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CAS No.: 664969-54-4

4-(3-Phenylallyl)-N-(4-sulfamoylphenyl)piperazine-1-carbothioamide Catalog No. CSN22542

Synonyms: LF3

LF3 is an inhibitor of canonical wnt signaling pathway with IC50 of less than 2 μM. It can disrupt the interaction between β-catenin and TCF4.

规格 价格 促销价格 库存 数量
纯度 & 质量文件 批次:

靶点选择性

生物活性

  • 描述
  • 动物研究
    剂量

    NOD/SCID Mice: 50 mg/kg[1] (i.v.)

    给药途径

    i.v.

  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02683616Obstructive Sleep Apnea ... more >> Fatty Acid Metabolism Continuous Positive Airway Pressure Collapse <<Not ApplicableRecruitingDecember 2019Czechia ... more >> FN Kralovske Vinohrady Recruiting Prague, Czechia, 10034 Contact: Jan Polak, MD, PhD    +420267162710    jan.polak@lf3.cuni.cz    Contact: Jan Gojda, MD, PhD    +420267168144    jan.gojda@lf3.cuni.cz Collapse <<
    NCT03710850Insulin Resistance ... more >> Microbiome Collapse <<Not ApplicableRecruitingDecember 31, 2021Czechia ... more >> University Hospital Kralovske Vinohrady Recruiting Prague, Czechia, 10084 Contact: Jana Potočková    +420267163031    klinicka.fyziologie@lf3.cuni.cz Collapse <<
    NCT03386461Metabolism Disorder ... more >> Adiposity Inflammatory Response Collapse <<Not ApplicableRecruitingDecember 2019Czechia ... more >> Third Faculty of Medicine, Charles University Recruiting Prague, Czechia, 100 00 Contact: Michaela Siklova, PhD    +420 267 102 211    michaela.siklova@lf3.cuni.cz    Contact: Lenka Rossmeislova, PhD    +420 267 102 211    lenka.rossmeislova@lf3.cuni.cz    Principal Investigator: Michaela Siklova, PhD          Sub-Investigator: Martin Rossmeisl, PhD          Sub-Investigator: Vladimir Stich, prof. MUDr. Collapse <<
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实验方案

技术信息

CAS号 664969-54-4 储存条件
分子式 C20H24N4O2S2 运输 蓝冰
分子量 416.56 别名 LF3
溶解度
DMSO50.0 mg/mL (120.0 mM)
Waterinsoluble
动物实验配方

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