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CAS No.: 1415558-82-5

2-Keto Crizotinib Catalog No. CSN22484

Synonyms: PF-06260182

PF-06260182 is a lactam metabolite of crizotinib.

规格 价格 促销价格 库存 数量
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靶点选择性

生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02511184ALK-positive Advanced NSCLCPhase 1Terminated(Decision based on t... more >>he low enrollment mainly due to high efficacy drugs available in 1st line ALK-positive NSCLC (eg alectinib), not due to any safety concerns) Collapse <<-United States, Alabama ... more >> University of Alabama at Birmingham Birmingham, Alabama, United States, 35233 University of Alabama at Birmingham, IDS Pharmacy Birmingham, Alabama, United States, 35249 University of Alabama at Birmingham Birmingham, Alabama, United States, 35249 United States, California City of Hope National Medical Center Duarte, California, United States, 91010 UC San Diego Moores Cancer Center - Investigational Drug Services La Jolla, California, United States, 92037-0845 UC San Diego Medical Center - La Jolla(Thornton Hospital) La Jolla, California, United States, 92037 University Of California / San Diego Moores Cancer Center La Jolla, California, United States, 92093 UC San Diego Medical Center - Hillcrest San Diego, California, United States, 92103 United States, Georgia Emory University Hospital Midtown Atlanta, Georgia, United States, 30308 Emory University Hospital Atlanta, Georgia, United States, 30322 The Emory Clinic Atlanta, Georgia, United States, 30322 Winship Cancer Institute of Emory University Atlanta, Georgia, United States, 30322 United States, Ohio The Cleveland Clinic Foundation Cleveland, Ohio, United States, 44195 United States, Washington Swedish Cancer Institute Seattle, Washington, United States, 98104 Swedish Investigational Drug Services Pharmacy Seattle, Washington, United States, 98104 Collapse <<
    NCT01549574HealthyPhase 1Completed-Belgium ... more >> Pfizer Investigational Site Bruxelles, Belgium, B-1070 Collapse <<
    NCT01419041Renal ImpairmentPhase 1Completed-United States, California ... more >> Pfizer Investigational Site Anaheim, California, United States, 92801 United States, Florida Pfizer Investigational Site DeLand, Florida, United States, 32720 United States, Minnesota Pfizer Investigational Site Saint Paul, Minnesota, United States, 55114 Collapse <<
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实验方案

技术信息

CAS号 1415558-82-5 储存条件
分子式 C21H20Cl2FN5O2 运输 蓝冰
分子量 464.32 别名 PF-06260182

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