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CAS No.: 1797989-42-4
Synonyms: CHIR-99021 monohydrochloride;CT99021 monohydrochloride;CHIR-99021 HCl
CHIR-99021 HCl is HCl of CHIR-99021, which is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM and shows greater than 500-fold selectivity for GSK-3 versus its closest homologs Cdc2 and ERK2.
生物活性
实验方案
技术信息
CAS号 | 1797989-42-4 | 储存条件 |
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分子式 | C22H19Cl3N8 | 运输 | 蓝冰 | |||||||||
分子量 | 501.80 | 别名 | CHIR-99021 monohydrochloride;CT99021 monohydrochloride;CHIR-99021 HCl;CHIR-911;CT- 99021;CHIR-73911;GSK 3 inhibitor XVI;GSK 3IXV | |||||||||
溶解度 |
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动物实验配方 |
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Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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22RV1 | - | Growth Inhibition Assay | - | IC50=197.424 μM | SANGER |
23132-87 | - | Growth Inhibition Assay | - | IC50=93.168 μM | SANGER |
3T3-L1 | 3 μM | Function Assay | 4 h | Inhibits preadipocyte differentiation | 12055200 |
5637 | - | Growth Inhibition Assay | - | IC50=233.003 μM | SANGER |
639-V | - | Growth Inhibition Assay | - | IC50=148.705 μM | SANGER |
647-V | - | Growth Inhibition Assay | - | IC50=314.673 μM | SANGER |
697 | - | Growth Inhibition Assay | - | IC50=54.1555 μM | SANGER |
769-P | - | Growth Inhibition Assay | - | IC50=0.58499 μM | SANGER |
786-0 | - | Growth Inhibition Assay | - | IC50=113.453 μM | SANGER |
8305C | - | Growth Inhibition Assay | - | IC50=18.5305 μM | SANGER |
8505C | - | Growth Inhibition Assay | - | IC50=35.9294 μM | SANGER |
8-MG-BA | - | Growth Inhibition Assay | - | IC50=76.1096 μM | SANGER |
A101D | - | Growth Inhibition Assay | - | IC50=19.243 μM | SANGER |
A172 | - | Growth Inhibition Assay | - | IC50=3.75498 μM | SANGER |
A204 | - | Growth Inhibition Assay | - | IC50=29.6828 μM | SANGER |
A2058 | - | Growth Inhibition Assay | - | IC50=95.4617 μM | SANGER |
A253 | - | Growth Inhibition Assay | - | IC50=110.479 μM | SANGER |
A2780 | - | Growth Inhibition Assay | - | IC50=192.891 μM | SANGER |
A375 | - | Growth Inhibition Assay | - | IC50=54.8059 μM | SANGER |
A388 | - | Growth Inhibition Assay | - | IC50=312.022 μM | SANGER |
A3-KAW | - | Growth Inhibition Assay | - | IC50=460.841 μM | SANGER |
A427 | - | Growth Inhibition Assay | - | IC50=184.631 μM | SANGER |
A431 | - | Growth Inhibition Assay | - | IC50=211.299 μM | SANGER |
A498 | - | Growth Inhibition Assay | - | IC50=1.30469 μM | SANGER |
A4-Fuk | - | Growth Inhibition Assay | - | IC50=454.507 μM | SANGER |
A549 | 5 µM | Apoptosis Assay | 24 h | Increases cell apoptosis | 24367688 |
A673 | - | Growth Inhibition Assay | - | IC50=267.025 μM | SANGER |
A704 | - | Growth Inhibition Assay | - | IC50=3.0812 μM | SANGER |
ABC-1 | - | Growth Inhibition Assay | - | IC50=291.069 μM | SANGER |
ACHN | - | Growth Inhibition Assay | - | IC50=9.30546 μM | SANGER |
ACN | - | Growth Inhibition Assay | - | IC50=59.1587 μM | SANGER |
AGS | - | Growth Inhibition Assay | - | IC50=222.523 μM | SANGER |
ALL-PO | - | Growth Inhibition Assay | - | IC50=4.83858 μM | SANGER |
AM-38 | - | Growth Inhibition Assay | - | IC50=438.54 μM | SANGER |
AN3-CA | - | Growth Inhibition Assay | - | IC50=64.3035 μM | SANGER |
ARH-77 | - | Growth Inhibition Assay | - | IC50=337.32 μM | SANGER |
AsPC-1 | - | Growth Inhibition Assay | - | IC50=152.764 μM | SANGER |
ATN-1 | - | Growth Inhibition Assay | - | IC50=117.828 μM | SANGER |
AU565 | - | Growth Inhibition Assay | - | IC50=163.64 μM | SANGER |
BB30-HNC | - | Growth Inhibition Assay | - | IC50=134.116 μM | SANGER |
BB49-HNC | - | Growth Inhibition Assay | - | IC50=147.404 μM | SANGER |
BB65-RCC | - | Growth Inhibition Assay | - | IC50=6.53195 μM | SANGER |
BC-1 | - | Growth Inhibition Assay | - | IC50=220.799 μM | SANGER |
BC-3 | - | Growth Inhibition Assay | - | IC50=805.203 μM | SANGER |
BCPAP | - | Growth Inhibition Assay | - | IC50=1.66898 μM | SANGER |
BE-13 | - | Growth Inhibition Assay | - | IC50=41.4473 μM | SANGER |
Becker | - | Growth Inhibition Assay | - | IC50=20.1777 μM | SANGER |
BEN | - | Growth Inhibition Assay | - | IC50=276.461 μM | SANGER |
BFTC-905 | - | Growth Inhibition Assay | - | IC50=84.0172 μM | SANGER |
BFTC-909 | - | Growth Inhibition Assay | - | IC50=243.118 μM | SANGER |
BHT-101 | - | Growth Inhibition Assay | - | IC50=140.208 μM | SANGER |
BHY | - | Growth Inhibition Assay | - | IC50=323.175 μM | SANGER |
BL-41 | - | Growth Inhibition Assay | - | IC50=5.81266 μM | SANGER |
BL-70 | - | Growth Inhibition Assay | - | IC50=439.429 μM | SANGER |
BOKU | - | Growth Inhibition Assay | - | IC50=92.6957 μM | SANGER |
BPH-1 | - | Growth Inhibition Assay | - | IC50=21.7035 μM | SANGER |
BT-20 | - | Growth Inhibition Assay | - | IC50=210.986 μM | SANGER |
BT-474 | - | Growth Inhibition Assay | - | IC50=332.418 μM | SANGER |
BV-173 | - | Growth Inhibition Assay | - | IC50=57.5142 μM | SANGER |
BxPC-3 | - | Growth Inhibition Assay | - | IC50=4.70391 μM | SANGER |
C2BBe1 | - | Growth Inhibition Assay | - | IC50=300.691 μM | SANGER |
C32 | - | Growth Inhibition Assay | - | IC50=28.0826 μM | SANGER |
C-33-A | - | Growth Inhibition Assay | - | IC50=90.54 μM | SANGER |
C3A | - | Growth Inhibition Assay | - | IC50=215.575 μM | SANGER |
C-4-II | - | Growth Inhibition Assay | - | IC50=69.3607 μM | SANGER |
C8166 | - | Growth Inhibition Assay | - | IC50=13.2318 μM | SANGER |
CA46 | - | Growth Inhibition Assay | - | IC50=504.407 μM | SANGER |
Ca9-22 | - | Growth Inhibition Assay | - | IC50=164.321 μM | SANGER |
CAKI-1 | - | Growth Inhibition Assay | - | IC50=30.2656 μM | SANGER |
CAL-120 | - | Growth Inhibition Assay | - | IC50=155.821 μM | SANGER |
CAL-12T | - | Growth Inhibition Assay | - | IC50=268.366 μM | SANGER |
CAL-148 | - | Growth Inhibition Assay | - | IC50=565.089 μM | SANGER |
CAL-27 | - | Growth Inhibition Assay | - | IC50=253.485 μM | SANGER |
CAL-33 | - | Growth Inhibition Assay | - | IC50=93.0601 μM | SANGER |
CAL-39 | - | Growth Inhibition Assay | - | IC50=260.272 μM | SANGER |
CAL-51 | - | Growth Inhibition Assay | - | IC50=321.403 μM | SANGER |
CAL-54 | - | Growth Inhibition Assay | - | IC50=345.879 μM | SANGER |
CAL-62 | - | Growth Inhibition Assay | - | IC50=162.613 μM | SANGER |
