400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / Neuronal Signaling / Secretase / AZD3839
CAS No.: 1227163-84-9
Synonyms: AZD-3839 Free Base
AZD3839 is an inhibitor of BACE1 with IC50 of 23.6 uM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01348737 | Alzheimer's Disease ... more >> Safety Tolerability Blood Concentration Healthy Volunteers Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
实验方案
技术信息
CAS号 | 1227163-84-9 | 储存条件 |
|
|||||||
分子式 | C24H16F3N5 | 运输 | 蓝冰 | |||||||
分子量 | 431.41 | 别名 | AZD-3839 Free Base | |||||||
溶解度 |
|
动物实验配方 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
---|
CHO cells | - | Function assay | - | Inhibition of human ERG expressed in CHO cells by IonWorks assay, IC50=4.8 μM | 22924815 |
SH-SY5Y cells | - | Function assay | 16 h | Inhibition of BACE1 in human SH-SY5Y cells assessed as inhibition of sAPPbeta release after 16 hrs by immunoassay, IC50=0.0167 μM | 22924815 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01348737 | Alzheimer's Disease ... more >> Safety Tolerability Blood Concentration Healthy Volunteers Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网