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CAS No.: 72509-76-3
Synonyms: 非洛地平
Felodipine is a long-acting 1,4-dihydropyridine calcium channel blocker.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02988102 | - | - | Unknown | August 2017 | Albania ... more >> Fatos Kelmendi Recruiting Tirana, Kosovo Prishtina, Albania, 10 000 Contact: Agon Mekaj, PhD +37744373545 dragonmekaj@gmail.com Contact: Ridvan Alimehmeti, PhD +355692102140 ridvanalimehmeti@hotmail.com Collapse << |
NCT00695656 | - | - | Completed | - | - |
NCT00000620 | Atherosclerosis ... more >> Cardiovascular Diseases Hypercholesterolemia Hypertension Diabetes Mellitus, Type 2 Diabetes Mellitus Coronary Disease Collapse << | Phase 3 | Completed | - | United States, Minnesota ... more >> Minneapolis Medical Research Foundation Minneapolis, Minnesota, United States, 55404 United States, New York Columbia University New York, New York, United States, 10027 United States, North Carolina Wake Forest University Winston-Salem, North Carolina, United States, 27106 United States, Ohio Case Western Reserve University Cleveland, Ohio, United States, 44106 United States, Tennessee Veterans Affairs Memphis, Tennessee, United States, 38104 United States, Washington University of Washington Seattle, Washington, United States, 98195 Canada, Ontario McMaster University Hamilton, Ontario, Canada Collapse << |
实验方案
技术信息
CAS号 | 72509-76-3 | 储存条件 |
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分子式 | C18H19Cl2NO4 | 运输 | 蓝冰 | |||||||
分子量 | 384.25 | 别名 | 非洛地平 | |||||||
溶解度 |
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动物实验配方 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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H9C2 cells | - | Function assay | - | Inhibition of L-VDCC in rat H9C2 cells assessed as effect on calcium level by Fluo-4 fluorescence assay | 19880323 |
HepG2 (DPX-2) cells | - | Function assay | 24 h | Activation of human PXR expressed in human HepG2 (DPX-2) cells assessed as induction of CYP3A4 after 24 hrs by luminescent analysis, EC50=1.9 μM | 20966043 |
HepG2 cells | - | Function assay | 24 h | Activation of rat PXR expressed in human HepG2 cells after 24 hrs by luciferase reporter gene based luminescent analysis, EC50=23.4 μM | 20966043 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02988102 | - | - | Unknown | August 2017 | Albania ... more >> Fatos Kelmendi Recruiting Tirana, Kosovo Prishtina, Albania, 10 000 Contact: Agon Mekaj, PhD +37744373545 dragonmekaj@gmail.com Contact: Ridvan Alimehmeti, PhD +355692102140 ridvanalimehmeti@hotmail.com Collapse << |
NCT00695656 | - | - | Completed | - | - |
NCT00000620 | Atherosclerosis ... more >> Cardiovascular Diseases Hypercholesterolemia Hypertension Diabetes Mellitus, Type 2 Diabetes Mellitus Coronary Disease Collapse << | Phase 3 | Completed | - | United States, Minnesota ... more >> Minneapolis Medical Research Foundation Minneapolis, Minnesota, United States, 55404 United States, New York Columbia University New York, New York, United States, 10027 United States, North Carolina Wake Forest University Winston-Salem, North Carolina, United States, 27106 United States, Ohio Case Western Reserve University Cleveland, Ohio, United States, 44106 United States, Tennessee Veterans Affairs Memphis, Tennessee, United States, 38104 United States, Washington University of Washington Seattle, Washington, United States, 98195 Canada, Ontario McMaster University Hamilton, Ontario, Canada Collapse << |
NCT00000620 | - | - | Completed | - | - |
NCT00770250 | - | - | Completed | - | - |
NCT00882128 | - | - | Completed | - | - |
NCT00582114 | Hemodialysis ... more >>Hypertension Left Ventricular Hypertrophy Collapse << | Phase 3 | Terminated(Stopped by data saf... more >>ety monitoring board) Collapse << | - | United States, Indiana ... more >> Indiana University Indianapolis, Indiana, United States, 46202 Collapse << |
