400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / Epigenetics / HDAC / 贝利司他
CAS No.: 866323-14-0
Synonyms: PXD101;PX105684;NSC726630
Belinostat is a pan-HDAC inhibitor with IC50 of 27 nM, with activity demonstrated in cisplatin-resistant tumors.
生物活性
靶点 | HDAC IC50:27nM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03432741 | Breast Adenocarcinoma ... more >> Recurrent Breast Carcinoma Recurrent Hodgkin Lymphoma Recurrent Mycosis Fungoides Recurrent Non-Hodgkin Lymphoma Recurrent Primary Cutaneous T-Cell Non-Hodgkin Lymphoma Refractory Hodgkin Lymphoma Refractory Mycosis Fungoides Refractory Nodal Marginal Zone Lymphoma Refractory Non-Hodgkin Lymphoma Refractory Primary Cutaneous T-Cell Non-Hodgkin Lymphoma Stage IV Breast Cancer AJCC v6 and v7 Collapse << | Phase 1 | Recruiting | May 1, 2019 | United States, Minnesota ... more >> Mayo Clinic Recruiting Rochester, Minnesota, United States, 55905 Contact: Clinical Trials Referral Office 855-776-0015 Principal Investigator: Grzegorz S. Nowakowski Collapse << |
NCT00131261 | Multiple Myeloma | Phase 2 | Completed | - | United States, California ... more >> James Berenson, MD, Inc West Hollywood, California, United States, 90069 United States, Florida H. Lee Moffitt Cancer Center Tampa, Florida, United States, 33612 United States, Illinois Northwestern University Chicago, Illinois, United States, 60611 United States, New York Research Facility New York, New York, United States, 10021 Denmark Rigshospitalet Copenhagen, Denmark, 2100 Norway Research Facility Bergen, Norway, N-5021 Research Facility Oslo, Norway, N-0407 Research Facility Trondheim, Norway, N-7006 United Kingdom Christie Hospital NHS Trust Manchester, United Kingdom, M20 4BX The Royal Marsden NHS Trust Surrey, United Kingdom, SM2 5NG Collapse << |
NCT00354185 | Adult Nasal Type Extranodal NK... more >>/T-cell Lymphoma Anaplastic Large Cell Lymphoma Angioimmunoblastic T-cell Lymphoma Extranodal Marginal Zone B-cell Lymphoma of Mucosa-associated Lymphoid Tissue Intraocular Lymphoma Nodal Marginal Zone B-cell Lymphoma Post-transplant Lymphoproliferative Disorder Recurrent Adult Burkitt Lymphoma Recurrent Adult Diffuse Large Cell Lymphoma Recurrent Adult Diffuse Mixed Cell Lymphoma Recurrent Adult Diffuse Small Cleaved Cell Lymphoma Recurrent Adult Grade III Lymphomatoid Granulomatosis Recurrent Adult Hodgkin Lymphoma Recurrent Adult Immunoblastic Large Cell Lymphoma Recurrent Adult Lymphoblastic Lymphoma Recurrent Adult T-cell Leukemia/Lymphoma Recurrent Cutaneous T-cell Non-Hodgkin Lymphoma Recurrent Grade 1 Follicular Lymphoma Recurrent Grade 2 Follicular Lymphoma Recurrent Grade 3 Follicular Lymphoma Recurrent Mantle Cell Lymphoma Recurrent Marginal Zone Lymphoma Recurrent Mycosis Fungoides/Sezary Syndrome Recurrent Small Lymphocytic Lymphoma Small Intestine Lymphoma Splenic Marginal Zone Lymphoma Stage III Adult Burkitt Lymphoma Stage III Adult Diffuse Large Cell Lymphoma Stage III Adult Diffuse Mixed Cell Lymphoma Stage III Adult Diffuse Small Cleaved Cell Lymphoma Stage III Adult Hodgkin Lymphoma Stage III Adult Immunoblastic Large Cell Lymphoma Stage III Adult Lymphoblastic Lymphoma Stage III Adult T-cell Leukemia/Lymphoma Stage III Cutaneous T-cell Non-Hodgkin Lymphoma Stage III Grade 1 Follicular Lymphoma Stage III Grade 2 Follicular Lymphoma Stage III Grade 3 Follicular Lymphoma Stage III Mantle Cell Lymphoma Stage III Marginal Zone Lymphoma Stage III Mycosis Fungoides/Sezary Syndrome Stage III Small Lymphocytic Lymphoma Stage IV Adult Burkitt Lymphoma Stage IV Adult Diffuse Large Cell Lymphoma Stage IV Adult Diffuse Mixed Cell Lymphoma Stage IV Adult Diffuse Small Cleaved Cell Lymphoma Stage IV Adult Hodgkin Lymphoma Stage IV Adult Immunoblastic Large Cell Lymphoma Stage IV Adult Lymphoblastic Lymphoma Stage IV Adult T-cell Leukemia/Lymphoma Stage IV Cutaneous T-cell Non-Hodgkin Lymphoma Stage IV Grade 1 Follicular Lymphoma Stage IV Grade 2 Follicular Lymphoma Stage IV Grade 3 Follicular Lymphoma Stage IV Mantle Cell Lymphoma Stage IV Marginal Zone Lymphoma Stage IV Mycosis Fungoides/Sezary Syndrome Stage IV Small Lymphocytic Lymphoma Unspecified Adult Solid Tumor, Protocol Specific Waldenström Macroglobulinemia Collapse << | Phase 1 | Terminated | - | United States, Wisconsin ... more >> University of Wisconsin Hospital and Clinics Madison, Wisconsin, United States, 53792 Collapse << |
