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Histamine Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN12228 | Zaltidine | 85604-00-8 | Zaltidine is a H2-receptor antagonist, which has the antisecretory action. |
| CSN12374 | Tripelennamine HCl | 154-69-8 | Tripelennamine HCl is an antagonist of H1-receptor that used as a psychoactive drug with antipruritic activity. |
| CSN12316 | Rupatadine Fumarate | 182349-12-8 | Rupatadine fumarate is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively. |
| CSN11869 | Roxatidine acetate | 78628-28-1 | Roxatidine acetate is a specific and competitive histamine H2 receptor antagonist drug that is used to treat gastric ulcers, Zollinger–Ellison syndrome, erosive esophagitis, gastro-oesophageal reflux disease, and gastritis. |
| CSN13086 | Roxatidine Acetate HCl | 93793-83-0 | Roxatidine acetate HCl is a slective antagonist of histamin H2 receptor. |
| CSN13516 | N-(2-(((5-((Dimethylamino)methyl)furan-2-yl)methyl)thio)ethyl)-N'-methyl-2-nitroethene-1,1-diamine hydrochloride | 66357-59-3 | Ranitidine HCl is an antagonist of histamine H2-receptor that can inhibit stomach acid production. |
| CSN11722 | Pimethixene | 314-03-4 | Pimethixene is an antihistamine and anticholinergic agent, that is often used to treat hyperactivity, anxiety, sleep disorders, and allergy. |
| CSN11691 | Pheniramine maleate | 132-20-7 | Pheniramine maleate can acts as an antihistamine and vasoconstrictor. |
| CSN11668 | Pemirolast potassium | 100299-08-9 | Pemirolast potassium is an antagonist of histamine H1 and mast cell stabilizer with antiallergic effect. |
| CSN11604 | Olopatadine HCl | 140462-76-6 | Olopatadine HCl can block the release of histamine (IC50 = 559 µM) and stabilize mast cell. |
| CSN11565 | Nizatidine | 76963-41-2 | Nizatidine is an antagonist of histamine H2 receptor that can inhibit the secretion of gastric acid. |
| CSN12482 | Mizolastine | 108612-45-9 | Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions. |
| CSN11437 | Mianserin | 24219-97-4 | Mianserin is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant. |
| CSN10479 | 2-Methyl-1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyrazino[1,2-a]azepine hydrochloride | 21535-47-7 | Mianserin HCl is inverse agonist of H1 receptor and can be act as a psychoactive agent of the tetracyclic antidepressant. |
| CSN11423 | Metiamide | 34839-70-8 | Metiamide is a histamine H2-receptor antagonist developed from another H2 antagonist, burimamide. |
| CSN11382 | Mequitazine | 29216-28-2 | Mequitazine is a potent, nonsedative and long-acting histamine H1 antagonist. |
| CSN11809 | Mepyramine maleate | 59-33-6 | Mepyramine maleate is an antagonist of histamine H1 receptor. |
| CSN11366 | 1-((4-Chlorophenyl)(phenyl)methyl)-4-(3-methylbenzyl)piperazine dihydrochloride | 1104-22-9 | Meclizine 2HCl is a histamine H1 receptor antagonist with Ki of 250 nM and is used to treat nausea and motion sickness. |
| CSN12956 | Ethyl 4-(8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)piperidine-1-carboxylate | 79794-75-5 | Loratadine is an inverse agonist of peripheral histamine H1-receptor with IC50 of > 32 μM. |
| CSN11321 | Lodoxamide tromethamine | 63610-09-3 | Lodoxamide tromethamine is used as an ophthalmic solution that specially applying to the eye. |
| CSN13135 | Levodropropizine | 99291-25-5 | Levodropropizine is a histamine receptor inhibitor, and is an effective and very well tolerated peripheral antitussive drug. |
| CSN11264 | Lafutidine | 118288-08-7 | Lafutidine is an antagonist of histamine H(2)-receptor that inhibits gastric acid secretion. |
| CSN11177 | Hydroxyzine pamoate | 10246-75-0 | Hydroxyzine pamoate is a histamine H1-receptor antagonist. |
| CSN11153 | Histamine Diphosphate | 51-74-1 | Histamine phosphate can dilate arteries and capillaries mediated by H1- and H2-receptors. |
| CSN13756 | Histamine 2HCl | 56-92-8 | Histamine 2HCl is the 2HCl form of histamine which is an organic nitrogen compound that articipates in immune responses and inflammatory reactions and also can be used as neurotransmitters |
