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Opioid Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN18678 | [D-Ala2]leucine-enkephalin | 64963-01-5 | [D-Ala2]Leucine-Enkephalin is a potent, long-acting Leu-enkephalin analog agonist of delta opioid receptor. |
| CSN12642 | Trimebutine maleate | 34140-59-5 | Trimebutine Maleate is an agonist effect on peripheral μ, k and δ opiate receptors, and also shows antimuscarinic effect. |
| CSN12147 | Trimebutine | 39133-31-8 | Trimebutine is an agonist effect on peripheral μ, k and δ opiate receptors, and also shows antimuscarinic effect. |
| CSN21185 | SR17018 | 2134602-45-0 | SR17018 is brain-penetrant μ-opioid receptor agonist EC50 of 97 nM. |
| CSN17907 | Nalfurafine hydrochloride | 152658-17-8 | Nalfurafine HCl is a moderately selective kappa opioid receptor agonist. |
| CSN11162 | Tyr-Gly-Gly-Phe-Met-OH | 58569-55-4 | Met-enkephalin is an Opioid related peptide work as a potent agonist of the δ-opioid receptor, and to a lesser extent the μ-opioid receptor, with little to no effect on the κ-opioid receptor. |
| CSN11381 | 3-(3-Ethyl-1-methylazepan-3-yl)phenol hydrochloride | 59263-76-2 | Meptazinol HCl is both a partial agonist of μ1 opioid receptor and an AChE inhibitor. |
| CSN17469 | (R)-1-(1-(1-Methylcyclooctyl)piperidin-4-yl)-2-(piperidin-3-yl)-1H-benzo[d]imidazole trihydrochloride | 1108147-88-1 | MCOPPB 3HCl is a nociceptin receptor agonist with pKi of 10.07, displaying weaker activity at other opioid receptors. |
| CSN17719 | LY2795050 | 1346133-08-1 | LY2795050 is a selective κ-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo. |
| CSN11328 | Loperamide HCl | 34552-83-5 | Loperamide HCl is a potent and selective μ-opioid receptor agonist. |
| CSN16622 | JTC-801 | 244218-51-7 | JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, and weakly inhibits receptors δ, κ, and μ. |
| CSN18435 | JDTic 2HCl | 785835-79-2 | JDTic 2HCl is a highly selective antagonist for the κ-opioid receptor without affecting the μ- or δ-opioid receptors. |
| CSN19796 | N-((3,5-Difluoro-3'-(1H-1,2,4-triazol-5-yl)-[1,1'-biphenyl]-4-yl)methyl)-2,3-dihydro-1H-inden-2-amine | 1007573-18-3 | GSK-1521498 is a μ-opioid receptor antagonist. It has been shown to attenuate reward-driven compulsive behaviours, such as stimulant drug seeking or binge eating, in animals and humans. |
| CSN10947 | Ethyl 1-methyl-4-phenylazepane-4-carboxylate | 77-15-6 | Ethoheptazine is an opioid analgesic from the phenazepane family. |
| CSN19110 | Cebranopadol ((1α,4α)stereoisomer) | 863513-93-3 | Cebranopadol(1α,4α)stereoisomer is a stereoisomer of cebranopadol. |
| CSN13503 | Cebranopadol | 863513-91-1 | Cebranopadol is an analgesic NOP and opioid receptor agonist with Kis/EC50s of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, 18 nM/110 nM for human NOP, MOP, KOP and delta-opioid peptide (DOP) receptor, respectively. |
| CSN17791 | BAN ORL 24 | 1401463-54-4 | BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively). |
| CSN13513 | Alvimopan | 156053-89-3 | Alvimopan is a peripherally selective opioid mu receptor antagonist. |
| CSN13650 | Alvimopan dihydrate | 170098-38-1 | Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. |
| CSN12425 | ADL-5859 Hydrochloride | 850173-95-4 | ADL-5859 HCl is both a δ-opioid receptor agonist (Ki=0.84 nM, EC50=20 nM) and selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel with IC50 value of 78 µM. |
| CSN18860 | (R)-ZINC-3573 | 2089389-15-9 | (R)-ZINC-3573 can activate endogenous MRGPRX2 in a human mast cell line and induce degranulation and calcium release. |
| CSN11317 | (1R,2S,5R)-2-Isopropyl-5-methylcyclohexanol | 2216-51-5 | (-)-Menthol is a natural product obtained from the oils of corn mint, peppermint, or other mints, as a weak kappa opioid receptor agonist. It has local anesthetic and counterirritant qualities, and used to relieve minor throat irritation. |
| CSN19330 | (41S,7aS,13aR,13bR)-Dodecahydro-1H-dipyrido[2,1-f:3',2',1'-ij][1,6]naphthyridin-10(41H)-one | 519-02-8 | (+)-Matrine is a naturally occuring κ-opioid and μ-opioid receptor agonist. |
| CSN50018 | 2-((3-(2,3-Dichlorophenoxy)propyl)amino)ethan-1-ol hydrochloride | 1009555-55-8 |