实验方案
技术信息
CAS号 | 866323-14-0 | 储存条件 |
|
|||||
分子式 | C15H14N2O4S | 运输 | 蓝冰 | |||||
分子量 | 318.35 | 别名 | PXD101;PX105684;NSC726630;brand name: Beleodaq;贝利司他 | |||||
溶解度 |
|
动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03432741 | Breast Adenocarcinoma ... more >> Recurrent Breast Carcinoma Recurrent Hodgkin Lymphoma Recurrent Mycosis Fungoides Recurrent Non-Hodgkin Lymphoma Recurrent Primary Cutaneous T-Cell Non-Hodgkin Lymphoma Refractory Hodgkin Lymphoma Refractory Mycosis Fungoides Refractory Nodal Marginal Zone Lymphoma Refractory Non-Hodgkin Lymphoma Refractory Primary Cutaneous T-Cell Non-Hodgkin Lymphoma Stage IV Breast Cancer AJCC v6 and v7 Collapse << | Phase 1 | Recruiting | May 1, 2019 | United States, Minnesota ... more >> Mayo Clinic Recruiting Rochester, Minnesota, United States, 55905 Contact: Clinical Trials Referral Office 855-776-0015 Principal Investigator: Grzegorz S. Nowakowski Collapse << |
NCT00131261 | Multiple Myeloma | Phase 2 | Completed | - | United States, California ... more >> James Berenson, MD, Inc West Hollywood, California, United States, 90069 United States, Florida H. Lee Moffitt Cancer Center Tampa, Florida, United States, 33612 United States, Illinois Northwestern University Chicago, Illinois, United States, 60611 United States, New York Research Facility New York, New York, United States, 10021 Denmark Rigshospitalet Copenhagen, Denmark, 2100 Norway Research Facility Bergen, Norway, N-5021 Research Facility Oslo, Norway, N-0407 Research Facility Trondheim, Norway, N-7006 United Kingdom Christie Hospital NHS Trust Manchester, United Kingdom, M20 4BX The Royal Marsden NHS Trust Surrey, United Kingdom, SM2 5NG Collapse << |
NCT00354185 | Adult Nasal Type Extranodal NK... more >>/T-cell Lymphoma Anaplastic Large Cell Lymphoma Angioimmunoblastic T-cell Lymphoma Extranodal Marginal Zone B-cell Lymphoma of Mucosa-associated Lymphoid Tissue Intraocular Lymphoma Nodal Marginal Zone B-cell Lymphoma Post-transplant Lymphoproliferative Disorder Recurrent Adult Burkitt Lymphoma Recurrent Adult Diffuse Large Cell Lymphoma Recurrent Adult Diffuse Mixed Cell Lymphoma Recurrent Adult Diffuse Small Cleaved Cell Lymphoma Recurrent Adult Grade III Lymphomatoid Granulomatosis Recurrent Adult Hodgkin Lymphoma Recurrent Adult Immunoblastic Large Cell Lymphoma Recurrent Adult Lymphoblastic Lymphoma Recurrent Adult T-cell Leukemia/Lymphoma Recurrent Cutaneous T-cell Non-Hodgkin Lymphoma Recurrent Grade 1 Follicular Lymphoma Recurrent Grade 2 Follicular Lymphoma Recurrent Grade 3 Follicular Lymphoma Recurrent Mantle Cell Lymphoma Recurrent Marginal Zone Lymphoma Recurrent Mycosis Fungoides/Sezary Syndrome Recurrent Small Lymphocytic Lymphoma Small Intestine Lymphoma Splenic Marginal Zone Lymphoma Stage III Adult Burkitt Lymphoma Stage III Adult Diffuse Large Cell Lymphoma Stage III Adult Diffuse Mixed Cell Lymphoma Stage III Adult Diffuse Small Cleaved Cell Lymphoma Stage III Adult Hodgkin Lymphoma Stage III Adult Immunoblastic Large Cell Lymphoma Stage III Adult Lymphoblastic Lymphoma Stage III Adult T-cell Leukemia/Lymphoma Stage III Cutaneous T-cell Non-Hodgkin Lymphoma Stage III Grade 1 Follicular Lymphoma Stage III Grade 2 Follicular Lymphoma Stage III Grade 3 Follicular Lymphoma Stage III Mantle Cell Lymphoma Stage III Marginal Zone Lymphoma Stage III Mycosis Fungoides/Sezary Syndrome Stage III Small Lymphocytic Lymphoma Stage IV Adult Burkitt Lymphoma Stage IV Adult Diffuse Large Cell Lymphoma Stage IV Adult Diffuse Mixed Cell Lymphoma Stage IV Adult Diffuse Small Cleaved Cell Lymphoma Stage IV Adult Hodgkin Lymphoma Stage IV Adult Immunoblastic Large Cell Lymphoma Stage IV Adult Lymphoblastic Lymphoma Stage IV Adult T-cell Leukemia/Lymphoma Stage IV Cutaneous T-cell Non-Hodgkin Lymphoma Stage IV Grade 1 Follicular Lymphoma Stage IV Grade 2 Follicular Lymphoma Stage IV Grade 3 Follicular Lymphoma Stage IV Mantle Cell Lymphoma Stage IV Marginal Zone Lymphoma Stage IV Mycosis Fungoides/Sezary Syndrome Stage IV Small Lymphocytic Lymphoma Unspecified Adult Solid Tumor, Protocol Specific Waldenström Macroglobulinemia Collapse << | Phase 1 | Terminated | - | United States, Wisconsin ... more >> University of Wisconsin Hospital and Clinics Madison, Wisconsin, United States, 53792 Collapse << |
