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CAS No.: 3544-24-9
Synonyms: PARP-IN-1;3-ABA;3-amino Benzamide
INO-1001 is a potent inhibitor of PARP with IC50 of < 50 nM in CHO cells and a mediator of oxidant-induced myocyte dysfunction during reperfusion.
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00272415 | Melanoma | Phase 1 | Terminated | - | - |
NCT00271765 | Acute Myocardial Infarction | Phase 2 | Completed | - | United States, Florida ... more >> Holy Cross Hospital Fort Lauderdale, Florida, United States, 33308 United States, Indiana Porter Hospital Valparaiso, Indiana, United States, 46383 United States, Minnesota St. Paul Heart Clinic St. Paul, Minnesota, United States, 55102 United States, New Jersey Newark, New Jersey, United States United States, Ohio Toledo Hospital Toledo, Ohio, United States, 43606 United States, Pennsylvania Hospital of the University of Pennsylvania Philadelphia, Pennsylvania, United States United States, South Dakota Black Hills Cardiovascular Research Rapid City, South Dakota, United States, 57701 United States, Vermont Burlington, Vermont, United States United States, Virginia Sentara Norfolk General Hospital Norfolk, Virginia, United States United States, West Virginia West Virginia University Morgantown, West Virginia, United States, 26506 Israel Rambam Medical Center Haifa, Israel, 31096 Meir Medical Center Kfar Saba, Israel, 95847 Hasharon Medical Center Petach Tikva, Israel, 49100 Rabin Medical Center Petach Tikva, Israel, 49100 Rehovot, Israel Assaf Harofe Medical Centre Zerifin, Israel Collapse << |
NCT00271167 | Heart Diseases ... more >> Postoperative Complications Collapse << | Phase 2 | Terminated(It was determined t... more >>hat the study was not appropriate for demonstrating therapeutic benefit in the cardiopulmonary bypass patient population.) Collapse << | - | United States, Massachusetts ... more >> Beth Israel Deaconess Medical Center Boston, Massachusetts, United States, 02215 United States, Oklahoma University of Oklahoma Oklahoma, Oklahoma, United States, 73152 United States, Pennsylvania University of Pennsylvania Philadelphia, Pennsylvania, United States, 19104 United States, South Dakota Rapid City Regional Hospital Rapid City, South Dakota, United States United States, Texas Methodist Hospital Houston, Texas, United States, 77030 Australia, New South Wales Sydney, New South Wales, Australia Australia, South Australia Ashford Cardiac Clinic / Adelaide Cardiac Adelaide, South Australia, Australia Australia, Victoria St. Vincent's Hospital Melbourne, Victoria, Australia, 3065 Australia, Western Australia Royal Perth Hospital Perth, Western Australia, Australia, 6000 India Care Hospital Hyderabad, India Escorts Heart Institute and Research Centre New Delhi, India, 110029 Israel Wolfson Medical Centre Holon, Israel, 58100 Jerusalem, Israel Collapse << |
实验方案
技术信息
CAS号 | 3544-24-9 | 储存条件 |
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分子式 | C7H8N2O | 运输 | 蓝冰 | |||||
分子量 | 136.15 | 别名 | PARP-IN-1;3-ABA;3-amino Benzamide;3-(Aminocarbonyl) Aniline;3-Carboxamidoaniline | |||||
溶解度 |
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动物实验配方 |