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CAS No.: 945595-80-2
Synonyms: AMG-900
AMG-900 is a potent and highly selective pan-Aurora kinases inhibitor for Aurora A/B/C with IC50 of 5 nM/4 nM /1 nM, and is > 10-fold selective for Aurora kinases than p38α, Tyk2, JNK2, Met and Tie2.
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00858377 | Advanced Malignancy ... more >> Advanced Solid Tumors Cancer Solid Tumors Tumors Collapse << | Phase 1 | Active, not recruiting | May 1, 2019 | United States, Arizona ... more >> Research Site Tucson, Arizona, United States, 85724 United States, California Research Site Los Angeles, California, United States, 90095 United States, Maryland Research Site Baltimore, Maryland, United States, 21231 United States, Nevada Research Site Las Vegas, Nevada, United States, 89148 United States, New Mexico Research Site Albuquerque, New Mexico, United States, 87131 Australia, South Australia Research Site Kurralta Park, South Australia, Australia, 5037 Australia, Victoria Research Site Bentleigh East, Victoria, Australia, 3165 Research Site Parkville, Victoria, Australia, 3050 Collapse << |
NCT01380756 | Cancer Hemato... more >>logic Malignancies Leukemia Myeloid Leukemia Collapse << | Phase 1 | Completed | - | United States, New York ... more >> Research Site Stony Brook, New York, United States, 11794 United States, Ohio Research Site Cleveland, Ohio, United States, 44195 United States, Texas Research Site Houston, Texas, United States, 77030 Collapse << |
实验方案
技术信息
CAS号 | 945595-80-2 | 储存条件 |
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分子式 | C28H21N7OS | 运输 | 蓝冰 | |||||||||
分子量 | 503.58 | 别名 | AMG-900 | |||||||||
溶解度 |
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动物实验配方 |
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