NCT00303953 | Recurrent Adult Burkitt Lympho... more >>ma Recurrent Adult Diffuse Large Cell Lymphoma Collapse << | Phase 2 | Completed | - | - |
NCT00926640 | Carcinoma Neuroendocrine ... more >> Small Cell Lung Carcinoma Malignant Epithelial Neoplasms Collapse << | Phase 1 | Completed | - | United States, Maryland ... more >> National Institutes of Health Clinical Center, 9000 Rockville Pike Bethesda, Maryland, United States, 20892 Collapse << |
NCT00351975 | Accelerated Phase of Disease ... more >> Adult Acute Myeloid Leukemia With Inv(16)(p13.1q22); CBFB-MYH11 Adult Acute Myeloid Leukemia With t(16;16)(p13.1;q22); CBFB-MYH11 Adult Acute Myeloid Leukemia With t(8;21)(q22;q22); RUNX1-RUNX1T1 Adult Acute Myeloid Leukemia With t(9;11)(p22;q23); MLLT3-MLL Adult Acute Promyelocytic Leukemia With t(15;17)(q22;q12); PML-RARA Atypical Chronic Myeloid Leukemia, BCR-ABL1 Negative Blastic Phase Chronic Myelogenous Leukemia, BCR-ABL1 Positive Chronic Myelomonocytic Leukemia de Novo Myelodysplastic Syndrome Myelodysplastic/Myeloproliferative Neoplasm, Unclassifiable Philadelphia Chromosome Negative, BCR-ABL1 Positive Chronic Myelogenous Leukemia Previously Treated Myelodysplastic Syndrome Primary Myelofibrosis Recurrent Adult Acute Lymphoblastic Leukemia Recurrent Adult Acute Myeloid Leukemia Recurrent Disease Secondary Acute Myeloid Leukemia Secondary Myelodysplastic Syndrome Collapse << | Phase 1 | Completed | - | United States, Illinois ... more >> University of Chicago Comprehensive Cancer Center Chicago, Illinois, United States, 60637 United States, Wisconsin University of Wisconsin Hospital and Clinics Madison, Wisconsin, United States, 53792 Canada, Ontario University Health Network-Princess Margaret Hospital Toronto, Ontario, Canada, M5G 2M9 New Zealand Princess Margaret Hospital Cashmere, Canterbury, New Zealand, 8022 Collapse << |
NCT00365053 | Advanced Malignant Mesotheliom... more >>a Epithelial Mesothelioma Recurrent Malignant Mesothelioma Sarcomatous Mesothelioma Collapse << | Phase 2 | Completed | - | United States, California ... more >> City of Hope Duarte, California, United States, 91010 Collapse << |
NCT00303953 | - | - | Completed | - | - |
NCT00357032 | Adult Acute Myeloid Leukemia W... more >>ith 11q23 (MLL) Abnormalities Adult Acute Myeloid Leukemia With Del(5q) Adult Acute Myeloid Leukemia With Inv(16)(p13;q22) Adult Acute Myeloid Leukemia With t(15;17)(q22;q12) Adult Acute Myeloid Leukemia With t(16;16)(p13;q22) Adult Acute Myeloid Leukemia With t(8;21)(q22;q22) Recurrent Adult Acute Myeloid Leukemia Untreated Adult Acute Myeloid Leukemia Collapse << | Phase 2 | Completed | - | United States, California ... more >> City of Hope Duarte, California, United States, 91010 Collapse << |
NCT00365053 | - | - | Completed | - | - |
NCT00348985 | Adult Grade III Lymphomatoid G... more >>ranulomatosis Anaplastic Large Cell Lymphoma Angioimmunoblastic T-cell Lymphoma Extranodal Marginal Zone B-cell Lymphoma of Mucosa-associated Lymphoid Tissue Intraocular Lymphoma Nodal Marginal Zone B-cell Lymphoma Post-transplant Lymphoproliferative Disorder Primary Central Nervous System Hodgkin Lymphoma Primary Central Nervous System Non-Hodgkin Lymphoma Recurrent Adult Burkitt Lymphoma Recurrent Adult Diffuse Large Cell Lymphoma Recurrent Adult Diffuse Mixed Cell Lymphoma Recurrent Adult Diffuse Small Cleaved Cell Lymphoma Recurrent Adult Grade III Lymphomatoid Granulomatosis Recurrent Adult Hodgkin Lymphoma Recurrent Adult Immunoblastic Large Cell Lymphoma Recurrent Adult Lymphoblastic Lymphoma Recurrent Adult T-cell Leukemia/Lymphoma Recurrent Cutaneous T-cell Non-Hodgkin Lymphoma Recurrent