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CAS No.: 193022-04-7
Synonyms: Ro 1130830;RS 130830
CTS-1027 is a potent small molecule inhibitor of MMPs (IC50=0.4 nM/0.6 nM for MMP2/MMP13), displaying > 1,000 fold selectivity over MMP1.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01273064 | Hepatitis C | Phase 2 | Terminated(Risk-benefit ratio) | - | - |
NCT01273064 | - | - | Terminated(Risk-benefit ratio) | - | - |
NCT00925990 | Hepatitis C | Phase 2 | Completed | - | - |
实验方案
技术信息
CAS号 | 193022-04-7 | 储存条件 |
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分子式 | C19H20ClNO6S | 运输 | 蓝冰 | |
分子量 | 425.88 | 别名 | Ro 1130830;RS 130830 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01273064 | Hepatitis C | Phase 2 | Terminated(Risk-benefit ratio) | - | - |
NCT01273064 | - | - | Terminated(Risk-benefit ratio) | - | - |
NCT00925990 | Hepatitis C | Phase 2 | Completed | - | - |
NCT00925990 | - | - | Completed | - | - |
NCT01051921 | Hepatitis C | Phase 2 | Completed | - | United States, California ... more >> Scripps Clinic La Jolla, California, United States, 92037 VA Medical Center, San Diego San Diego, California, United States, 92161 United States, Colorado University of Colorado Health Science Center Denver, Colorado, United States, 80262 South Denver Gastroenterology Englewood, Colorado, United States, 80113 United States, Georgia Digestive Healthcare of Georgia Atlanta, Georgia, United States, 30309 United States, Louisiana Tulane University Health Sciences Center New Orleans, Louisiana, United States, 70112 United States, Michigan Henry Ford Medical Center-Columbus Novi, Michigan, United States, 48377 United States, Minnesota MN Clinical Research Center Plymouth, Minnesota, United States, 55446 United States, Missouri St. Louis University St. Louis, Missouri, United States, 63104 United States, Ohio Consultants of Clinical Research, Ohio GI and Liver Institute Cincinnati, Ohio, United States, 45219 United States, Texas Advanced Liver Therapies - Baylor College of Medicine Houston, Texas, United States, 77030 VA Medical Center, Houston Houston, Texas, United States, 77030 United States, Utah University of Utah Health Science Center Salt Lake City, Utah, United States, 84132 United States, Virginia Liver Institute of Virginia Newport News, Virginia, United States, 23602 Puerto Rico Fundacion de Investigacion de Diego Santurce, Puerto Rico, 00909 Collapse << |
NCT00570336 | Chronic Hepatitis C Virus Infe... more >>ction Collapse << | Phase 2 | Completed | - | United States, Alabama ... more >> University of Alabama at Birmingham Birmingham, Alabama, United States, 35233 United States, California Scripps Clinic La Jolla, California, United States, 92037 Kaiser Permanente San Diego, California, United States, 92154 California Pacific Medical Center San Francisco, California, United States, 94115 United States, Colorado University of Colorado Denver Aurora, Colorado, United States, 80045 United States, Florida University of Miami Miami, Florida, United States, 33136 United States, Georgia Digestive Healthcare of Georgia Atlanta, Georgia, United States, 30309 United States, Louisiana Tulane University Health Sciences Center New Orleans, Louisiana, United States, 70112 United States, Massachusetts Beth Israel Deaconess Medical Center Boston, Massachusetts, United States, 02215 United States, Michigan Henry Ford Health System West Bloomfield, Michigan, United States, 48322 United States, Minnesota Mayo Clinic Rochester, Minnesota, United States, 55905 United States, New York Bronx VA Medical Center Bronx, New York, United States, 10468 Mt. Sinai School of Medicine New York, New York, United States, 10019 United States, North Carolina Duke University Medical Center Durham, North Carolina, United States, 27710 United States, Ohio Consultants of Clinical Research Cincinnati, Ohio, United States, 45219 Cleveland Clinic Cleveland, Ohio, United States, 44195 United States, Texas Advanced Liver Therapies - Baylor College of Medicine Houston, Texas, United States, 77030 VAMC - Baylor College of Medicine Houston, Texas, United States, 77030 United States, Virginia McGuire Hospital DVAMC Richmond, Virginia, United States, 23249 Collapse << |
NCT01051921 | - | - | Completed | - | - |
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