CAL-72 | - | Growth Inhibition Assay | - | IC50=8.76113 μM | SANGER |
CAL-85-1 | - | Growth Inhibition Assay | - | IC50=6.60936 μM | SANGER |
Calu-1 | - | Growth Inhibition Assay | - | IC50=154.003 μM | SANGER |
Calu-3 | - | Growth Inhibition Assay | - | IC50=168.311 μM | SANGER |
Calu-6 | - | Growth Inhibition Assay | - | IC50=116.798 μM | SANGER |
CAMA-1 | - | Growth Inhibition Assay | - | IC50=278.279 μM | SANGER |
Caov-3 | - | Growth Inhibition Assay | - | IC50=149.714 μM | SANGER |
Caov-4 | - | Growth Inhibition Assay | - | IC50=95.685 μM | SANGER |
CAPAN-1 | - | Growth Inhibition Assay | - | IC50=187.453 μM | SANGER |
Capan-2 | - | Growth Inhibition Assay | - | IC50=133.975 μM | SANGER |
CaR-1 | - | Growth Inhibition Assay | - | IC50=221.251 μM | SANGER |
CAS-1 | - | Growth Inhibition Assay | - | IC50=31.7665 μM | SANGER |
Ca-Ski | - | Growth Inhibition Assay | - | IC50=138.831 μM | SANGER |
CCF-STTG1 | - | Growth Inhibition Assay | - | IC50=143.334 μM | SANGER |
CCRF-CEM | - | Growth Inhibition Assay | - | IC50=16.6702 μM | SANGER |
CESS | - | Growth Inhibition Assay | - | IC50=52.145 μM | SANGER |
CGTH-W-1 | - | Growth Inhibition Assay | - | IC50=6.417 μM | SANGER |
ChaGo-K-1 | - | Growth Inhibition Assay | - | IC50=363.924 μM | SANGER |
CHL-1 | - | Growth Inhibition Assay | - | IC50=228.13 μM | SANGER |
CHP-126 | - | Growth Inhibition Assay | - | IC50=53.5169 μM | SANGER |
CHP-212 | - | Growth Inhibition Assay | - | IC50=163.626 μM | SANGER |
CMK | - | Growth Inhibition Assay | - | IC50=38.4162 μM | SANGER |
COLO-205 | - | Growth Inhibition Assay | - | IC50=9.43821 μM | SANGER |
COLO-320-HSR | - | Growth Inhibition Assay | - | IC50=551.35 μM | SANGER |
COLO-668 | - | Growth Inhibition Assay | - | IC50=193.157 μM | SANGER |
COLO-678 | - | Growth Inhibition Assay | - | IC50=357.863 μM | SANGER |
COLO-679 | - | Growth Inhibition Assay | - | IC50=200.859 μM | SANGER |
COLO-680N | - | Growth Inhibition Assay | - | IC50=302.893 μM | SANGER |
COLO-684 | - | Growth Inhibition Assay | - | IC50=448.888 μM | SANGER |
COLO-741 | - | Growth Inhibition Assay | - | IC50=177.561 μM | SANGER |
COLO-792 | - | Growth Inhibition Assay | - | IC50=27.7728 μM | SANGER |
COLO-800 | - | Growth Inhibition Assay | - | IC50=45.5898 μM | SANGER |
COLO-824 | - | Growth Inhibition Assay | - | IC50=53.6976 μM | SANGER |
COLO-829 | - | Growth Inhibition Assay | - | IC50=2.7654 μM | SANGER |
COR-L105 | - | Growth Inhibition Assay | - | IC50=48.973 μM | SANGER |
COR-L23 | - | Growth Inhibition Assay | - | IC50=250.412 μM | SANGER |
COR-L279 | - | Growth Inhibition Assay | - | IC50=464.847 μM | SANGER |
COR-L88 | - | Growth Inhibition Assay | - | IC50=383.677 μM | SANGER |
CP50-MEL-B | - | Growth Inhibition Assay | - | IC50=134.2 μM | SANGER |
CP66-MEL | - | Growth Inhibition Assay | - | IC50=168.415 μM | SANGER |
CPC-N | - | Growth Inhibition Assay | - | IC50=502.063 μM | SANGER |
CTB-1 | - | Growth Inhibition Assay | - | IC50=132.897 μM | SANGER |
CTV-1 | - | Growth Inhibition Assay | - | IC50=9.43894 μM | SANGER |
CW-2 | - | Growth Inhibition Assay | - | IC50=356.529 μM | SANGER |
D-247MG | - | Growth Inhibition Assay | - | IC50=0.94852 μM | SANGER |
D-263MG | - | Growth Inhibition Assay | - | IC50=108.961 μM | SANGER |
D-283MED | - | Growth Inhibition Assay | - | IC50=488.924 μM | SANGER |
D-336MG | - | Growth Inhibition Assay | - | IC50=0.8462 μM | SANGER |
D-392MG | - | Growth Inhibition Assay | - | IC50=5.49145 μM | SANGER |
D-502MG | - | Growth Inhibition Assay | - | IC50=345.812 μM | SANGER |
D-542MG | - | Growth Inhibition Assay | - | IC50=47.4589 μM | SANGER |
Daoy | - | Growth Inhibition Assay | - | IC50=169.891 μM | SANGER |
Daudi | - | Growth Inhibition Assay | - | IC50=17.6149 μM | SANGER |
DB | - | Growth Inhibition Assay | - | IC50=51.9855 μM | SANGER |
DBTRG-05MG | - | Growth Inhibition Assay | - | IC50=9.7777 μM | SANGER |
DEL | - | Growth Inhibition Assay | - | IC50=700.838 μM | SANGER |
Detroit562 | - | Growth Inhibition Assay | - | IC50=141.466 μM | SANGER |
DG-75 | - | Growth Inhibition Assay | - | IC50=156.694 μM | SANGER |
DJM-1 | - | Growth Inhibition Assay | - | IC50=209.897 μM | SANGER |
DK-MG | - | Growth Inhibition Assay | - | IC50=155.183 μM | SANGER |
DMS-114 | - | Growth Inhibition Assay | - | IC50=147.441 μM | SANGER |
DMS-153 | - | Growth Inhibition Assay | - | IC50=217.836 μM | SANGER |
DMS-273 | - | Growth Inhibition Assay | - | IC50=115.617 μM | SANGER |
DMS-53 | - | Growth Inhibition Assay | - | IC50=358.711 μM | SANGER |
DMS-79 | - | Growth Inhibition Assay | - | IC50=449.68 μM | SANGER |
DN3 | 10 μM | Function Assay | 96 h | Increases cell development and proliferation | 23526989 |
DOHH-2 | - | Growth Inhibition Assay | - | IC50=346.65 μM | SANGER |
DOK | - | Growth Inhibition Assay | - | IC50=184.643 μM | SANGER |
DoTc2-4510 | - | Growth Inhibition Assay | - | IC50=56.6057 μM | SANGER |
DSH1 | - | Growth Inhibition Assay | - | IC50=13.3879 μM | SANGER |
DU-145 | - | Growth Inhibition Assay | - | IC50=109.945 μM | SANGER |
DU-4475 | - | Growth Inhibition Assay | - | IC50=511.101 μM | SANGER |
DV-90 | - | Growth Inhibition Assay | - | IC50=55.8917 μM | SANGER |
EB2 | - | Growth Inhibition Assay | - | IC50=241.907 μM | SANGER |
EB-3 | - | Growth Inhibition Assay | - | IC50=127.013 μM | SANGER |
ECC12 | - | Growth Inhibition Assay | - | IC50=310.254 μM | SANGER |
ECC4 | - | Growth Inhibition Assay | - | IC50=408.458 μM | SANGER |
EC-GI-10 | - | Growth Inhibition Assay | - | IC50=502.169 μM | SANGER |
EFE-184 | - | Growth Inhibition Assay | - | IC50=35.917 μM | SANGER |
EFM-19 | - | Growth Inhibition Assay | - | IC50=9.75566 μM | SANGER |
EFO-21 | - | Growth Inhibition Assay | - | IC50=165.45 μM | SANGER |
EFO-27 | - | Growth Inhibition Assay | - | IC50=160.584 μM | SANGER |
EGI-1 | - | Growth Inhibition Assay | - | IC50=204.833 μM | SANGER |
EHEB | - | Growth Inhibition Assay | - | IC50=507.208 μM | SANGER |
EKVX | - | Growth Inhibition Assay | - | IC50=61.4958 μM | SANGER |
EM-2 | - | Growth Inhibition Assay | - | IC50=18.6248 μM | SANGER |
embryonic stem cells (ESC) | 3 µM | Function Assay | 11 d | Promotes self-renewal of naïve-type mouse embryonic stem cells (ESC) | 23843312 |