Grade 1 Follicular Lymphoma Recurrent Grade 2 Follicular Lymphoma Recurrent Grade 3 Follicular Lymphoma Recurrent Mantle Cell Lymphoma Recurrent Marginal Zone Lymphoma Recurrent Mycosis Fungoides/Sezary Syndrome Recurrent Small Lymphocytic Lymphoma Splenic Marginal Zone Lymphoma Stage III Adult Burkitt Lymphoma Stage III Adult Diffuse Large Cell Lymphoma Stage III Adult Diffuse Mixed Cell Lymphoma Stage III Adult Diffuse Small Cleaved Cell Lymphoma Stage III Adult Hodgkin Lymphoma Stage III Adult Immunoblastic Large Cell Lymphoma Stage III Adult Lymphoblastic Lymphoma Stage III Adult T-cell Leukemia/Lymphoma Stage III Cutaneous T-cell Non-Hodgkin Lymphoma Stage III Grade 1 Follicular Lymphoma Stage III Grade 2 Follicular Lymphoma Stage III Grade 3 Follicular Lymphoma Stage III Mantle Cell Lymphoma Stage III Marginal Zone Lymphoma Stage III Mycosis Fungoides/Sezary Syndrome Stage III Small Lymphocytic Lymphoma Stage IV Adult Burkitt Lymphoma Stage IV Adult Diffuse Large Cell Lymphoma Stage IV Adult Diffuse Mixed Cell Lymphoma Stage IV Adult Diffuse Small Cleaved Cell Lymphoma Stage IV Adult Hodgkin Lymphoma Stage IV Adult Immunoblastic Large Cell Lymphoma Stage IV Adult Lymphoblastic Lymphoma Stage IV Adult T-cell Leukemia/Lymphoma Stage IV Cutaneous T-cell Non-Hodgkin Lymphoma Stage IV Grade 1 Follicular Lymphoma Stage IV Grade 2 Follicular Lymphoma Stage IV Grade 3 Follicular Lymphoma Stage IV Mantle Cell Lymphoma Stage IV Marginal Zone Lymphoma Stage IV Mycosis Fungoides/Sezary Syndrome Stage IV Small Lymphocytic Lymphoma Unspecified Adult Solid Tumor, Protocol Specific Waldenström Macroglobulinemia Collapse << | Phase 1 | Completed | - | United States, Colorado ... more >> University of Colorado Denver, Colorado, United States, 80217-3364 Collapse << |
NCT00357032 | - | - | Completed | - | - |
NCT00589290 | - | - | Completed | - | - |
NCT00413322 | Tumor | Phase 1 | Completed | - | United States, Arizona ... more >> Mayo Clinic Arizona Scottsdale, Arizona, United States, 85259 United States, Nebraska University of Nebraska Omaha, Nebraska, United States, 68198-7680 United States, New Hampshire Portsmouth Regional Hospital Hematology/Oncology Clinic Portsmouth, New Hampshire, United States, 03801 Collapse << |
NCT00589290 | Thymoma Thymi... more >>c Carcinoma Collapse << | Phase 2 | Completed | - | United States, Indiana ... more >> Indiana University Cancer Center Indianapolis, Indiana, United States, 46202-5262 United States, Maryland National Institutes of Health Clinical Center, 9000 Rockville Pike Bethesda, Maryland, United States, 20892 Collapse << |
NCT00873119 | Carcinoma of Unknown Primary | Phase 2 | Completed | - | United States, Florida ... more >> Florida Cancer Specialists Fort Myers, Florida, United States, 33619 United States, Georgia Northwest Georgia Oncology Centers Marietta, Georgia, United States, 30060 United States, Louisiana Baton Rouge Medical Center Baton Rouge, Louisiana, United States, 70809 United States, Maryland Center for Cancers and Blood Disorders Bethesda, Maryland, United States, 20817 United States, Missouri Research Medical Center Kansas City, Missouri, United States, 64132 United States, Ohio Oncology Hematology Care Inc. Cincinnati, Ohio, United States, 45242 United States, South Carolina South Carolina Oncology Associates Columbia, South Carolina, United States, 29210 United States, Tennessee Chattanooga Oncology & Hematology Associates, PC Chattanooga, Tennessee, United States, 37404 Tennessee Oncology Sarah Cannon Research Nashville, Tennessee, United States, 37203 United States, Texas South Texas Oncology and Hematology San Antonio, Texas, United States, 78258 United States, Virginia Virginia Cancer Institute Richmond, Virginia, United States, 23230 Denmark H:S Rigshospital, The Finsen Centre Copenhagen, Denmark, DK-2100 France CRLCC Francois Baclesse, Oncologie medicale Caen, France, 14000 Centre Oscar Lambert Lille, France, 59020 Centre Léon Bérard, Oncologie Lyon, France, 69008 Centre Eugène Marquis Rennes cedex, France, 35042 Centre Henri Becquerel, Oncologie Médicale Rouen, France, 76038 Institut de Cancerologie de la Loire Saint Priest en Jarez, France, 42270 Institut Gustave Roussy IGR Villejuif cedex, France, 94805 Germany Carl-Gustav-Carus Medicinische Klinik und Poliklinik I Dresden, Germany, 01307 Kliniken Essen-Mitte Essen, Germany, 45136 ASKLEPIOS Klinik Altona Hamburg, Germany, 22763 Ostholstein-Onkologie Oldenburg in Holstein, Germany, 23758 Collapse << |