| CSN11010 | 2-(4-(1-Hydroxy-4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)butyl)phenyl)-2-methylpropanoic acid | 83799-24-0 | Fexofenadine is an antihistamine pharmaceutical drug used in the treatment of allergy symptoms, such as hay fever, nasal congestion, and urticaria. |
| CSN12462 | Fexofenadine HCl | 153439-40-8 | Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM. |
| CSN10917 | Epinastine HCl | 108929-04-0 | Epinastine HCl is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis. |
| CSN10884 | Ebrotidine | 100981-43-9 | Ebrotidine is a competitive H2-receptor antagonist (Ki= 127.5 nM) with a potent antisecretory activity and evidenced gastroprotection. |
| CSN10883 | Ebastine | 90729-43-4 | Ebastine is a selective H1-histamine receptor antagonist. |
| CSN10864 | Doxylamine succinate | 562-10-7 | Doxylamine Succinate Salt is an antihistamine which inhibits histamine H1 receptors. It can be used as a short-term sedative and anticholinergic agent. |
| CSN12731 | Dimenhydrinate | 523-87-5 | Dimenhydrinate is an anti-emetic and anti-histamine. |
| CSN10783 | Dexchlorpheniramine maleate | 2438-32-6 | Dexchlorpheniramine maleate is an antihistamine, with anticholinergic properties, used to treat allergic conditions. |
| CSN10775 | Desloratadine | 100643-71-8 | Desloratadine is an antagonist of histamine H1 receptor that is used to treat allergies. |
| CSN10757 | Decloxizine | 3733-63-9 | Decloxizine is a histamine 1 receptor antagonist. |
| CSN13624 | 2-(2-(4-Benzhydrylpiperazin-1-yl)ethoxy)ethanol dihydrochloride | 13073-96-6 | Decloxizine 2HCl is a histamine 1 receptor antagonist. |
| CSN10664 | Clemizole | 442-52-4 | Clemizole is an antagonist of H1 histamine receptor that can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication. |
| CSN10663 | (R)-2-(2-((R)-1-(4-Chlorophenyl)-1-phenylethoxy)ethyl)-1-methylpyrrolidine fumarate | 14976-57-9 | Clemastine fumarate is a selective antagonist of histamine H1 receptor with IC50 of 3 nM. |
| CSN12549 | 1-Benzhydryl-4-cinnamylpiperazine | 298-57-7 | Cinnarizine, an antihistamine, can block calcium channel and promote cerebral blood flow. It is used to treat post-trauma cerebral symptoms and cerebral arteriosclerosis. |
| CSN10624 | Chlorphenoxamine | 77-38-3 | Chlorphenoxamine is an antihistamine and anticholinergic and can be used as antipruritic and antiparkinsonian agent. |
| CSN10600 | Cetirizine | 83881-51-0 | Cetirizine, a second-generation antihistamine, is a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria. |
| CSN12995 | Cetirizine 2HCl | 83881-52-1 | Cetirizine 2HCl, a metabolite of hydroxyzine, is racemic selective and inverse agonist of H1 receptor used in the treatment of allergies and hay fever. |
| CSN10548 | Carbinoxamine maleate salt | 3505-38-2 | Carbinoxamine maleate is a blocker of histamine-H1 receptor with antihistamine and anticholinergic effects. |
| CSN10500 | Buclizine 2HCl | 129-74-8 | Buclizine 2HCl, the derivative of piperazine, is an antihistamine and anticholinergic agent. |
| CSN10492 | Brompheniramine maleate | 980-71-2 | Brompheniramine maleate is an antagonist of histamine H1 receptors. |
| CSN10402 | 2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoic acid | 202189-78-4 | Bilastine selectively antagonizes histamine H1 receptor and it is used to treat allergic rhinoconjunctivitis and urticaria. |
| CSN10415 | Bepotastine besilate | 190786-44-8 | Bepotastine besilate is a selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7. |
| CSN10365 | Azatadine | 3964-81-6 | Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively. |
| CSN10364 | Azatadine dimaleate | 3978-86-7 | Azatadine dimaleate is an inhibitor of histamine and cholinergic with IC50 of 6.5 nM and 10 nM, respectively. |
| CSN12361 | ABT-239 | 460746-46-7 | ABT-239 is a highly efficacious, non-imidazole class of H3R antagonist. |