Endothelial cell(EC) | 3 μM | Function Assay | - | Promotes endothelial cell (EC) differentiation | 22052006 |
EoL-1- | - | Growth Inhibition Assay | - | IC50=21.8385 μM | SANGER |
ES1 | - | Growth Inhibition Assay | - | IC50=312.189 μM | SANGER |
ES3 | - | Growth Inhibition Assay | - | IC50=270.358 μM | SANGER |
ES4 | - | Growth Inhibition Assay | - | IC50=159.396 μM | SANGER |
ES5 | - | Growth Inhibition Assay | - | IC50=245.038 μM | SANGER |
ES6 | - | Growth Inhibition Assay | - | IC50=55.8899 μM | SANGER |
ES7 | - | Growth Inhibition Assay | - | IC50=214.878 μM | SANGER |
ES8 | - | Growth Inhibition Assay | - | IC50=27.7814 μM | SANGER |
ES-CCE | 10 μM | Cytotoxic Assay | 3 d | Induces moderate cytotoxicity | 24779365 |
ES-CCE | 5 μM | Function Assay | 3 d | Strongly induces the activity of Wnt/beta-catenin pathway | 24779365 |
ES-D3 | 10 μM | Cytotoxic Assay | 3 d | Induces moderate cytotoxicity with IC50 of 4.9 μM | 24779365 |
ES-D3 | 5 μM | Function Assay | 3 d | Strongly induces the activity of Wnt/beta-catenin pathway | 24779365 |
ESS-1 | - | Growth Inhibition Assay | - | IC50=44.2062 μM | SANGER |
ETK-1 | - | Growth Inhibition Assay | - | IC50=190.181 μM | SANGER |
EVSA-T | - | Growth Inhibition Assay | - | IC50=543.684 μM | SANGER |
EW-1 | - | Growth Inhibition Assay | - | IC50=452.888 μM | SANGER |
EW-11 | - | Growth Inhibition Assay | - | IC50=552.399 μM | SANGER |
EW-13 | - | Growth Inhibition Assay | - | IC50=322.424 μM | SANGER |
EW-16 | - | Growth Inhibition Assay | - | IC50=71.7415 μM | SANGER |
EW-18 | - | Growth Inhibition Assay | - | IC50=210.763 μM | SANGER |
EW-24 | - | Growth Inhibition Assay | - | IC50=320.07 μM | SANGER |
EW-3 | - | Growth Inhibition Assay | - | IC50=176.555 μM | SANGER |
EW-7 | - | Growth Inhibition Assay | - | IC50=285.232 μM | SANGER |
FADU | - | Growth Inhibition Assay | - | IC50=403.083 μM | SANGER |
FTC-133 | - | Growth Inhibition Assay | - | IC50=108.488 μM | SANGER |
G-361 | - | Growth Inhibition Assay | - | IC50=7.46561 μM | SANGER |
G-401 | - | Growth Inhibition Assay | - | IC50=145.835 μM | SANGER |
G-402 | - | Growth Inhibition Assay | - | IC50=135.295 μM | SANGER |
GAK | - | Growth Inhibition Assay | - | IC50=151.374 μM | SANGER |
GAMG | - | Growth Inhibition Assay | - | IC50=148.247 μM | SANGER |
GB-1 | - | Growth Inhibition Assay | - | IC50=235.177 μM | SANGER |
GCIY | - | Growth Inhibition Assay | - | IC50=147.797 μM | SANGER |
GCT | - | Growth Inhibition Assay | - | IC50=0.30672 μM | SANGER |
GDM-1 | - | Growth Inhibition Assay | - | IC50=151.135 μM | SANGER |
GI-1 | - | Growth Inhibition Assay | - | IC50=22.7841 μM | SANGER |
GI-ME-N | - | Growth Inhibition Assay | - | IC50=181.672 μM | SANGER |
GMS-10 | - | Growth Inhibition Assay | - | IC50=287.183 μM | SANGER |
GOTO | - | Growth Inhibition Assay | - | IC50=390.641 μM | SANGER |
GP5d | - | Growth Inhibition Assay | - | IC50=242.616 μM | SANGER |
GR-ST | - | Growth Inhibition Assay | - | IC50=410.497 μM | SANGER |
GT3TKB | - | Growth Inhibition Assay | - | IC50=338.412 μM | SANGER |
H157 | 5 µM | Growth Inhibition Assay | 24 h | Promotes cell proliferation | 24367688 |
H157 | 5 µM | Apoptosis Assay | 24 h | Does not significantly affect apoptosis | 24367688 |
H4 | - | Growth Inhibition Assay | - | IC50=45.3296 μM | SANGER |
H460 | 5 µM | Growth Inhibition Assay | 24 h | Promotes cell proliferation | 24367688 |
H460 | 5 µM | Apoptosis Assay | 24 h | Attenuates cell apoptosis | 24367688 |
H4IIE | 10 μM | Function Assay | 24 h | Regulates β-catenin activity and TIRE containing promoter activity | 15350195 |
HAL-01 | - | Growth Inhibition Assay | - | IC50=122.499 μM | SANGER |
HC-1 | - | Growth Inhibition Assay | - | IC50=290.602 μM | SANGER |
HCC1143 | - | Growth Inhibition Assay | - | IC50=32.7979 μM | SANGER |
HCC1187 | - | Growth Inhibition Assay | - | IC50=20.3589 μM | SANGER |
HCC1395 | - | Growth Inhibition Assay | - | IC50=1.78273 μM | SANGER |
HCC1419 | - | Growth Inhibition Assay | - | IC50=156.077 μM | SANGER |
HCC1569 | - | Growth Inhibition Assay | - | IC50=3.48305 μM | SANGER |
HCC1599 | - | Growth Inhibition Assay | - | IC50=117.156 μM | SANGER |
HCC1806 | - | Growth Inhibition Assay | - | IC50=71.4587 μM | SANGER |
HCC1937 | - | Growth Inhibition Assay | - | IC50=224.389 μM | SANGER |
HCC1954 | - | Growth Inhibition Assay | - | IC50=323.582 μM | SANGER |
HCC2157 | - | Growth Inhibition Assay | - | IC50=378.161 μM | SANGER |
HCC2218 | - | Growth Inhibition Assay | - | IC50=40.5849 μM | SANGER |
HCC2998 | - | Growth Inhibition Assay | - | IC50=48.2982 μM | SANGER |
HCC38 | - | Growth Inhibition Assay | - | IC50=157.369 μM | SANGER |
HCC70 | - | Growth Inhibition Assay | - | IC50=159.242 μM | SANGER |
HCE-4 | - | Growth Inhibition Assay | - | IC50=190.992 μM | SANGER |
HCE-T | - | Growth Inhibition Assay | - | IC50=80.1588 μM | SANGER |
HCT-116 | - | Growth Inhibition Assay | - | IC50=43.2099 μM | SANGER |
HCT-15 | - | Growth Inhibition Assay | - | IC50=110.661 μM | SANGER |
HDLM-2 | - | Growth Inhibition Assay | - | IC50=480.869 μM | SANGER |
HD-MY-Z | - | Growth Inhibition Assay | - | IC50=321.409 μM | SANGER |
HEC-1 | - | Growth Inhibition Assay | - | IC50=129.198 μM | SANGER |
HEL | - | Growth Inhibition Assay | - | IC50=11.6579 μM | SANGER |
HGC-27 | - | Growth Inhibition Assay | - | IC50=195.538 μM | SANGER |
HH | - | Growth Inhibition Assay | - | IC50=173.848 μM | SANGER |
hiPSC-NPs | 3 μM | Growth Inhibition Assay | 72 h | Increases cell proliferation | 22642687 |
HL-60 | - | Growth Inhibition Assay | - | IC50=522.924 μM | SANGER |
HLE | - | Growth Inhibition Assay | - | IC50=301.818 μM | SANGER |
HMC1.2 | 30 μM | Growth Inhibition Assay | 72 h | Reduces cell survival | 22039301 |
HMV-II | - | Growth Inhibition Assay | - | IC50=24.2163 μM | SANGER |
HN | - | Growth Inhibition Assay | - | IC50=242.991 μM | SANGER |
HO-1-N-1 | - | Growth Inhibition Assay | - | IC50=212.894 μM | SANGER |
HOP-62 | - | Growth Inhibition Assay | - | IC50=3.36054 μM | SANGER |
HOP-92 | - | Growth Inhibition Assay | - | IC50=108.475 μM | SANGER |
HOS | - | Growth Inhibition Assay | - | IC50=218.9 μM | SANGER |
HPAF-II | - | Growth Inhibition Assay | - | IC50=209.671 μM | SANGER |
Hs-578-T | - | Growth Inhibition Assay | - | IC50=70.3 μM | SANGER |
HSC-2 | - | Growth Inhibition Assay | - | IC50=258.584 μM | SANGER |