NCT00431340 | Multiple Myeloma | Phase 2 | Terminated(Terminated due to d... more >>ose limiting toxicity) Collapse << | - | United States, California ... more >> Oncotherapeutics West Hollywood, California, United States, 90069 United States, Maryland Center for cancer and blood disorders Bethesda, Maryland, United States, 20817 United States, Texas Baylor University Medical Center Dallas, Texas, United States, 75246 Collapse << |
NCT00873119 | - | - | Completed | - | - |
NCT01075425 | Acute Lymphocytic Leukemia ... more >> Acute Myeloid Leukemia Myelodysplastic Syndrome Chronic Myelogenous Leukemia Collapse << | Phase 1 | Completed | - | United States, Texas ... more >> M D Anderson Cancer Center Houston, Texas, United States, 77030 United States, Virginia Virginia Commonwealth University Richmond, Virginia, United States, 23298 Collapse << |
NCT00993616 | - | - | Completed | - | - |
NCT00334789 | Adult Solid Neoplasm | Phase 1 | Completed | - | United States, California ... more >> City of Hope Comprehensive Cancer Center Duarte, California, United States, 91010 USC / Norris Comprehensive Cancer Center Los Angeles, California, United States, 90033 University of California Davis Comprehensive Cancer Center Sacramento, California, United States, 95817 City of Hope South Pasadena South Pasadena, California, United States, 91030 United States, Pennsylvania University of Pittsburgh Cancer Institute (UPCI) Pittsburgh, Pennsylvania, United States, 15232 Collapse << |
NCT01100944 | Thymoma Thymi... more >>c Carcinoma Collapse << | Phase 1 Phase 2 | Terminated(Principal investiga... more >>tor left the National Institutes of Health (NIH).) Collapse << | - | United States, Maryland ... more >> National Institutes of Health Clinical Center, 9000 Rockville Pike Bethesda, Maryland, United States, 20892 Collapse << |
NCT00878722 | Acute Myeloid Leukemia | Phase 1 Phase 2 | Completed | - | France ... more >> CHU Lapeyronie Montpellier, France, 34295 Hôpital St. Louis Paris, France, 75475 Germany Uniklinik Homburg Homburg, Germany, 66424 Uni Hospital Marburg Marburg, Germany, 35043 Universitätsklinikum Ulm Ulm, Germany, 89081 United Kingdom Christie Hospital NHS Trust Manchester, United Kingdom, M20 4BX Collapse << |
NCT00357162 | de Novo Myelodysplastic Syndro... more >>mes Previously Treated Myelodysplastic Syndromes Secondary Myelodysplastic Syndromes Collapse << | Phase 2 | Completed | - | United States, Minnesota ... more >> Mayo Clinic Rochester, Minnesota, United States, 55905 Collapse << |
NCT00993616 | Brenner Tumor ... more >> Fallopian Tube Cancer Ovarian Clear Cell Cystadenocarcinoma Ovarian Endometrioid Adenocarcinoma Ovarian Mixed Epithelial Carcinoma Ovarian Mucinous Cystadenocarcinoma Ovarian Serous Cystadenocarcinoma Ovarian Undifferentiated Adenocarcinoma Primary Peritoneal Cavity Cancer Recurrent Ovarian Epithelial Cancer Collapse << | Phase 2 | Completed | - | - |
NCT01310244 | Stage IV Non-small Cell Lung C... more >>ancer Collapse << | Phase 1 Phase 2 | Completed | - | United States, Alabama ... more >> Clearview Cancer Institute (CCI) Huntsville, Alabama, United States, 35805 United States, California Sarcoma Oncology Center Santa Monica, California, United States, 90403 United States, Florida University Cancer Insitute Boynton Beach, Florida, United States, 33426 United States, Missouri Washington University School of Medicine St. Louis, Missouri, United States, 63110 Collapse << |
