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CAS No.: 1166227-08-2
Synonyms: A66
A66 is a potent and specific p110α inhibitor with IC50 of 32 nM, > 100 fold selectivity for p110α over other class-I PI3K isoforms.
生物活性
靶点 | PI3Kα IC50:32nM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01898520 | Cerebral Palsy | Phase 3 | Completed | - | Czechia ... more >> Center 14 Prague, Czechia Israel Center 7 Tel Aviv, Israel Center 8 Tel Hashomer, Israel United Kingdom Center 2 Bristol, United Kingdom Center 6 Cambridge, United Kingdom Center 10 Exeter, United Kingdom Center 13 Glasgow, United Kingdom Center 3 Liverpool, United Kingdom Center 1 London, United Kingdom Center 5 London, United Kingdom Center 12 Norwich, United Kingdom Center 9 Nottingham, United Kingdom Center 11 Salisbury, United Kingdom Center 4 Sheffield, United Kingdom Collapse << |
NCT02391649 | Schizophrenia ... more >> Psychotic Disorders Collapse << | Not Applicable | Active, not recruiting | March 31, 2019 | Hong Kong ... more >> Li Ka Shing Specialty OPD Sha Tin, NT, Hong Kong TM Psy Centre Tuen Mun, NT, Hong Kong Collapse << |
NCT03528135 | Human Immunodeficiency Virus ... more >> Sexually Transmitted Infections Anxiety Depression Substance Use Disorders Collapse << | Not Applicable | Recruiting | April 30, 2019 | United States, Texas ... more >> Avenue 360, University of Houston Recruiting Houston, Texas, United States, 77204 Contact: Joe C Fuentes, MBA 832-384-1389 jfuentes@avenue360.org Collapse << |
实验方案
技术信息
CAS号 | 1166227-08-2 | 储存条件 |
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分子式 | C17H23N5O2S2 | 运输 | 蓝冰 | |||||||
分子量 | 393.53 | 别名 | A66 | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01898520 | Cerebral Palsy | Phase 3 | Completed | - | Czechia ... more >> Center 14 Prague, Czechia Israel Center 7 Tel Aviv, Israel Center 8 Tel Hashomer, Israel United Kingdom Center 2 Bristol, United Kingdom Center 6 Cambridge, United Kingdom Center 10 Exeter, United Kingdom Center 13 Glasgow, United Kingdom Center 3 Liverpool, United Kingdom Center 1 London, United Kingdom Center 5 London, United Kingdom Center 12 Norwich, United Kingdom Center 9 Nottingham, United Kingdom Center 11 Salisbury, United Kingdom Center 4 Sheffield, United Kingdom Collapse << |
NCT02391649 | Schizophrenia ... more >> Psychotic Disorders Collapse << | Not Applicable | Active, not recruiting | March 31, 2019 | Hong Kong ... more >> Li Ka Shing Specialty OPD Sha Tin, NT, Hong Kong TM Psy Centre Tuen Mun, NT, Hong Kong Collapse << |
NCT03528135 | Human Immunodeficiency Virus ... more >> Sexually Transmitted Infections Anxiety Depression Substance Use Disorders Collapse << | Not Applicable | Recruiting | April 30, 2019 | United States, Texas ... more >> Avenue 360, University of Houston Recruiting Houston, Texas, United States, 77204 Contact: Joe C Fuentes, MBA 832-384-1389 jfuentes@avenue360.org Collapse << |
NCT01046383 | NON-SMALL CELL LUNG CANCER | Phase 3 | Terminated(Slower than anticip... more >>ated recruitment) Collapse << | - | Canada, British Columbia ... more >> British Columbia Cancer Agency Vancouver, British Columbia, Canada, V5Z 1L3 Canada, Ontario Juravinski Cancer Centre Hamilton, Ontario, Canada, L8V 5C2 Canada, Quebec CHUM - Hopital Notre Dame Montreal, Quebec, Canada, H2L 4M1 Jewish General Hospital Montreal, Quebec, Canada, H3T 1E2 Canada, Saskatchewan Allan Blair Cancer Centre Regina, Saskatchewan, Canada, S4T 7T1 Collapse << |
NCT03611478 | Mental Fatigue ... more >> Cognitive Function Mood Collapse << | Phase 2 | Recruiting | May 2019 | Australia, Victoria ... more >> Centre for Human Psychopharmacology, Swinburne University of Technology Recruiting Hawthorn, Victoria, Australia, 3122 Contact: Naomi L Perry, PhD +61 3 9214 8930 nlperry@swin.edu.au Collapse << |
