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CAS No.: 289656-45-7
Synonyms: ICA-17043
Senicapoc is a potent and selective Gardos channel blocker and blocks Ca(2+)-induced rubidium flux from human RBCs/ inhibited RBC dehydration with IC50s of 11 nM/30 nM, respectively.
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00102791 | Sickle Cell Disease | Phase 3 | Terminated(Because of the low ... more >>probability of achieving the primary endpoint.) Collapse << | - | - |
NCT00294541 | Sickle Cell Disease ... more >> Sickle Cell Anemia Collapse << | Phase 3 | Terminated(Lack of efficacy de... more >>monstrated in study ICA-17043-10) Collapse << | - | - |
NCT00040677 | Sickle Cell Disease ... more >> Sickle Cell Anemia Collapse << | Phase 2 | Completed | - | United States, Alabama ... more >> Study Site Birmingham, Alabama, United States United States, California Study Site Oakland, California, United States Study Site San Francisco, California, United States United States, District of Columbia Study Site Washington, District of Columbia, United States United States, Georgia Study Site Augusta, Georgia, United States United States, Illinois Study Site Chicago, Illinois, United States United States, Maryland Study Site Baltimore, Maryland, United States United States, Massachusetts Study Site Boston, Massachusetts, United States United States, Michigan Study Site Detroit, Michigan, United States United States, Mississippi Study Site Jackson, Mississippi, United States United States, New York Study Site Brooklyn, New York, United States Study Site New York, New York, United States United States, North Carolina Study Site Chapel Hill, North Carolina, United States Study Site Durham, North Carolina, United States United States, Pennsylvania Study Site Philadelphia, Pennsylvania, United States Study Site Pittsburgh, Pennsylvania, United States United States, Tennessee Study Site Nashville, Tennessee, United States United States, Texas Study Site Houston, Texas, United States United States, Virginia Study Site Richmond, Virginia, United States Collapse << |
实验方案
技术信息
CAS号 | 289656-45-7 | 储存条件 |
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分子式 | C20H15F2NO | 运输 | 蓝冰 | |||
分子量 | 323.34 | 别名 | ICA-17043 | |||
溶解度 |
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动物实验配方 |