NCT00301756 | Fallopian Tube Carcinoma ... more >> Primary Peritoneal Carcinoma Recurrent Borderline Ovarian Surface Epithelial-Stromal Tumor Recurrent Ovarian Carcinoma Stage III Borderline Ovarian Surface Epithelial-Stromal Tumor Stage III Ovarian Cancer Stage IV Borderline Ovarian Surface Epithelial-Stromal Tumor Stage IV Ovarian Cancer Collapse << | Phase 2 | Completed | - | Canada, Ontario ... more >> Juravinski Cancer Centre at Hamilton Health Sciences Hamilton, Ontario, Canada, L8V 5C2 Odette Cancer Centre- Sunnybrook Health Sciences Centre Toronto, Ontario, Canada, M4N 3M5 University Health Network Princess Margaret Cancer Center P2C Toronto, Ontario, Canada, M5G 2M9 University Health Network-Princess Margaret Hospital Toronto, Ontario, Canada, M5G 2M9 Collapse << |
NCT02532192 | Lymphoma | Phase 1 | Withdrawn(Withdrawal of study ... more >>support.) Collapse << | - | - |
NCT00321594 | Adult Primary Hepatocellular C... more >>arcinoma Advanced Adult Primary Liver Cancer Localized Unresectable Adult Primary Liver Cancer Recurrent Adult Primary Liver Cancer Collapse << | Phase 1 Phase 2 | Completed | - | United States, Wisconsin ... more >> University of Wisconsin Hospital and Clinics Madison, Wisconsin, United States, 53792 Singapore Cancer Therapeutics Research Group Singapore, Singapore, 119074 Collapse << |
NCT00357162 | - | - | Completed | - | - |
NCT00321594 | - | - | Completed | - | - |
NCT00878800 | Dose Escalation: Solid Tumors ... more >> MTD: Soft Tissue Sarcomas Collapse << | Phase 1 Phase 2 | Completed | - | Denmark ... more >> Herlev Hospital, Department of Oncology Herlev, Denmark, DK-2730 Århus Hospital, Department of Oncology Århus, Denmark, DK-8000 C United Kingdom The Royal Marsden NHS Trust, Cancer Research Surrey, United Kingdom, SM2 5PT Surrey Collapse << |
NCT01100944 | - | - | Terminated(Principal investiga... more >>tor left the National Institutes of Health (NIH).) Collapse << | - | - |
NCT00878722 | - | - | Completed | - | - |
NCT00878800 | - | - | Completed | - | - |
NCT00274651 | Cutaneous T-Cell Lymphoma ... more >> Peripheral T-Cell Lymphoma Non-Hodgkin's Lymphoma Collapse << | Phase 2 | Terminated(Enrollment stopped ... more >>prior to reaching expected number of patients, study had accumulated sufficient data to allow a registration study in PTCL (PXD101-CLN-19)) Collapse << | - | United States, California ... more >> Leland Stanford Junior University Stanford, California, United States, 94305 United States, Connecticut Yale University School of Medicine New Haven, Connecticut, United States, 06520 United States, Kansas Kansas City Cancer Center Lenexa, Kansas, United States, 66214 United States, Massachusetts Dana Farber Cancer Institute Boston, Massachusetts, United States, 02115 Boston University Medical Center Boston, Massachusetts, United States, 02118 United States, New York NYU Medical Center New York, New York, United States, 10016 United States, Ohio Cleveland Clinic Foundation Cleveland, Ohio, United States, 44195 United States, Texas MD Anderson Cancer Center Houston, Texas, United States, 77030 France Hopitaux du Haut Leveque Pessac, France, 33604 Hospital Purpan Toulouse, France, 31059 Germany Universitatsklinikum Essen Essen, Germany, 45147 Israel Hadassah University Hospital Ein Kerem Jerusalem, Israel, 91120 Rabin Medical Center Petach Tikva, Israel, 49100 Thailand Songklanagarind Hospital, Prince of Songkla University Hat Yai, Thailand, 90110 King Chulalongkorn Memorial Hospital Patumwan, Thailand, 10330 Collapse << |
NCT00421889 | Ovarian Cancer ... more >> Epithelial Ovarian Cancer Fallopian Tube Cancer Bladder Cancer Collapse << | Phase 1 Phase 2 | Completed | - | United States, California ... more >> Gynecologic Oncology Associates Newport Beach, California, United States, 92663 United States, Florida Research Facility Orlando, Florida, United States, 32804 United States, Louisiana Hematology and Oncology Specialists, LLC Covington, Louisiana, United States, 70433 Hematology & Oncology Specialists, LLC Metairie, Louisiana, United States, 70006 United States, Maryland Greater Baltimore Medical Center Baltimore, Maryland, United States, 21204 United States, Massachusetts Massachusetts General Hospital Cancer Center Boston, Massachusetts, United States, 02114 United States, Rhode Island Women & Infants Hospital of Rhode Island Providence, Rhode Island, United States, 02905 Denmark The Finsen Center, Rigshospitalet Copenhagen, Denmark, 2100 Research Facility, Herlev University Hospital Herlev, Denmark, 2730 United Kingdom The Beatson West of Scotland Cancer Centre Glasgow, United Kingdom, G120YN The Royal Marsden NHS Trust Surrey, United Kingdom, SM2 5PT Collapse << |
