术信息
CAS号 | 2095432-75-8 | 储存条件 |
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分子式 | C19H19ClN4O3 | 运输 | 蓝冰 | |||||||||
分子量 | 386.83 | 别名 | Wnt Agonist 1;BML 284;CID 11210285;AMBMP hydrochloride | |||||||||
溶解度 |
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动物实验配方 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01358045 | Basal Cell Carcinoma | Phase 2 | Completed | - | Netherlands ... more >> Maastricht University Medical Center Maastricht, Limburg, Netherlands, 6202 AZ Collapse << |
NCT01878617 | Medulloblastoma | Phase 2 | Recruiting | December 2026 | - |
NCT00085202 | Brain and Central Nervous Syst... more >>em Tumors Collapse << | Phase 3 | Active, not recruiting | January 2023 | United States, North Carolina ... more >> Duke Comprehensive Cancer Center Durham, North Carolina, United States, 27710 United States, Pennsylvania Children's Hospital of Philadelphia Philadelphia, Pennsylvania, United States, 19104 United States, Tennessee St. Jude Children's Research Hospital Memphis, Tennessee, United States, 38105 United States, Texas Texas Children's Cancer Center and Hematology Service at Texas Children's Hospital Houston, Texas, United States, 77030-2399 Australia, New South Wales Sydney Children's Hospital Randwick, New South Wales, Australia, 2031 Children's Hospital at Westmead Westmead, New South Wales, Australia, 2145 Australia, Queensland Lady Cilento Children's Hospital, Brisbane Brisbane, Queensland, Australia, 4029 Australia, Victoria Royal Children's Hospital Parkville, Victoria, Australia, 3052 Canada, Ontario Hospital for Sick Children Toronto, Ontario, Canada, M5G 1X8 Collapse << |
NCT00085202 | - | - | Active, not recruiting | - | - |
NCT02897700 | Breast Cancer | Phase 1 | Recruiting | December 2020 | China, Jiangxi ... more >> Ganzhou City People's Hospital Recruiting Ganzhou, Jiangxi, China, 341000 Contact: Xiao-Ming Zhong, M.D 86-18160779919 jxthrz@qq.com China, Jilin China-Japan Union Hospital, Jilin University Recruiting Changchun, Jilin, China, 130033 Contact: Xian-Ling Cong, M.D 86-0431-89876626 congxl888@hotmail.com China Shanghai 10th People's Hospital, Tongji University School of Medicine Recruiting Shanghai, China, 200072 Contact: Da Fu, Ph.D 86-15921527578 fu800da900@126.com Collapse << |
NCT02724579 | Medulloblastoma ... more >> Untreated Childhood Medulloblastoma Collapse << | Phase 2 | Recruiting | May 31, 2025 | - |
NCT02212574 | Medulloblastoma | Not Applicable | Recruiting | May 2022 | United States, Arizona ... more >> Phoenix Childrens Hospital Hematology/Oncology Recruiting Phoenix, Arizona, United States, 85016-7710 Contact: Michael Etzl, Dr 602-546-0920 metzl@phoenixchildrens.com United States, Colorado Children's Hospital Colorado Center for Cancer & Blood Disorders Recruiting Aurora, Colorado, United States, 80045 Contact: Kathleen Dorris, M.D., M.S. 720-777-6772 kathleen.dorris@childrenscolorado.org United States, Florida M D Anderson Cancer Center-Orlando Pediatric Hematology/Oncology Not yet recruiting Orlando, Florida, United States, 32806 Contact: Amy Smith, Dr 321-841-8588 amy.smith@orlandohealth.com All Children's Hospital Pediatric Hematology/Oncology Recruiting Saint Petersburg, Florida, United States, 33701 Contact: Stacie Stapleton, Dr 727-767-4176 Stacie.Stapleton@allkids.org United States, Georgia Children's Healthcare of Atlanta- Egleston Pediatric Neuro-Oncology Recruiting Atlanta, Georgia, United States, 30322 Contact: Tobey MacDonald, Dr 404-727-1447 tobey.macdonald@emory.edu United States, Illinois Ann and Robert H Lurie Children's Hospital of Chicago Hematology/Oncology Recruiting Chicago, Illinois, United States, 60611 Contact: Stewart Goldman, Dr 312-227-4844 sgoldman@northwestern.edu United States, Maryland Johns Hopkins University Recruiting Baltimore, Maryland, United States, 21287 Contact: Kenneth Cohen, MD, MBA 410-614-5055 kcohen@jhmi.edu Contact: Tammy Scott, RN 4140-614-5990 scottta@jhmi.edu United States, Massachusetts Dana-Farber Cancer Institute Recruiting Boston, Massachusetts, United States, 02215 Contact: Pratiti Bandopadhayay, MBBS, PhD United States, Missouri Washington University School of Medicine Pediatric Hematology/Oncology Recruiting Saint Louis, Missouri, United States, 63110 Contact: Joshua Rubin, Dr 314-454-6018 rubin_j@kids.wustl.edu United States, New Jersey Hackensack University Medical Center Recruiting Hackensack, New Jersey, United States, 07601 Contact: Derek Hanson, MD 551-996-5437 dhanson@hackensackumc.org United States, New York Memorial Sloan Kettering Cancer Center Recruiting New York, New York, United States, 10065 Contact: Kevin De Braganca, MD 212-639-3449 debragak@mskcc.org United States, North Carolina Duke University Medical Center Recruiting Durham, North Carolina, United States, 27705 Contact: David Ashley, MD, PhD david.ashley@duke.edu Principal Investigator: David Ashley, MD, PhD United States, Ohio Nationwide Children's Hospital Recruiting Columbus, Ohio, United States, 43205 Contact: Mohamed S AbdelBaki, MBBCh 614-722-3250 mohamed.abdelbaki@nationwidechildrens.org United States, Oregon Oregon Health and Science University Pediatric Hematology/Oncology Not yet recruiting Portland, Oregon, United States, 97239-3098 Contact: Kellie Nazemi, Dr 503-494-0714 nazemik@ohsu.edu United States, Washington Seattle Children's Hospital Hematology/Oncology Recruiting Seattle, Washington, United States, 98105 Contact: Sarah Leary, Dr 206-987-2106 sarah.leary@seattlechildrens.org United States, Wisconsin Childrens Hospital of Wisconsin (Medical College of Wisconsin) Recruiting Milwaukee, Wisconsin, United States, 53226 Contact: Jeffrey Knipstein, MD 414-955-4108 jknipstein@jhmi.edu Collapse << |
NCT03315702 | - | - | Active, not recruiting | October 31, 2017 | China, Shanghai ... more >> Department of Anesthesia, Shanghai Xinhua hospital Shanghai, Shanghai, China, 200082 Collapse << |
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