NCT02283437 | Schizophrenia Spectrum Disorde... more >>rs Family Caregivers Collapse << | Not Applicable | Active, not recruiting | December 31, 2018 | Hong Kong ... more >> KH; LKS Specialty OPD Shatin And Mongkok, NT/Kln, Hong Kong Li Ka Shing Specialty OPD Sha Tin, NT, Hong Kong Collapse << |
NCT01497015 | Breast Cancer | Not Applicable | Completed | - | United States, Indiana ... more >> Indiana University Indianapolis, Indiana, United States, 46202 Collapse << |
NCT03726996 | Infantile Neuroaxonal Dystroph... more >>y Collapse << | Phase 4 | Not yet recruiting | November 30, 2020 | United States, North Carolina ... more >> Duke University Health Center Not yet recruiting Durham, North Carolina, United States, 27710 Contact: Janet Wootton, RN 919-668-4809 janet.wootton@duke.edu Collapse << |
NCT03255590 | Cerebral Stroke | Not Applicable | Recruiting | December 2018 | United States, Maryland ... more >> Kennedy Krieger Institute Recruiting Baltimore, Maryland, United States, 21205 Contact: Manuel Anaya, MD 443-923-2723 BrainStimulationLab@jhmi.edu Contact: Peggy Foltyn (410) 502-2446 pfoltyn@jhmi.ed Collapse << |
NCT01578850 | Rheumatoid Arthritis | Phase 4 | Completed | - | - |
NCT01953653 | HIV Infection | Not Applicable | Completed | - | United States, Colorado ... more >> Children's Hospital of Denver Aurora, Colorado, United States, 80045 United States, Michigan Wayne State University Detroit, Michigan, United States, 48201 United States, Pennsylvania Childrens Hospital of Philadelphia Philadelphia, Pennsylvania, United States, 19104 Collapse << |
NCT02560935 | Sickle Cell Disease ... more >> Stroke Collapse << | Phase 3 | Active, not recruiting | December 2021 | Nigeria ... more >> Barau Dikko Teaching Hospital/Kaduna State University Kaduna, Nigeria Aminu Kano Teaching Hospital Kano, Nigeria Murtala Muhammad Specialist Hospital Kano, Nigeria Collapse << |
NCT03555474 | Strokes Thrombotic | Not Applicable | Completed | - | - |
NCT01578850 | - | - | Completed | - | - |
NCT03371940 | Type2 Diabetes ... more >> Depression Collapse << | Not Applicable | Completed | - | United States, Indiana ... more >> Indiana University Indianapolis, Indiana, United States, 46202 United States, Ohio Ohio University Athens, Ohio, United States, 45701 United States, West Virginia West Virginia University Morgantown, West Virginia, United States, 26506 Collapse << |
NCT03663179 | Attention Deficit Disorder Wit... more >>h Hyperactivity (ADHD) Collapse << | Not Applicable | Recruiting | June 2019 | United States, Pennsylvania ... more >> University of Pennsylvania Recruiting Philadelphia, Pennsylvania, United States, 19104 Contact: Mary Falcone, PhD 215-746-3782 mfalc@pennmedicine.upenn.edu Contact: Leah Bernardo, BA 215-746-7162 lleah@pennmedicine.upenn.edu Principal Investigator: Caryn Lerman, PhD Sub-Investigator: Mario Cristancho, MD Sub-Investigator: Anthony Rostain, MD Sub-Investigator: James Loughead, PhD Sub-Investigator: Rebecca Ashare, PhD Sub-Investigator: Roy Hamilton, MD Sub-Investigator: J. Russell Ramsay, PhD Collapse << |
NCT01590433 | Obesity | Phase 4 | Active, not recruiting | June 2019 | United States, Massachusetts ... more >> Beth Israel Deaconess Medical Center Boston, Massachusetts, United States, 02215 Collapse << |
NCT01773369 | Perinatal Stroke | Not Applicable | Active, not recruiting | December 2021 | Canada, Alberta ... more >> Alberta Children's Hospital Calgary, Alberta, Canada University of Alberta Edmonton, Alberta, Canada, T6G 2G4 Collapse << |
