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CAS No.: 602306-29-6
AZD5438 is a potent inhibitor of CDK1/2/9 with IC50 of 16/6/20 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00088790 | Neoplasms | Phase 1 | Completed | - | United States, Massachusetts ... more >> Research Site Boston, Massachusetts, United States United States, New York Research Site New York City, New York, United States Collapse << |
实验方案
技术信息
CAS号 | 602306-29-6 | 储存条件 |
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分子式 | C18H21N5O2S | 运输 | 蓝冰 | |||||
分子量 | 371.46 | 别名 | ||||||
溶解度 |
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动物实验配方 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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human LoVo cells | - | Proliferation assay | 48 h | Antiproliferative activity against human LoVo cells assessed as BrdU incorporation after 48 hrs, IC50=0.63 μM | 18815031 |
human LoVo cells | - | Proliferation assay | 48 h | Antiproliferative activity against human LoVo cells assessed as inhibition of BrdU incorporation after 48 hrs, IC50=0.8 μM | 18996007 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00088790 | Neoplasms | Phase 1 | Completed | - | United States, Massachusetts ... more >> Research Site Boston, Massachusetts, United States United States, New York Research Site New York City, New York, United States Collapse << |
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