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CAS No.: 878385-84-3
Synonyms: AZD5069
AZD 5069 is a selective and reversible antagonist of CXCR2 that can inhibit CXCL8 binding to CXCR2 with pIC50 of 9.1.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02499328 | Advanced Solid Tumors & Metast... more >>atic Squamous Cell Carcinoma of the Head and Neck Collapse << | Phase 1 Phase 2 | Recruiting | October 31, 2019 | - |
NCT01962935 | Chronic Obstructive Pulmonary ... more >>Disease (COPD). Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
NCT01989520 | Uncontrolled and Persistent As... more >>thma Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
实验方案
技术信息
CAS号 | 878385-84-3 | 储存条件 |
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分子式 | C18H22F2N4O5S2 | 运输 | 蓝冰 | |||||||
分子量 | 476.52 | 别名 | AZD5069 | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02499328 | Advanced Solid Tumors & Metast... more >>atic Squamous Cell Carcinoma of the Head and Neck Collapse << | Phase 1 Phase 2 | Recruiting | October 31, 2019 | - |
NCT01962935 | Chronic Obstructive Pulmonary ... more >>Disease (COPD). Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
NCT01989520 | Uncontrolled and Persistent As... more >>thma Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
NCT02583477 | Metastatic Pancreatic Ductal A... more >>denocarcinoma Collapse << | Phase 1 Phase 2 | Completed | - | United States, New York ... more >> Research Site Rochester, New York, United States, 14642 United Kingdom Research Site Cambridge, United Kingdom, CB2 0QQ Research Site Glasgow, United Kingdom, G12 0YN Research Site London, United Kingdom, SE1 9RY Research Site London, United Kingdom, W12 0NN Research Site Manchester, United Kingdom, M20 4BX Research Site Wirral, United Kingdom, CH63 4JY Collapse << |
NCT01255592 | Bronchiectasis ... more >> Lung Disease Respiratory Diseases Collapse << | Phase 2 | Completed | - | Czech Republic ... more >> Research Site Ostrava, Czech Republic Research Site Prague, Czech Republic Poland Research Site Krakow, Poland Research Site Lodz, Poland Research Site Warszawa, Poland United Kingdom Research Site Hull, East Yorkshire, United Kingdom Research Site Leicester, Leicestershire, United Kingdom Research Site Birmingham, Wstmid, United Kingdom Research Site Belfast, United Kingdom Research Site Bristol, United Kingdom Research Site Cambridge, United Kingdom Research Site London, United Kingdom Research Site Newcastle-upon-tyne, United Kingdom Research Site Salford, United Kingdom Research Site Wolverhampton, United Kingdom Collapse << |
NCT01233232 | - | - | Completed | - | - |
NCT01255592 | - | - | Completed | - | - |
NCT01890148 | Asthma | Phase 1 | Completed | - | Germany ... more >> Research Site Grosshansdorf, Germany Collapse << |
NCT01233232 | Scientific Terminology Chronic... more >> Obstructive Pulmonary Disease (COPD) Laymen Terminology Chronic Bronchitis and Emphysema Collapse << | Phase 2 | Completed | - | Bulgaria ... more >> Research Site Sofia, Bulgaria Germany Research Site Berlin, Germany Research Site GROßHANSDORF, Germany Hungary Research Site Debrecen, Hungary Research Site Pécs, Hungary Research Site Szeged, Hungary Research Site Százhalombatta, Hungary Ukraine Research Site Kyiv, Ukraine Collapse << |
NCT01890148 | - | - | Completed | - | - |
NCT00953888 | Healthy | Phase 1 | Completed | - | United Kingdom ... more >> Research Site Nottingham, United Kingdom Collapse << |
NCT01480739 | Chemokine Receptor 2 (CXCR2) A... more >>ntagonist Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> London, UK, United Kingdom Collapse << |
NCT01051505 | Healthy | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London Bridge, United Kingdom Collapse << |
NCT01100047 | Healthy | Phase 1 | Completed | - | United Kingdom ... more >> Research Site Croydon, United Kingdom Collapse << |
NCT01704495 | - | - | Completed | - | - |
NCT01704495 | Asthma | Phase 2 | Completed | - | - |
NCT01332903 | Healthy | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
NCT03177187 | Metastatic Castration Resistan... more >>t Prostate Cancer Collapse << | Phase 1 Phase 2 | Not yet recruiting | December 2020 | - |
NCT01735240 | Asthma, Pharm... more >>acokinetics, Cmax, Tmax, λz, AUC, Ketoconazole, Metabolite Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> London, United Kingdom Collapse << |
NCT01083238 | Chronic Obstructive Pulmonary ... more >>Disease Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Research Site London, United Kingdom Collapse << |
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