HSC-3 | - | Growth Inhibition Assay | - | IC50=77.0282 μM | SANGER |
HSC-4 | - | Growth Inhibition Assay | - | IC50=539.293 μM | SANGER |
HT | - | Growth Inhibition Assay | - | IC50=622.785 μM | SANGER |
HT-1080 | - | Growth Inhibition Assay | - | IC50=132.204 μM | SANGER |
HT-1197 | - | Growth Inhibition Assay | - | IC50=292.879 μM | SANGER |
HT-1376 | - | Growth Inhibition Assay | - | IC50=59.0921 μM | SANGER |
HT-144 | - | Growth Inhibition Assay | - | IC50=38.2575 μM | SANGER |
HT-29 | - | Growth Inhibition Assay | - | IC50=122.778 μM | SANGER |
HT-3 | - | Growth Inhibition Assay | - | IC50=10.6179 μM | SANGER |
HT55 | - | Growth Inhibition Assay | - | IC50=199.192 μM | SANGER |
HTC-C3 | - | Growth Inhibition Assay | - | IC50=145.075 μM | SANGER |
HuCCT1 | - | Growth Inhibition Assay | - | IC50=67.0374 μM | SANGER |
HuH-7 | - | Growth Inhibition Assay | - | IC50=260.996 μM | SANGER |
HuO-3N1 | - | Growth Inhibition Assay | - | IC50=172.273 μM | SANGER |
HuO9 | - | Growth Inhibition Assay | - | IC50=337.47 μM | SANGER |
HuP-T3 | - | Growth Inhibition Assay | - | IC50=292.146 μM | SANGER |
HuP-T4 | - | Growth Inhibition Assay | - | IC50=121.55 μM | SANGER |
HUTU-80 | - | Growth Inhibition Assay | - | IC50=171.032 μM | SANGER |
IA-LM | - | Growth Inhibition Assay | - | IC50=197.822 μM | SANGER |
IGR-1 | - | Growth Inhibition Assay | - | IC50=99.3119 μM | SANGER |
IGROV-1 | - | Growth Inhibition Assay | - | IC50=35.3416 μM | SANGER |
IM-9 | - | Growth Inhibition Assay | - | IC50=651.541 μM | SANGER |
IMR-5 | - | Growth Inhibition Assay | - | IC50=315.38 μM | SANGER |
INS-1E | 2.5 μM | Function Assay | 24 h | Induces a reduction of NP1 overexpression | 22427704 |
insulin receptor–expressing CHO-IR | 500 nM | Function Assay | 30 min | Activates Glycogen Synthase (GS) | 12606497 |
IPC-298 | - | Growth Inhibition Assay | - | IC50=242.072 μM | SANGER |
IST-MEL1 | - | Growth Inhibition Assay | - | IC50=42.6938 μM | SANGER |
IST-MES1 | - | Growth Inhibition Assay | - | IC50=29.7092 μM | SANGER |
IST-SL1 | - | Growth Inhibition Assay | - | IC50=394.406 μM | SANGER |
IST-SL2 | - | Growth Inhibition Assay | - | IC50=372.926 μM | SANGER |
J82 | - | Growth Inhibition Assay | - | IC50=93.7811 μM | SANGER |
JAR | - | Growth Inhibition Assay | - | IC50=474.788 μM | SANGER |
JEG-3 | - | Growth Inhibition Assay | - | IC50=134.359 μM | SANGER |
JiyoyeP-2003 | - | Growth Inhibition Assay | - | IC50=29.6719 μM | SANGER |
J-RT3-T3-5 | - | Growth Inhibition Assay | - | IC50=313.521 μM | SANGER |
JVM-2 | - | Growth Inhibition Assay | - | IC50=167.451 μM | SANGER |
JVM-3 | - | Growth Inhibition Assay | - | IC50=198.419 μM | SANGER |
K052 | - | Growth Inhibition Assay | - | IC50=579.213 μM | SANGER |
K5 | - | Growth Inhibition Assay | - | IC50=23.5486 μM | SANGER |
K-562 | - | Growth Inhibition Assay | - | IC50=62.2452 μM | SANGER |
KALS-1 | - | Growth Inhibition Assay | - | IC50=73.5475 μM | SANGER |
KARPAS-299 | - | Growth Inhibition Assay | - | IC50=22.1954 μM | SANGER |
KARPAS-422 | - | Growth Inhibition Assay | - | IC50=789.315 μM | SANGER |
KARPAS-45 | - | Growth Inhibition Assay | - | IC50=618.221 μM | SANGER |
KASUMI-1 | - | Growth Inhibition Assay | - | IC50=24.9328 μM | SANGER |
KE-37 | - | Growth Inhibition Assay | - | IC50=102.95 μM | SANGER |
KG-1 | - | Growth Inhibition Assay | - | IC50=189.798 μM | SANGER |
KGN | - | Growth Inhibition Assay | - | IC50=53.959 μM | SANGER |
KINGS-1 | - | Growth Inhibition Assay | - | IC50=167.354 μM | SANGER |
KLE | - | Growth Inhibition Assay | - | IC50=27.2565 μM | SANGER |
KM12 | - | Growth Inhibition Assay | - | IC50=38.5998 μM | SANGER |
KM-H2 | - | Growth Inhibition Assay | - | IC50=699.059 μM | SANGER |
KMOE-2 | - | Growth Inhibition Assay | - | IC50=81.8531 μM | SANGER |
KMS-12-PE | - | Growth Inhibition Assay | - | IC50=456.822 μM | SANGER |
KNS-42 | - | Growth Inhibition Assay | - | IC50=31.8662 μM | SANGER |
KNS-81-FD | - | Growth Inhibition Assay | - | IC50=119.417 μM | SANGER |
KOSC-2 | - | Growth Inhibition Assay | - | IC50=195.818 μM | SANGER |
KP-4 | - | Growth Inhibition Assay | - | IC50=343.733 μM | SANGER |
KP-N-YS | - | Growth Inhibition Assay | - | IC50=78.5878 μM | SANGER |
KS-1 | - | Growth Inhibition Assay | - | IC50=50.2225 μM | SANGER |
KU-19-19 | - | Growth Inhibition Assay | - | IC50=33.7534 μM | SANGER |
KU812 | - | Growth Inhibition Assay | - | IC50=13.5175 μM | SANGER |
KURAMOCHI | - | Growth Inhibition Assay | - | IC50=22.7069 μM | SANGER |
KY821 | - | Growth Inhibition Assay | - | IC50=414.086 μM | SANGER |
KYSE-140 | - | Growth Inhibition Assay | - | IC50=122.141 μM | SANGER |
KYSE-150 | - | Growth Inhibition Assay | - | IC50=169.636 μM | SANGER |
KYSE-180 | - | Growth Inhibition Assay | - | IC50=1.72788 μM | SANGER |
KYSE-270 | - | Growth Inhibition Assay | - | IC50=45.0437 μM | SANGER |
KYSE-410 | - | Growth Inhibition Assay | - | IC50=80.2857 μM | SANGER |
KYSE-450 | - | Growth Inhibition Assay | - | IC50=21.5354 μM | SANGER |
KYSE-510 | - | Growth Inhibition Assay | - | IC50=247.517 μM | SANGER |
KYSE-520 | - | Growth Inhibition Assay | - | IC50=148.54 μM | SANGER |
KYSE-70 | - | Growth Inhibition Assay | - | IC50=203.879 μM | SANGER |
L-363 | - | Growth Inhibition Assay | - | IC50=648.064 μM | SANGER |
L-428 | - | Growth Inhibition Assay | - | IC50=600.671 μM | SANGER |
L-540 | - | Growth Inhibition Assay | - | IC50=149.75 μM | SANGER |
LAMA-84 | - | Growth Inhibition Assay | - | IC50=202.073 μM | SANGER |
LAN-6 | - | Growth Inhibition Assay | - | IC50=336.977 μM | SANGER |
LB1047-RCC | - | Growth Inhibition Assay | - | IC50=9.99798 μM | SANGER |
LB2241-RCC | - | Growth Inhibition Assay | - | IC50=185.145 μM | SANGER |
LB2518-MEL | - | Growth Inhibition Assay | - | IC50=5.72627 μM | SANGER |
LB373-MEL-D | - | Growth Inhibition Assay | - | IC50=31.0047 μM | SANGER |
LB647-SCLC | - | Growth Inhibition Assay | - | IC50=148.562 μM | SANGER |
LB771-HNC | - | Growth Inhibition Assay | - | IC50=217.893 μM | SANGER |
LB831-BLC | - | Growth Inhibition Assay | - | IC50=43.697 μM | SANGER |
LB996-RCC | - | Growth Inhibition Assay | - | IC50=9.52397 μM | SANGER |
LC-1F | - | Growth Inhibition Assay | - | IC50=248.156 μM | SANGER |
LC-2-ad | - | Growth Inhibition Assay | - | IC50=336.591 μM | SANGER |