NCT00274651 | - | - | Terminated(Enrollment stopped ... more >>prior to reaching expected number of patients, study had accumulated sufficient data to allow a registration study in PTCL (PXD101-CLN-19)) Collapse << | - | - |
NCT01686165 | Anaplastic Large Cell Lymphoma... more >> Recurrent Adult Diffuse Large Cell Lymphoma Recurrent Mantle Cell Lymphoma Collapse << | Phase 2 | Completed | - | United States, Arizona ... more >> University of Arizona Cancer Center Tucson, Arizona, United States, 85724-5024 Collapse << |
NCT02875002 | Relapsed and Refractory Aggres... more >>sive B- and T-cell Lymphomas Lymphoma Collapse << | Phase 1 | Withdrawn | September 2018 | United States, Connecticut ... more >> Yale Cancer Center New Haven, Connecticut, United States, 06511 United States, Maryland Sidney Kimmel Comprehensive Cancer Baltimore, Maryland, United States, 21287 United States, Virginia Massey Cancer Center Richmond, Virginia, United States, 23298 Collapse << |
NCT00421889 | - | - | Completed | - | - |
NCT02701673 | Lymphoma | Phase 1 Phase 2 | Withdrawn | - | - |
NCT01686165 | - | - | Completed | - | - |
NCT00301756 | - | - | Completed | - | - |
NCT00413075 | Solid Tumor L... more >>ymphoma Collapse << | Phase 1 | Completed | - | United States, Connecticut ... more >> Yale New Haven Hospital New Haven, Connecticut, United States, 06520 United States, New York Columbia University - Herbert Irving Cancer Center New York, New York, United States, 01132 New York University Cancer Institute New York, New York, United States, 10016 United States, Texas M.D. Anderson Cancer Center Houston, Texas, United States, 77230-1402 Denmark Research Facility Copenhagen, Denmark United Kingdom Research Facility London, Surrey, United Kingdom, SW3 6JJ Collapse << |
NCT01188707 | Non Small Cell Lung Cancer | Phase 1 Phase 2 | Terminated(Dose over MTD reach... more >>ed) Collapse << | August 2012 | Denmark ... more >> Dept of Oncology Copenhagen University Hospital Herlev Herlev, Copenhagen, Denmark, 2730 Collapse << |
NCT01273155 | Neoplasms Lym... more >>phomas Collapse << | Phase 1 | Completed | - | United States, California ... more >> University of California, Davis Davis, California, United States, 95616 City of Hope National Medical Center Duarte, California, United States, 91010 USC Norris Cancer Center Los Angeles, California, United States United States, Georgia Emory University Atlanta, Georgia, United States, 30322-1102 United States, Maryland National Institutes of Health Clinical Center, 9000 Rockville Pike Bethesda, Maryland, United States, 20892 United States, Michigan Karmanos Cancer Institute Detroit, Michigan, United States, 48201 United States, New York Albert Einstein College of Medicine Bronx, New York, United States, 10461 Collapse << |
NCT01090830 | Non-Small-Cell Lung Carcinoma | Phase 1 Phase 2 | Terminated(Principal Investiga... more >>tor has left institution. IND withdrawn.) Collapse << | - | United States, Florida ... more >> Holy Cross Hospital, Inc Fort Lauderdale, Florida, United States, 33308 Collapse << |
NCT02137759 | Glioblastoma Multiforme of Bra... more >>in Collapse << | Phase 2 | Recruiting | June 2022 | United States, Georgia ... more >> Emory University/Winship Cancer Institute Recruiting Atlanta, Georgia, United States, 30322 Contact: Rikesh Patel 404-778-2981 rikesh.b.patel@emory.edu Contact: Lily Masoumy 404-778-1960 lily.masoumy@emory.edu United States, Maryland Johns Hopkins Sidney Kimmel Comprehensive Cancer Center Recruiting Baltimore, Maryland, United States, 21287 Contact: Matthias Holdhoff, MD, PhD 410-955-8837 mholdho1@jhmi.edu Collapse << |
