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CAS No.: 1026016-83-0
Synonyms: (+)-TBZ;(3R,11bR)-TBZ;(3R,11bR)-Tetrabenazine
Tetrabenazine (+)- is a potent, selective and reversible VMAT-2 (vesicular monoamine transporter-2) inhibitor with Ki value of 100 nM.
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT03567291 | Tourette Syndrome | Phase 3 | Recruiting | May 22, 2021 | United States, Alabama ... more >> Teva Investigational Site 046-0104 Recruiting Dothan, Alabama, United States, 36303 United States, California Teva Investigational Site 046-0101 Recruiting Sacramento, California, United States, 95815 United States, Georgia Teva Investigational Site 046-0116 Recruiting Atlanta, Georgia, United States, 30331 United States, New York Teva Investigational Site 046-0102 Recruiting Rochester, New York, United States, 14618 United States, Texas Teva Investigational Site 060-0163 Recruiting Fort Worth, Texas, United States, 76104 United States, Washington Teva Investigational Site 060-0162 Recruiting Everett, Washington, United States, 98201-4077 Canada Teva Investigational Site 046-0201 Recruiting Ajax, Canada, L1Z0M1 Teva Investigational Site 046-0202 Recruiting Ottawa, Canada, K2G 1W2 Collapse << |
NCT01688037 | - | - | Completed | - | - |
NCT01688037 | Tardive Dyskinesia | Phase 2 | Completed | - | - |
实验方案
技术信息
CAS号 | 1026016-83-0 | 储存条件 |
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分子式 | C19H27NO3 | 运输 | 蓝冰 | |||
分子量 | 317.42 | 别名 | (+)-TBZ;(3R,11bR)-TBZ;(3R,11bR)-Tetrabenazine;Tetrabenazine ((+)-);(+)-丁苯那嗪 | |||
溶解度 |
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动物实验配方 |