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CAS No.: 500017-70-9
DC_517 is a selective non-nucleoside inhibitor of DNA methyltransferase 1 (DNMT1) (IC50 = 1.7 μM).
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00032630 | - | - | Completed | - | - |
NCT00032630 | Ischemic Heart Disease | Phase 3 | Completed | - | United States, California ... more >> VA Palo Alto Health Care System Palo Alto, California, United States, 94304-1290 VA Medical Center, San Francisco San Francisco, California, United States, 94121 VA Greater Los Angeles HCS, Sepulveda Sepulveda, California, United States, 91343 United States, Colorado VA Eastern Colorado Health Care System, Denver Denver, Colorado, United States, 80220 United States, District of Columbia VA Medical Center, DC Washington, District of Columbia, United States, 20422 United States, Florida North Florida/South Georgia Veterans Health System Gainesville, Florida, United States, 32608 VA Medical Center, Miami Miami, Florida, United States, 33125 James A. Haley Veterans Hospital, Tampa Tampa, Florida, United States, 33612 United States, New Mexico New Mexico VA Health Care System, Albuquerque Albuquerque, New Mexico, United States, 87108-5153 United States, North Carolina VA Medical Center, Asheville Asheville, North Carolina, United States, 28805 VA Medical Center, Durham Durham, North Carolina, United States, 27705 United States, Ohio VA Medical Center, Cleveland Cleveland, Ohio, United States, 44106 United States, Oregon VA Medical Center, Portland Portland, Oregon, United States, 97201 United States, Pennsylvania VA Pittsburgh Health Care System Pittsburgh, Pennsylvania, United States, 15240 United States, Texas VA North Texas Health Care System, Dallas Dallas, Texas, United States, 75216 VA South Texas Health Care System, San Antonio San Antonio, Texas, United States, 78229 United States, Wisconsin Zablocki VA Medical Center, Milwaukee Milwaukee, Wisconsin, United States, 53295-1000 Collapse << |
实验方案
技术信息
CAS号 | 500017-70-9 | 储存条件 |
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分子式 | C33H35N3O2 | 运输 | 蓝冰 | |
分子量 | 505.65 | 别名 |