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CAS No.: 330942-05-7
Synonyms: PRT054021;MK-4448;PRT-021
Betrixaban is a highly potent, selective, and orally efficacious factor Xa inhibitor with IC50 of 1.2 nM (inhibition of Factor 10a).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03728166 | Venous Thromboembolism | Phase 4 | Not yet recruiting | February 1, 2021 | - |
NCT03397888 | Hepatic Impairment | Phase 1 | Completed | - | United States, Florida ... more >> Clinical Pharmacology of Miami Hialeah, Florida, United States, 33014 Collapse << |
NCT03613402 | - | - | Suspended(Due to slow enrollme... more >>nt.) Collapse << | January 2020 | United States, North Carolina ... more >> Durham Durham, North Carolina, United States, 27705 Collapse << |
实验方案
技术信息
CAS号 | 330942-05-7 | 储存条件 |
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分子式 | C23H22ClN5O3 | 运输 | 蓝冰 | |||||
分子量 | 451.91 | 别名 | PRT054021;MK-4448;PRT-021;MLN-1021;贝曲西班 | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03728166 | Venous Thromboembolism | Phase 4 | Not yet recruiting | February 1, 2021 | - |
NCT03397888 | Hepatic Impairment | Phase 1 | Completed | - | United States, Florida ... more >> Clinical Pharmacology of Miami Hialeah, Florida, United States, 33014 Collapse << |
NCT03613402 | - | - | Suspended(Due to slow enrollme... more >>nt.) Collapse << | January 2020 | United States, North Carolina ... more >> Durham Durham, North Carolina, United States, 27705 Collapse << |
NCT00375609 | Thromboembolism | Phase 2 | Completed | - | Canada, Quebec ... more >> Montreal General Hospital Montreal, Quebec, Canada, H3Y 3B8 Collapse << |
NCT00375609 | - | - | Completed | - | - |
NCT01229254 | - | - | Completed | - | - |
NCT03330457 | Bleeding | Phase 2 | Recruiting | September 2018 | United States, California ... more >> WCCT Global Recruiting Cypress, California, United States, 90630 Contact 714-252-0700 Collapse << |
NCT01765855 | Health Volunteers | Phase 1 | Completed | - | - |
NCT00742859 | - | - | Completed | - | - |
NCT00742859 | Atrial Fibrillation | Phase 2 | Completed | - | United States, California ... more >> Portola Investigational Site Anaheim, California, United States, 92801 United States, Colorado Portola Investigational Site Colorado Springs, Colorado, United States, 80909 United States, Florida Portola Investigational Site Melbourne, Florida, United States, 32901 Portola Investigational Site Miami, Florida, United States, 33173 Portola Investigational Site Ormond Beach, Florida, United States, 32174 Portola Investigational Site Pensacola, Florida, United States, 32501 Portola Investigational Site Port Charlotte, Florida, United States, 33952 United States, Illinois Portola Investigational Site Aurora, Illinois, United States, 60504 United States, Maine Portola Investigational Site Auburn, Maine, United States, 04210 United States, Maryland Portola Investigational Site Columbia, Maryland, United States, 21044 Portola Investigational Site Salisbury, Maryland, United States, 21804 Portola Investigational Site Towson, Maryland, United States, 21204 United States, Mississippi Portola Investigational Site Tupelo, Mississippi, United States, 38801 United States, Missouri Portola Investigational Site Saint Louis, Missouri, United States, 63110 United States, New York Portola Investigational Site Poughkeepsie, New York, United States, 12601 United States, Oregon Portola Investigational Site Hillsboro, Oregon, United States, 97123 United States, Pennsylvania Portola Investigational Site Wynnewood, Pennsylvania, United States, 19096 United States, South Dakota Portola Investigational Site Rapid City, South Dakota, United States, 57701 United States, Virginia Portola Investigational Site Norfolk, Virginia, United States, 23507 Canada, Quebec Portola Investigational Site Longueuil, Quebec, Canada Portola Investigational Site Montreal, Quebec, Canada Collapse << |
NCT01765868 | Healthy Subjects | Phase 1 | Completed | - | - |
NCT03346083 | VTE Prophylaxis | Phase 1 | Recruiting | April 2022 | Russian Federation ... more >> Children's Hospital of Tatarstan Republic Recruiting Kazan, Russian Federation Federal State Institution Recruiting Kemerovo, Russian Federation State Budgetary Institution Recruiting Nizhnii Novgorod, Russian Federation Federal State Budgetary Institution Recruiting Saint Petersburg, Russian Federation Collapse << |
NCT01229254 | Atrial Fibrillation ... more >> Atrial Flutter Collapse << | Phase 2 | Completed | - | - |
NCT00999336 | Renal Impairment | Phase 1 | Completed | - | Germany ... more >> APEX GmbH Munich, Germany Collapse << |
NCT01583218 | Venous Thromboembolism (VTE) | Phase 3 | Completed | - | - |
NCT01583218 | - | - | Completed | - | - |
NCT02596100 | Healthy | Phase 1 | Completed | - | - |
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