LC4-1 | - | Growth Inhibition Assay | - | IC50=49.8912 μM | SANGER |
LCLC-103H | - | Growth Inhibition Assay | - | IC50=30.2059 μM | SANGER |
LCLC-97TM1 | - | Growth Inhibition Assay | - | IC50=59.0553 μM | SANGER |
LK-2 | - | Growth Inhibition Assay | - | IC50=147.143 μM | SANGER |
LN-405 | - | Growth Inhibition Assay | - | IC50=269.708 μM | SANGER |
LNCaP-Clone-FGC | - | Growth Inhibition Assay | - | IC50=175.861 μM | SANGER |
LOUCY | - | Growth Inhibition Assay | - | IC50=182.688 μM | SANGER |
LoVo | - | Growth Inhibition Assay | - | IC50=15.2659 μM | SANGER |
LOXIMVI | - | Growth Inhibition Assay | - | IC50=0.58832 μM | SANGER |
LP-1 | - | Growth Inhibition Assay | - | IC50=603.587 μM | SANGER |
LS-1034 | - | Growth Inhibition Assay | - | IC50=202.553 μM | SANGER |
LS-123 | - | Growth Inhibition Assay | - | IC50=328.164 μM | SANGER |
LS-411N | - | Growth Inhibition Assay | - | IC50=74.2528 μM | SANGER |
LS-513 | - | Growth Inhibition Assay | - | IC50=22.6192 μM | SANGER |
LU-134-A | - | Growth Inhibition Assay | - | IC50=59.6016 μM | SANGER |
LU-139 | - | Growth Inhibition Assay | - | IC50=24.835 μM | SANGER |
LU-165 | - | Growth Inhibition Assay | - | IC50=267.941 μM | SANGER |
LU-65 | - | Growth Inhibition Assay | - | IC50=101.081 μM | SANGER |
LU-99A | - | Growth Inhibition Assay | - | IC50=129.931 μM | SANGER |
LXF-289 | - | Growth Inhibition Assay | - | IC50=55.5066 μM | SANGER |
M059J | - | Growth Inhibition Assay | - | IC50=10.6102 μM | SANGER |
M14 | - | Growth Inhibition Assay | - | IC50=23.1132 μM | SANGER |
MC116 | - | Growth Inhibition Assay | - | IC50=7.28691 μM | SANGER |
MC-CAR | - | Growth Inhibition Assay | - | IC50=27.7907 μM | SANGER |
MCF7 | - | Growth Inhibition Assay | - | IC50=51.7554 μM | SANGER |
MC-IXC | - | Growth Inhibition Assay | - | IC50=54.4364 μM | SANGER |
MDA-MB-134-VI | - | Growth Inhibition Assay | - | IC50=431.033 μM | SANGER |
MDA-MB-157 | - | Growth Inhibition Assay | - | IC50=112.49 μM | SANGER |
MDA-MB-175-VII | - | Growth Inhibition Assay | - | IC50=85.7426 μM | SANGER |
MDA-MB-231 | - | Growth Inhibition Assay | - | IC50=200.902 μM | SANGER |
MDA-MB-361 | - | Growth Inhibition Assay | - | IC50=153.164 μM | SANGER |
MDA-MB-415 | - | Growth Inhibition Assay | - | IC50=184.651 μM | SANGER |
MDA-MB-453 | - | Growth Inhibition Assay | - | IC50=186.941 μM | SANGER |
MDA-MB-468 | - | Growth Inhibition Assay | - | IC50=269.333 μM | SANGER |
ME-180 | - | Growth Inhibition Assay | - | IC50=174.016 μM | SANGER |
MEG-01 | - | Growth Inhibition Assay | - | IC50=8.99043 μM | SANGER |
MEL-HO | - | Growth Inhibition Assay | - | IC50=13.8829 μM | SANGER |
MEL-JUSO | - | Growth Inhibition Assay | - | IC50=94.954 μM | SANGER |
MES-SA | - | Growth Inhibition Assay | - | IC50=409.98 μM | SANGER |
Mewo | - | Growth Inhibition Assay | - | IC50=99.5603 μM | SANGER |
MFE-280 | - | Growth Inhibition Assay | - | IC50=201.961 μM | SANGER |
MFE-296 | - | Growth Inhibition Assay | - | IC50=64.4473 μM | SANGER |
MFH-ino | - | Growth Inhibition Assay | - | IC50=131.114 μM | SANGER |
MFM-223 | - | Growth Inhibition Assay | - | IC50=201.587 μM | SANGER |
MG-63 | - | Growth Inhibition Assay | - | IC50=53.9381 μM | SANGER |
MHH-CALL-2 | - | Growth Inhibition Assay | - | IC50=269.92 μM | SANGER |
MHH-ES-1 | - | Growth Inhibition Assay | - | IC50=4.04545 μM | SANGER |
MHH-NB-11 | - | Growth Inhibition Assay | - | IC50=19.5342 μM | SANGER |
MHH-PREB-1 | - | Growth Inhibition Assay | - | IC50=210.381 μM | SANGER |
MIA-PaCa-2 | - | Growth Inhibition Assay | - | IC50=1.75977 μM | SANGER |
MKN1 | - | Growth Inhibition Assay | - | IC50=36.8444 μM | SANGER |
MKN28 | - | Growth Inhibition Assay | - | IC50=8.88516 μM | SANGER |
MKN45 | - | Growth Inhibition Assay | - | IC50=103.584 μM | SANGER |
MKN7 | - | Growth Inhibition Assay | - | IC50=97.7439 μM | SANGER |
ML-2 | - | Growth Inhibition Assay | - | IC50=606.579 μM | SANGER |
MLMA | - | Growth Inhibition Assay | - | IC50=338.155 μM | SANGER |
MMAC-SF | - | Growth Inhibition Assay | - | IC50=261.192 μM | SANGER |
MN-60 | - | Growth Inhibition Assay | - | IC50=393.948 μM | SANGER |
MOLT-16 | - | Growth Inhibition Assay | - | IC50=3.88556 μM | SANGER |
MOLT-4 | - | Growth Inhibition Assay | - | IC50=241.209 μM | SANGER |
MONO-MAC-6 | - | Growth Inhibition Assay | - | IC50=187.392 μM | SANGER |
Mo-T | - | Growth Inhibition Assay | - | IC50=515.116 μM | SANGER |
MPP-89 | - | Growth Inhibition Assay | - | IC50=41.9211 μM | SANGER |
MRK-nu-1 | - | Growth Inhibition Assay | - | IC50=184.972 μM | SANGER |
MS-1 | - | Growth Inhibition Assay | - | IC50=454.385 μM | SANGER |
MSTO-211H | - | Growth Inhibition Assay | - | IC50=233.276 μM | SANGER |
MV-4-11 | - | Growth Inhibition Assay | - | IC50=8.54304 μM | SANGER |
MZ1-PC | - | Growth Inhibition Assay | - | IC50=94.5984 μM | SANGER |
MZ2-MEL | - | Growth Inhibition Assay | - | IC50=10.4677 μM | SANGER |
MZ7-mel | - | Growth Inhibition Assay | - | IC50=91.2676 μM | SANGER |
NALM-6 | - | Growth Inhibition Assay | - | IC50=30.4965 μM | SANGER |
NB1 | - | Growth Inhibition Assay | - | IC50=14.1935 μM | SANGER |
NB10 | - | Growth Inhibition Assay | - | IC50=177.846 μM | SANGER |
NB12 | - | Growth Inhibition Assay | - | IC50=80.9369 μM | SANGER |
NB13 | - | Growth Inhibition Assay | - | IC50=345.58 μM | SANGER |
NB5 | - | Growth Inhibition Assay | - | IC50=526.43 μM | SANGER |
NB6 | - | Growth Inhibition Assay | - | IC50=78.1299 μM | SANGER |
NB69 | - | Growth Inhibition Assay | - | IC50=277.405 μM | SANGER |
NCCIT | - | Growth Inhibition Assay | - | IC50=236.873 μM | SANGER |
NCI-H1092 | - | Growth Inhibition Assay | - | IC50=463.943 μM | SANGER |
NCI-H1155 | - | Growth Inhibition Assay | - | IC50=818.059 μM | SANGER |
NCI-H1299 | - | Growth Inhibition Assay | - | IC50=188.719 μM | SANGER |
NCI-H1304 | - | Growth Inhibition Assay | - | IC50=253.156 μM | SANGER |
NCI-H1355 | - | Growth Inhibition Assay | - | IC50=221.377 μM | SANGER |
NCI-H1395 | - | Growth Inhibition Assay | - | IC50=489.004 μM | SANGER |
NCI-H1417 | - | Growth Inhibition Assay | - | IC50=81.4368 μM | SANGER |
NCI-H1436 | - | Growth Inhibition Assay | - | IC50=523.064 μM | SANGER |
NCI-H1437 | - | Growth Inhibition Assay | - | IC50=134.59 μM | SANGER |
NCI-H1522 | - | Growth Inhibition Assay | - | IC50=334.339 μM | SANGER |