NCT03672877 | Spastic Diplegia ... more >> Periventricular Leukomalacia Collapse << | Not Applicable | Recruiting | December 31, 2024 | Canada, Alberta ... more >> Alberta Children's Hospital Not yet recruiting Calgary, Alberta, Canada, T3B 6A8 Contact: Donna Livingstone, BScPT 780-492-4858 carre@ualberta.ca Principal Investigator: Elizabeth Condliffe University of Alberta Recruiting Edmonton, Alberta, Canada, T6G 2G4 Contact: Donna Livingstone, BScPT 780-492-4858 carre@ualberta.ca Principal Investigator: Jaynie Yang, PhD Collapse << |
NCT03672864 | Perinatal Stroke | Not Applicable | Recruiting | December 2022 | Canada, Alberta ... more >> Alberta Children's Hospital Not yet recruiting Calgary, Alberta, Canada, T3B 6A8 Contact: Donna Livingstone, BScPT 780-492-4858 carre@ualberta.ca Principal Investigator: Elizabeth Condliffe, MD, Phd Glenrose Rehabilitation Hospital Recruiting Edmonton, Alberta, Canada Contact: Donna Livingstone 780-492-4858 carre@ualberta.ca Canada, Ontario Children's Hospital of Eastern Ontario Not yet recruiting Ottawa, Ontario, Canada Contact: Donna Livingstone, BScPT 780-492-4858 carre@ualberta.ca Principal Investigator: Anna McCormick, MD Collapse << |
NCT02304302 | Down Syndrome ... more >> Intellectual Disability Collapse << | Phase 2 | Recruiting | December 2019 | United States, Ohio ... more >> University Hospitals Case Medical Center Recruiting Cleveland, Ohio, United States, 44106 Contact: Melissa R Stasko, JD 216-844-7281 Melissa.Stasko@case.edu Contact: Alberto C Costa, MD, PhD (216) 844-7395 Alberto.Costa@case.edu Principal Investigator: Alberto C Costa, MD, PhD Sub-Investigator: Nancy J Roizen, MD Sub-Investigator: Stephen L Ruedrich, MD Sub-Investigator: Hudson G Taylor, PhD Sub-Investigator: Katherine Koenig, PhD Sub-Investigator: Richard Boada, PhD Brazil Sociedade Beneficente Israelita Brasileira Albert Einstein Recruiting São Paulo, SP, Brazil, 05652- 900 Contact: Fernanda F Assir, MS +1 55 11 2151-0724 ext 70724 fernanda.assir@einstein.br Principal Investigator: Ana C Brandão, MD Sub-Investigator: Patrícia Salmona, MD Sub-Investigator: Guilherme A Silveira, MD Collapse << |
NCT02096354 | Colorectal Neoplasms | Phase 2 | Active, not recruiting | January 2019 | United States, California ... more >> UCSD Moores Cancer Center La Jolla, California, United States, 92093 Stanford University Stanford, California, United States, 94305 United States, Hawaii Kaiser Permanete Honolulu, Hawaii, United States, 96819 United States, Maryland Walter Reed National Military Medical Center Bethesda, Maryland, United States, 20889 Aquilino Cancer Center, Maryland Oncology and Hematology PA Rockville, Maryland, United States, 20850 Collapse << |
NCT03166293 | Spastic Diplegia | Not Applicable | Active, not recruiting | December 31, 2019 | Canada, Alberta ... more >> Alberta Children's Hospital Calgary, Alberta, Canada University of Alberta Edmonton, Alberta, Canada, T6G 2G4 Collapse << |
NCT02475304 | Psoriatic Arthritis | Phase 2 | Withdrawn(Difficulties to enro... more >>l patients) Collapse << | June 2017 | Sweden ... more >> Department of Rheumatology, Skåne University Hospital Malmö, Sweden, 20502 Collapse << |
NCT01074359 | Neuromuscular Disease | Phase 2 | Terminated(Terminated for Comm... more >>ercial Reasons. There were no safety issues involved in the decision to terminate the study.) Collapse << | - | United Kingdom ... more >> University of Newcastle upon Tyne Newcastle, Framlington Place, United Kingdom, NE2 4HH Collapse << |
NCT02176304 | Knee Osteoarthritis | Phase 4 | Completed | - | Puerto Rico ... more >> University of Puerto Rico School Of Medicine Outpatient Clinics San Juan, Puerto Rico, 00918 Collapse << |
靶点 | Description | IC50 |
---|---|---|
PI3Kα | IC50:32nM |
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