NCT00684489 | Hypertension | Not Applicable | Completed | - | - |
NCT00582114 | - | - | Terminated(Stopped by data saf... more >>ety monitoring board) Collapse << | - | - |
NCT00679653 | Obesity Hyper... more >>tension Collapse << | Phase 3 | Completed | - | - |
NCT00348686 | - | - | Completed | - | - |
NCT00742066 | Hypertension ... more >>Insulin Resistance Microcirculation Collapse << | Not Applicable | Unknown | July 2009 | Netherlands ... more >> University Hospital Maastricht Maastricht, P.O. Box 5800, Netherlands, 6202 AZ Collapse << |
NCT00392262 | Hypertension | Phase 3 | Completed | - | Germany ... more >> Investigative Centers, Germany Switzerland Novartis Basel, Switzerland Collapse << |
NCT00367939 | Hypertension | Phase 3 | Completed | - | Germany ... more >> Investigative Centers, Germany Collapse << |
NCT00348686 | Hypertension ... more >>Left Ventricular Hypertrophy Collapse << | Phase 4 | Completed | - | Korea, Republic of ... more >> Research Site BuSan, Korea, Republic of Research Site CheonAn, Korea, Republic of Research Site CheongJu, Korea, Republic of Research Site Chunbuk, Korea, Republic of Research Site DaeGu, Korea, Republic of Research Site DaeJeon, Korea, Republic of Research Site Gyungsangnamdo, Korea, Republic of Research Site JeonJu, Korea, Republic of Research Site KwangJu, Korea, Republic of Research Site Pusan, Korea, Republic of Research Site Ulsan, Korea, Republic of Collapse << |
NCT02744872 | Disorder Related to Lung Trans... more >>plantation Collapse << | Phase 4 | Completed | - | Denmark ... more >> Department of Nephrology P, Copenhagen University Hospital, Rigshospitalet Copenhagen Ø, Copenhagen, Denmark, 2100 Collapse << |
NCT01238705 | Hypertension ... more >>Sexual Dysfunction Collapse << | Phase 4 | Unknown | November 2010 | China, Gansu ... more >> The Second Hospital of Lanzhou University Recruiting Lanzhou, Gansu, China, 730000 Contact: Ruixin Ma, Doctor +86 13893102690 mrxdr@sina.com Contact: Jing Yu, Professor +86 13893607559 yujing2304@126.com Principal Investigator: Jing Yu, Professor Sub-Investigator: Ruixin Ma, Doctor Collapse << |
NCT01630902 | Healthy | Phase 1 | Completed | - | India ... more >> Bio Evaluation Centre, Torrent Pharmaceuticals Ltd. Village Bhat, Gandhinagar, Gujarat, India Collapse << |
NCT00861016 | Hypertension | Phase 4 | Completed | - | - |
NCT01630655 | Healthy | Phase 1 | Completed | - | India ... more >> AXIS Clinicals Limited(formerly Trident Life Sciences Ltd.) Miyapur, Hyderabad, India, 500 050 Collapse << |
NCT00841880 | Hypertension | Phase 4 | Completed | - | Taiwan ... more >> Sanofi-Aventis Administrative Office Taipei, Taiwan Collapse << |
NCT00507845 | Hypertension | Phase 4 | Completed | - | Argentina ... more >> Sanofi-aventis administrative office Buenos Aires, Argentina Collapse << |
NCT02336607 | Hypertension | Not Applicable | Completed | - | - |
NCT01520285 | Hypertension | Phase 4 | Completed | - | China ... more >> Shanghai First People's Hospital Shanghai, China, 200000 Collapse << |
NCT02336607 | - | - | Completed | - | - |
NCT01136863 | Hypertension | Not Applicable | Completed | - | China ... more >> Fu Wai Hospital Beijing, China, 100037 Collapse << |
NCT00905333 | Healthy | Phase 1 | Completed | - | Brazil ... more >> Research Site Itatiba, SP, Brazil Research Site Americana, Brazil Collapse << |
NCT02311530 | Healthy | Not Applicable | Completed | - | - |
NCT02232269 | Food-Drug Interactions | Phase 1 | Completed | - | Canada, Ontario ... more >> Victoria Clinical Trials Centre London, Ontario, Canada Collapse << |
NCT02327247 | Healthy | Not Applicable | Completed | - | - |
靶点 | Description | IC50 |
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