NCI-H1563 | - | Growth Inhibition Assay | - | IC50=185.209 μM | SANGER |
NCI-H1581 | - | Growth Inhibition Assay | - | IC50=900.231 μM | SANGER |
NCI-H1618 | - | Growth Inhibition Assay | - | IC50=221.018 μM | SANGER |
NCI-H1623 | - | Growth Inhibition Assay | - | IC50=222.389 μM | SANGER |
NCI-H1648 | - | Growth Inhibition Assay | - | IC50=32.8467 μM | SANGER |
NCI-H1650 | - | Growth Inhibition Assay | - | IC50=51.5849 μM | SANGER |
NCI-H1651 | - | Growth Inhibition Assay | - | IC50=206.73 μM | SANGER |
NCI-H1693 | - | Growth Inhibition Assay | - | IC50=249.495 μM | SANGER |
NCI-H1694 | - | Growth Inhibition Assay | - | IC50=512.439 μM | SANGER |
NCI-H1703 | - | Growth Inhibition Assay | - | IC50=68.1171 μM | SANGER |
NCI-H1734 | - | Growth Inhibition Assay | - | IC50=61.9663 μM | SANGER |
NCI-H1755 | - | Growth Inhibition Assay | - | IC50=9.39986 μM | SANGER |
NCI-H1770 | - | Growth Inhibition Assay | - | IC50=26.8986 μM | SANGER |
NCI-H1792 | - | Growth Inhibition Assay | - | IC50=279.187 μM | SANGER |
NCI-H1793 | - | Growth Inhibition Assay | - | IC50=51.231 μM | SANGER |
NCI-H1838 | - | Growth Inhibition Assay | - | IC50=359.987 μM | SANGER |
NCI-H187 | - | Growth Inhibition Assay | - | IC50=256.76 μM | SANGER |
NCI-H1882 | - | Growth Inhibition Assay | - | IC50=286.035 μM | SANGER |
NCI-H1963 | - | Growth Inhibition Assay | - | IC50=24.2839 μM | SANGER |
NCI-H1993 | - | Growth Inhibition Assay | - | IC50=222.239 μM | SANGER |
NCI-H2009 | - | Growth Inhibition Assay | - | IC50=283.953 μM | SANGER |
NCI-H2030 | - | Growth Inhibition Assay | - | IC50=341.609 μM | SANGER |
NCI-H2052 | - | Growth Inhibition Assay | - | IC50=159.583 μM | SANGER |
NCI-H2081 | - | Growth Inhibition Assay | - | IC50=525.513 μM | SANGER |
NCI-H2087 | - | Growth Inhibition Assay | - | IC50=124.283 μM | SANGER |
NCI-H209 | - | Growth Inhibition Assay | - | IC50=226.53 μM | SANGER |
NCI-H2122 | - | Growth Inhibition Assay | - | IC50=2.27684 μM | SANGER |
NCI-H2126 | - | Growth Inhibition Assay | - | IC50=358.521 μM | SANGER |
NCI-H2141 | - | Growth Inhibition Assay | - | IC50=424.388 μM | SANGER |
NCI-H2170 | - | Growth Inhibition Assay | - | IC50=27.5282 μM | SANGER |
NCI-H2171 | - | Growth Inhibition Assay | - | IC50=512.705 μM | SANGER |
NCI-H2196 | - | Growth Inhibition Assay | - | IC50=352.624 μM | SANGER |
NCI-H2227 | - | Growth Inhibition Assay | - | IC50=530.254 μM | SANGER |
NCI-H2228 | - | Growth Inhibition Assay | - | IC50=250.864 μM | SANGER |
NCI-H226 | - | Growth Inhibition Assay | - | IC50=628.353 μM | SANGER |
NCI-H23 | - | Growth Inhibition Assay | - | IC50=108.357 μM | SANGER |
NCI-H2342 | - | Growth Inhibition Assay | - | IC50=69.3961 μM | SANGER |
NCI-H2347 | - | Growth Inhibition Assay | - | IC50=296.425 μM | SANGER |
NCI-H2405 | - | Growth Inhibition Assay | - | IC50=56.1693 μM | SANGER |
NCI-H2452 | - | Growth Inhibition Assay | - | IC50=5.45628 μM | SANGER |
NCI-H28 | - | Growth Inhibition Assay | - | IC50=10.4413 μM | SANGER |
NCI-H292 | - | Growth Inhibition Assay | - | IC50=99.3004 μM | SANGER |
NCI-H322M | - | Growth Inhibition Assay | - | IC50=228.019 μM | SANGER |
NCI-H345 | - | Growth Inhibition Assay | - | IC50=203.027 μM | SANGER |
NCI-H358 | - | Growth Inhibition Assay | - | IC50=355.356 μM | SANGER |
NCI-H441 | - | Growth Inhibition Assay | - | IC50=341.418 μM | SANGER |
NCI-H446 | - | Growth Inhibition Assay | - | IC50=477.08 μM | SANGER |
NCI-H460 | - | Growth Inhibition Assay | - | IC50=251.417 μM | SANGER |
NCI-H510A | - | Growth Inhibition Assay | - | IC50=524.696 μM | SANGER |
NCI-H520 | - | Growth Inhibition Assay | - | IC50=235.741 μM | SANGER |
NCI-H522 | - | Growth Inhibition Assay | - | IC50=181.059 μM | SANGER |
NCI-H524 | - | Growth Inhibition Assay | - | IC50=295.769 μM | SANGER |
NCI-H526 | - | Growth Inhibition Assay | - | IC50=11.1365 μM | SANGER |
NCI-H596 | - | Growth Inhibition Assay | - | IC50=385.34 μM | SANGER |
NCI-H630 | - | Growth Inhibition Assay | - | IC50=232.897 μM | SANGER |
NCI-H64 | - | Growth Inhibition Assay | - | IC50=9.42255 μM | SANGER |
NCI-H650 | - | Growth Inhibition Assay | - | IC50=89.8724 μM | SANGER |
NCI-H661 | - | Growth Inhibition Assay | - | IC50=81.344 μM | SANGER |
NCI-H69 | - | Growth Inhibition Assay | - | IC50=214.185 μM | SANGER |
NCI-H716 | - | Growth Inhibition Assay | - | IC50=410.075 μM | SANGER |
NCI-H719 | - | Growth Inhibition Assay | - | IC50=391.893 μM | SANGER |
NCI-H720 | - | Growth Inhibition Assay | - | IC50=349.846 μM | SANGER |
NCI-H727 | - | Growth Inhibition Assay | - | IC50=20.2169 μM | SANGER |
NCI-H747 | - | Growth Inhibition Assay | - | IC50=47.7264 μM | SANGER |
NCI-H748 | - | Growth Inhibition Assay | - | IC50=150.209 μM | SANGER |
NCI-H810 | - | Growth Inhibition Assay | - | IC50=143.687 μM | SANGER |
NCI-H82 | - | Growth Inhibition Assay | - | IC50=13.2909 μM | SANGER |
NCI-H838 | - | Growth Inhibition Assay | - | IC50=190.34 μM | SANGER |
NCI-H889 | - | Growth Inhibition Assay | - | IC50=547.23 μM | SANGER |
NCI-N87 | - | Growth Inhibition Assay | - | IC50=121.044 μM | SANGER |
NCI-SNU-1 | - | Growth Inhibition Assay | - | IC50=690.172 μM | SANGER |
NCI-SNU-16 | - | Growth Inhibition Assay | - | IC50=680.462 μM | SANGER |
NCI-SNU-5 | - | Growth Inhibition Assay | - | IC50=472.28 μM | SANGER |
NEC8 | - | Growth Inhibition Assay | - | IC50=112.624 μM | SANGER |
Neural progenitor cells | 3 μM | Function Assay | 10 d | Induces generation of neural progenitor cells | 24638034 |
NH-12 | - | Growth Inhibition Assay | - | IC50=16.0097 μM | SANGER |
NKM-1 | - | Growth Inhibition Assay | - | IC50=4.13971 μM | SANGER |
NMC-G1 | - | Growth Inhibition Assay | - | IC50=61.9242 μM | SANGER |
no-10 | - | Growth Inhibition Assay | - | IC50=38.1294 μM | SANGER |
no-11 | - | Growth Inhibition Assay | - | IC50=46.2031 μM | SANGER |
NOMO-1 | - | Growth Inhibition Assay | - | IC50=236.02 μM | SANGER |
NOS-1 | - | Growth Inhibition Assay | - | IC50=134.765 μM | SANGER |
NTERA-S-cl-D1 | - | Growth Inhibition Assay | - | IC50=326.489 μM | SANGER |
NUGC-3 | - | Growth Inhibition Assay | - | IC50=209.678 μM | SANGER |
NY | - | Growth Inhibition Assay | - | IC50=42.1801 μM | SANGER |
OAW-28 | - | Growth Inhibition Assay | - | IC50=28.0052 μM | SANGER |