NCT02381548 | Acute Myeloid Leukemia ... more >> Blast Phase Chronic Myelogenous Leukemia, BCR-ABL1 Positive Myelodysplastic Syndrome Previously Treated Myelodysplastic Syndrome Recurrent Adult Acute Myeloid Leukemia Recurrent Chronic Myelogenous Leukemia, BCR-ABL1 Positive Refractory Acute Myeloid Leukemia Refractory Chronic Myelogenous Leukemia, BCR-ABL1 Positive Secondary Acute Myeloid Leukemia Therapy-Related Acute Myeloid Leukemia Untreated Adult Acute Myeloid Leukemia Collapse << | Phase 1 | Terminated | - | United States, Florida ... more >> Moffitt Cancer Center Tampa, Florida, United States, 33612 United States, Virginia Virginia Commonwealth University/Massey Cancer Center Richmond, Virginia, United States, 23298 Collapse << |
NCT02737046 | Adult T-cell Leukemia-Lymphoma... more >> ATLL Collapse << | Phase 2 | Recruiting | November 2021 | United States, Florida ... more >> University of Miami Recruiting Miami, Florida, United States, 33136 Contact: Juan C Ramos, MD 305-243-6611 jramos2@med.miami.edu Principal Investigator: Juan C Ramos, MD Collapse << |
NCT01839097 | Peripheral T-cell Lymphoma | Phase 1 | Completed | - | United States, Connecticut ... more >> Yale University New Haven, Connecticut, United States, 06511 United States, Georgia Northeast Georgia Cancer Care, LLC Athens, Georgia, United States, 30607 United States, Minnesota Mayo Clinic Rochester, Minnesota, United States, 55905 United States, Missouri Washington University School of Medicine St. Louis, Missouri, United States, 63110 United States, New Jersey John Theurer Cancer Center at Hackensack University Medical Center Hackensack, New Jersey, United States, 07601 Hematology - Oncology Associates of Northern NJ P.A Morristown, New Jersey, United States, 07962 United States, New York Columbia University Medical Center/Center for Lymphiod Malignancies New York, New York, United States, 10019 United States, North Carolina Duke University Medical Center Durham, North Carolina, United States, 27705 Collapse << |
NCT01317927 | Solid Tumor H... more >>ematological Malignancy Collapse << | Phase 1 | Completed | - | United States, Utah ... more >> Huntsman Cancer Center, University of Utah Salt Lake City, Utah, United States, 84112 Collapse << |
NCT02680795 | Solid Tumors ... more >>Hematological Malignancies Collapse << | Phase 1 | Recruiting | June 2019 | United States, California ... more >> The Oncology Institute of Hope and Innovation Recruiting Whittier, California, United States Contact: Kirsten Bettino 562-693-4477 Principal Investigator: Richy Agajanian, MD United States, Ohio Gabrail Cancer Center Research Recruiting Canton, Ohio, United States, 44718 Contact: Carrie Smith 330-492-3345 Principal Investigator: Nashat Gabrail, MD Collapse << |
NCT01583777 | Advanced Cancer | Phase 1 | Completed | - | Spain ... more >> Hospital Universitario Madrid Sanchinarro Madrid, Spain, 28050 Collapse << |
NCT03772925 | Recurrent Acute Myeloid Leukem... more >>ia Recurrent Myelodysplastic Syndrome Refractory Acute Myeloid Leukemia Refractory Myelodysplastic Syndrome Collapse << | Phase 1 | Not yet recruiting | July 1, 2021 | - |
NCT00865969 | Peripheral T-cell Lymphoma | Phase 2 | Completed | - | - |
NCT02679131 | Relapsed/Refractory Solid Tumo... more >>rs/Hematological Malignancies Collapse << | Phase 1 | Terminated(Close out study wit... more >>hout completion of Cohort D; Severe Impairment (eGFR=15 to <30mL/min/1.73m²)) Collapse << | - | United States, California ... more >> Innovative Clinical Research Institute Whittier, California, United States, 90603 United States, Ohio Gabrail Cancer Center Research Canton, Ohio, United States, 44718 Collapse << |
NCT02142530 | Non-Hodgkin Lymphoma ... more >> Diffuse Large B-cell Lymphoma Mantle Cell Lymphoma Follicular Lymphoma Peripheral T-cell Lymphoma Collapse << | Phase 1 | Completed | - | United States, Massachusetts ... more >> Massachusetts General Hospital Boston, Massachusetts, United States, 02114 Beth-Israel Deaconess Medical Center Boston, Massachusetts, United States, 02115 Dana Farber Cancer Institute Boston, Massachusetts, United States, 02215 Collapse << |
靶点 | Description | IC50 |
---|---|---|
HDAC | IC50:27nM |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网