OAW-42 | - | Growth Inhibition Assay | - | IC50=137.856 μM | SANGER |
OCI-AML2 | - | Growth Inhibition Assay | - | IC50=141.507 μM | SANGER |
Oct4/Sox2/Klf4-infected MEFs | 10 μM | Function Assay | 28 d | Promotes MEFs reprogramming Transduced by Oct4, Sox2, and Klf4 | 19839055 |
OCUB-M | - | Growth Inhibition Assay | - | IC50=323.434 μM | SANGER |
OE19 | - | Growth Inhibition Assay | - | IC50=3.96451 μM | SANGER |
OE33 | - | Growth Inhibition Assay | - | IC50=141.798 μM | SANGER |
OMC-1 | - | Growth Inhibition Assay | - | IC50=145.967 μM | SANGER |
ONS-76 | - | Growth Inhibition Assay | - | IC50=182.387 μM | SANGER |
OPM-2 | - | Growth Inhibition Assay | - | IC50=123.176 μM | SANGER |
OS-RC-2 | - | Growth Inhibition Assay | - | IC50=97.461 μM | SANGER |
OVCAR-3 | - | Growth Inhibition Assay | - | IC50=119.915 μM | SANGER |
OVCAR-4 | - | Growth Inhibition Assay | - | IC50=140.749 μM | SANGER |
OVCAR-5 | - | Growth Inhibition Assay | - | IC50=168.309 μM | SANGER |
OVCAR-8 | - | Growth Inhibition Assay | - | IC50=117.668 μM | SANGER |
P12-ICHIKAWA | - | Growth Inhibition Assay | - | IC50=511.416 μM | SANGER |
P30-OHK | - | Growth Inhibition Assay | - | IC50=353.063 μM | SANGER |
P31-FUJ | - | Growth Inhibition Assay | - | IC50=376.964 μM | SANGER |
PA-1 | - | Growth Inhibition Assay | - | IC50=11.93 μM | SANGER |
PANC-03-27 | - | Growth Inhibition Assay | - | IC50=78.435 μM | SANGER |
PANC-08-13 | - | Growth Inhibition Assay | - | IC50=106.85 μM | SANGER |
PANC1 | 5 μM | Apoptosis Assay | 72 h | Triggers an apoptotic response | 22201186 |
PANC-10-05 | - | Growth Inhibition Assay | - | IC50=24.0898 μM | SANGER |
PC-14 | - | Growth Inhibition Assay | - | IC50=12.324 μM | SANGER |
PC-3 | - | Growth Inhibition Assay | - | IC50=99.0564 μM | SANGER |
PF-382 | - | Growth Inhibition Assay | - | IC50=344.422 μM | SANGER |
PFSK-1 | - | Growth Inhibition Assay | - | IC50=34.9241 μM | SANGER |
platelets | 10 μM | Function Assay | 15 min | Increases thrombin-mediated platelet aggregation and ATP secretion | 23239877 |
PLC-PRF-5 | - | Growth Inhibition Assay | - | IC50=304.907 μM | SANGER |
PSN1 | - | Growth Inhibition Assay | - | IC50=181.66 μM | SANGER |
QIMR-WIL | - | Growth Inhibition Assay | - | IC50=200.116 μM | SANGER |
Raji | - | Growth Inhibition Assay | - | IC50=338.38 μM | SANGER |
Ramos-2G6-4C10 | - | Growth Inhibition Assay | - | IC50=46.0755 μM | SANGER |
RCC10RGB | - | Growth Inhibition Assay | - | IC50=4.29479 μM | SANGER |
RCM-1 | - | Growth Inhibition Assay | - | IC50=56.0078 μM | SANGER |
RD | - | Growth Inhibition Assay | - | IC50=269.119 μM | SANGER |
REH | - | Growth Inhibition Assay | - | IC50=23.1699 μM | SANGER |
RERF-LC-MS | - | Growth Inhibition Assay | - | IC50=154.772 μM | SANGER |
RH-1 | - | Growth Inhibition Assay | - | IC50=435.09 μM | SANGER |
RKO | - | Growth Inhibition Assay | - | IC50=117.898 μM | SANGER |
RL | - | Growth Inhibition Assay | - | IC50=542.442 μM | SANGER |
RL95-2 | - | Growth Inhibition Assay | - | IC50=300.247 μM | SANGER |
RMG-I | - | Growth Inhibition Assay | - | IC50=95.1072 μM | SANGER |
RO82-W-1 | - | Growth Inhibition Assay | - | IC50=26.7377 μM | SANGER |
RPMI-2650 | - | Growth Inhibition Assay | - | IC50=205.467 μM | SANGER |
RPMI-6666 | - | Growth Inhibition Assay | - | IC50=491.398 μM | SANGER |
RPMI-7951 | - | Growth Inhibition Assay | - | IC50=2.70193 μM | SANGER |
RPMI-8226 | - | Growth Inhibition Assay | - | IC50=106.678 μM | SANGER |
RPMI-8402 | - | Growth Inhibition Assay | - | IC50=510.021 μM | SANGER |
RPMI-8866 | - | Growth Inhibition Assay | - | IC50=57.2412 μM | SANGER |
RS4-11 | - | Growth Inhibition Assay | - | IC50=1.95415 μM | SANGER |
RT-112 | - | Growth Inhibition Assay | - | IC50=7.16456 μM | SANGER |
RT4 | - | Growth Inhibition Assay | - | IC50=73.5742 μM | SANGER |
RVH-421 | - | Growth Inhibition Assay | - | IC50=33.168 μM | SANGER |
RXF393 | - | Growth Inhibition Assay | - | IC50=22.6068 μM | SANGER |
S-117 | - | Growth Inhibition Assay | - | IC50=0.92131 μM | SANGER |
Saos-2 | - | Growth Inhibition Assay | - | IC50=101.437 μM | SANGER |
SAS | - | Growth Inhibition Assay | - | IC50=223.796 μM | SANGER |
SBC-1 | - | Growth Inhibition Assay | - | IC50=84.0208 μM | SANGER |
SBC-5 | - | Growth Inhibition Assay | - | IC50=181.934 μM | SANGER |
Sca-1+ HPC | 2 μM | Growth Inhibition Assay | 6 d | Synergistically promotes Sca-1+ HPC proliferation and colony formation together with EGF | 21624348 |
SCC-15 | - | Growth Inhibition Assay | - | IC50=306.017 μM | SANGER |
SCC-25 | - | Growth Inhibition Assay | - | IC50=144.005 μM | SANGER |
SCC-3 | - | Growth Inhibition Assay | - | IC50=220.577 μM | SANGER |
SCC-4 | - | Growth Inhibition Assay | - | IC50=220.353 μM | SANGER |
SCC-9 | - | Growth Inhibition Assay | - | IC50=2.95485 μM | SANGER |
SCH | - | Growth Inhibition Assay | - | IC50=64.2351 μM | SANGER |
SCLC-21H | - | Growth Inhibition Assay | - | IC50=455.699 μM | SANGER |
SF126 | - | Growth Inhibition Assay | - | IC50=179.432 μM | SANGER |
SF268 | - | Growth Inhibition Assay | - | IC50=330.265 μM | SANGER |
SF295 | - | Growth Inhibition Assay | - | IC50=79.9553 μM | SANGER |
SF539 | - | Growth Inhibition Assay | - | IC50=14.0116 μM | SANGER |
SH-4 | - | Growth Inhibition Assay | - | IC50=283.123 μM | SANGER |
SHP-77 | - | Growth Inhibition Assay | - | IC50=295.597 μM | SANGER |
SIG-M5 | - | Growth Inhibition Assay | - | IC50=113.125 μM | SANGER |
SiHa | - | Growth Inhibition Assay | - | IC50=59.6487 μM | SANGER |
SIMA | - | Growth Inhibition Assay | - | IC50=17.9118 μM | SANGER |
SJRH30 | - | Growth Inhibition Assay | - | IC50=200.515 μM | SANGER |
SJSA-1 | - | Growth Inhibition Assay | - | IC50=360.939 μM | SANGER |
SK-CO-1 | - | Growth Inhibition Assay | - | IC50=41.7755 μM | SANGER |
SKG-IIIa | - | Growth Inhibition Assay | - | IC50=118.116 μM | SANGER |
SK-HEP-1 | - | Growth Inhibition Assay | - | IC50=246.043 μM | SANGER |
SK-LMS-1 | - | Growth Inhibition Assay | - | IC50=2.64128 μM | SANGER |
SK-LU-1 | - | Growth Inhibition Assay | - | IC50=188.428 μM | SANGER |
SK-MEL-1 | - | Growth Inhibition Assay | - | IC50=75.8019 μM | SANGER |
SK-MEL-2 | - | Growth Inhibition Assay | - | IC50=6.38344 μM | SANGER |
SK-MEL-24 | - | Growth Inhibition Assay | - | IC50=324.111 μM | SANGER |
SK-MEL-28 | - | Growth Inhibition Assay | - | IC50=21.6863 μM | SANGER |
SK-MEL-3 | - | Growth Inhibition Assay | - | IC50=275.457 μM | SANGER |
SK-MEL-30 | - | Growth Inhibition Assay | - | IC50=326.738 μM | SANGER |
SK-MES-1 | - | Growth Inhibition Assay | - | IC50=101.762 μM | SANGER |
SK-MM-2 | - | Growth Inhibition Assay | - | IC50=30.9792 μM | SANGER |
SK-N-AS | - | Growth Inhibition Assay | - | IC50=51.8281 μM | SANGER |
SK-N-DZ | - | Growth Inhibition Assay | - | IC50=9.65742 μM | SANGER |
SK-NEP-1 | - | Growth Inhibition Assay | - | IC50=177.806 μM | SANGER |
SK-N-FI | - | Growth Inhibition Assay | - | IC50=322.452 μM | SANGER |
SK-OV-3 | - | Growth Inhibition Assay | - | IC50=4.9934 μM | SANGER |
SK-PN-DW | - | Growth Inhibition Assay | - | IC50=347.426 μM | SANGER |
SK-UT-1 | - | Growth Inhibition Assay | - | IC50=36.3331 μM | SANGER |
SN12C | - | Growth Inhibition Assay | - | IC50=182.829 μM | SANGER |
SNB75 | - | Growth Inhibition Assay | - | IC50=48.4118 μM | SANGER |
SNG-M | - | Growth Inhibition Assay | - | IC50=27.2271 μM | SANGER |
SNU-387 | - | Growth Inhibition Assay | - | IC50=10.7235 μM | SANGER |
SNU-423 | - | Growth Inhibition Assay | - | IC50=2.49787 μM | SANGER |
SNU-449 | - | Growth Inhibition Assay | - | IC50=18.715 μM | SANGER |
SNU-475 | - | Growth Inhibition Assay | - | IC50=314.091 μM | SANGER |
SNU-C1 | - | Growth Inhibition Assay | - | IC50=49.3207 μM | SANGER |
SNU-C2B | - | Growth Inhibition Assay | - | IC50=105.023 μM | SANGER |
SR | - | Growth Inhibition Assay | - | IC50=43.8673 μM | SANGER |
ST486 | - | Growth Inhibition Assay | - | IC50=14.2251 μM | SANGER |
SU-DHL-1 | - | Growth Inhibition Assay | - | IC50=27.9474 μM | SANGER |
SUP-T1 | - | Growth Inhibition Assay | - | IC50=118.956 μM | SANGER |
SW1088 | - | Growth Inhibition Assay | - | IC50=195.677 μM | SANGER |
SW13 | - | Growth Inhibition Assay | - | IC50=147.253 μM | SANGER |
SW1417 | - | Growth Inhibition Assay | - | IC50=7.64584 μM | SANGER |
SW1463 | - | Growth Inhibition Assay | - | IC50=124.077 μM | SANGER |
SW1573 | - | Growth Inhibition Assay | - | IC50=82.5893 μM | SANGER |
SW1710 | - | Growth Inhibition Assay | - | IC50=5.42456 μM | SANGER |
SW1783 | - | Growth Inhibition Assay | - | IC50=234.41 μM | SANGER |
SW1990 | - | Growth Inhibition Assay | - | IC50=351.28 μM | SANGER |
SW48 | - | Growth Inhibition Assay | - | IC50=13.7265 μM | SANGER |
SW620 | - | Growth Inhibition Assay | - | IC50=171.535 μM | SANGER |
SW626 | - | Growth Inhibition Assay | - | IC50=296.115 μM | SANGER |
SW684 | - | Growth Inhibition Assay | - | IC50=22.2858 μM | SANGER |
SW756 | - | Growth Inhibition Assay | - | IC50=174.863 μM | SANGER |
SW780 | - | Growth Inhibition Assay | - | IC50=196.734 μM | SANGER |
SW837 | - | Growth Inhibition Assay | - | IC50=51.9785 μM | SANGER |
SW872 | - | Growth Inhibition Assay | - | IC50=28.5326 μM | SANGER |
SW948 | - | Growth Inhibition Assay | - | IC50=32.7548 μM | SANGER |
SW954 | - | Growth Inhibition Assay | - | IC50=237.868 μM | SANGER |
SW962 | - | Growth Inhibition Assay | - | IC50=398.69 μM | SANGER |
SW982 | - | Growth Inhibition Assay | - | IC50=0.21416 μM | SANGER |
T-24 | - | Growth Inhibition Assay | - | IC50=62.7126 μM | SANGER |
T47D | - | Growth Inhibition Assay | - | IC50=247.013 μM | SANGER |
T84 | - | Growth Inhibition Assay | - | IC50=284.665 μM | SANGER |
T98G | - | Growth Inhibition Assay | - | IC50=13.4717 μM | SANGER |
TALL-1 | - | Growth Inhibition Assay | - | IC50=455.297 μM | SANGER |
TCCSUP | - | Growth Inhibition Assay | - | IC50=211.533 μM | SANGER |
TE-1 | - | Growth Inhibition Assay | - | IC50=196.26 μM | SANGER |
TE-10 | - | Growth Inhibition Assay | - | IC50=276.439 μM | SANGER |
TE-11 | - | Growth Inhibition Assay | - | IC50=101.724 μM | SANGER |
TE-12 | - | Growth Inhibition Assay | - | IC50=89.3741 μM | SANGER |
TE-15 | - | Growth Inhibition Assay | - | IC50=3.95343 μM | SANGER |
TE-441-T | - | Growth Inhibition Assay | - | IC50=457.186 μM | SANGER |
TE-5 | - | Growth Inhibition Assay | - | IC50=198.033 μM | SANGER |
TE-6 | - | Growth Inhibition Assay | - | IC50=397.254 μM | SANGER |
TE-8 | - | Growth Inhibition Assay | - | IC50=43.7895 μM | SANGER |
TE-9 | - | Growth Inhibition Assay | - | IC50=149.443 μM | SANGER |
TGBC1TKB | - | Growth Inhibition Assay | - | IC50=252.875 μM | SANGER |
TGBC24TKB | - | Growth Inhibition Assay | - | IC50=21.8957 μM | SANGER |
TGW | - | Growth Inhibition Assay | - | IC50=283.058 μM | SANGER |
THP-1 | - | Growth Inhibition Assay | - | IC50=219.606 μM | SANGER |
TK10 | - | Growth Inhibition Assay | - | IC50=35.1322 μM | SANGER |
TT | - | Growth Inhibition Assay | - | IC50=153.49 μM | SANGER |
TUR | - | Growth Inhibition Assay | - | IC50=671.322 μM | SANGER |
TYK-nu | - | Growth Inhibition Assay | - | IC50=1.07912 μM | SANGER |
U031 | - | Growth Inhibition Assay | - | IC50=112.065 μM | SANGER |
U-118-MG | - | Growth Inhibition Assay | - | IC50=9.94444 μM | SANGER |
U251 | - | Growth Inhibition Assay | - | IC50=298.438 μM | SANGER |
U-266 | - | Growth Inhibition Assay | - | IC50=373.132 μM | SANGER |
U-2-OS | - | Growth Inhibition Assay | - | IC50=9.45006 μM | SANGER |
U-698-M | - | Growth Inhibition Assay | - | IC50=98.9489 μM | SANGER |
U-87-MG | - | Growth Inhibition Assay | - | IC50=694.585 μM | SANGER |
UACC-257 | - | Growth Inhibition Assay | - | IC50=217.43 μM | SANGER |
UACC-62 | - | Growth Inhibition Assay | - | IC50=46.8608 μM | SANGER |
UACC-812 | - | Growth Inhibition Assay | - | IC50=559.391 μM | SANGER |
UACC-893 | - | Growth Inhibition Assay | - | IC50=280.54 μM | SANGER |
UMC-11 | - | Growth Inhibition Assay | - | IC50=126.038 μM | SANGER |
UM-UC-3 | - | Growth Inhibition Assay | - | IC50=103.842 μM | SANGER |
VA-ES-BJ | - | Growth Inhibition Assay | - | IC50=261.918 μM | SANGER |
VM-CUB-1 | - | Growth Inhibition Assay | - | IC50=342.636 μM | SANGER |
VMRC-RCZ | - | Growth Inhibition Assay | - | IC50=130.375 μM | SANGER |
WM-115 | - | Growth Inhibition Assay | - | IC50=5.81509 μM | SANGER |
WSU-NHL | - | Growth Inhibition Assay | - | IC50=112.01 μM | SANGER |
YAPC | - | Growth Inhibition Assay | - | IC50=234.253 μM | SANGER |
YKG-1 | - | Growth Inhibition Assay | - | IC50=142.889 μM | SANGER |
YT | - | Growth Inhibition Assay | - | IC50=176.399 μM | SANGER |
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