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Cancer

货号 产品名 CAS号 信息
CSN22566 Vorasidenib 1644545-52-7 Vorasidenib is an isocitrate dehydrogenase (IDH) inhibitor.
CSN23793 SGC-GAK-1 2226517-76-4
CSN23766 BIBF0775 334951-90-5 BIBF0775 is an inhibitor of transforming growth factor β receptor I (TGFβRI) by soaking into the kinase domain of TGFβRI.
CSN23771 BAY8002 724440-27-1
CSN23239 Guanosine 118-00-3 Guanosine is a purine nucleoside.
CSN22468 MOZ-IN-2 2055397-88-9 MOZ-IN-2 is an inhibitor of protein MOZ, a member of histone acetyltransferases, with an IC50 of 125 μM.
CSN22526 Tucidinostat 1616493-44-7 Tucidinostat is an inhibitor of HDAC enzymes class I (HDAC1/2/3) and class IIb (HDAC10) inhibitor with IC50s of 95, 160, 67 and 78 nM, espectively.
CSN22506 SJ000291942 425613-09-8 SJ000291942 is an activator of the canonical bone morphogenetic proteins (BMP) signaling pathway. BMPs are members of the transforming growth factor beta (TGFβ) family of secreted signaling molecules.
CSN22537 α-2,3-sialyltransferase-IN-1 881179-06-2 α-2,3-sialyltransferase-IN-1 is a noncompetitive α-2,3-sialyltransferase inhibitor with an IC50 of 6 μM.
CSN22492 PROTAC Linker 1 1835705-53-7 PROTAC Linker 1 is a linker used to link the warhead and the E3 ligase ligand.
CSN22494 QX77 1798331-92-6 QX77 is a chaperone-mediated autophagy (CMA) activator.
CSN22505 SHIN1 2146095-85-2 SHIN1 is a human serine hydroxymethyltransferse 1 and 2 (SHMT1/2) inhibitor with IC50s of 5 and 13 nM, respectively, in an in vitro assay.
CSN22467 WM-1119 2055397-28-7 MOZ-IN-1 is an inhibitor of MOZ which is a member of histone acetyltransferases with IC50 of 0.051 μM.
CSN22532 Vecabrutinib 1510829-06-7 Vecabrutinib is a potent BTK inhibitor, with IC50s of 4.6 nM and 1.1 nM for WT BTK and C481S BTK, respectively, and also inhibits ITK activity (IC50, 24 nM).
CSN22485 PF-06459988 1428774-45-1 PF-06459988 is an irreversible inhibitor of T790M-Containing EGFR Mutants.
CSN22525 Troxacitabine 145918-75-8 Troxacitabine is nucleoside analog with potent anticancer activity.
CSN22507 SLV-2436 2095704-43-9 SLV-2436 is a highly potent and ATP-competitive inhibitor of MNK1 and MNK2 with IC50s of 10.8  nM and 5.4 nM, respectively.
CSN22470 NAV-2729 419547-11-8 NAV-2729 is a selective ARF6 inhibitor with IC50 of 1 μM.
CSN22456 M443 1820684-31-8 M443 is an irreversible and specific inhibitor of MRK, with an IC50<125 nM.
CSN22514 TAK-778 180185-61-9 TAK-778 is a derivative of ipriflavone and has been shown to induce bone growth in in vitro and in vivo models.
CSN22508 SM 16 614749-78-9 SM 16 is an an ATP-competitive ALK5/ALK4 inhibitor with IC50 value between 160 and 620 nM for inhibition of TGF-β1-induced Smad2/3 phosphorylation in cell study.
CSN22460 MAT2A Inhibitor 2201057-10-3 MAT2A inhibitor is a methionine adenosyltransferase 2A (MATA2) inhibitor.
CSN22484 PF-06260182 1415558-82-5 PF-06260182 is a lactam metabolite of crizotinib.
CSN22462 Mcl1-IN-4 1580484-04-3 Mcl1-IN-4 is an inhibitor of Mcl1 with an IC50 of 0.2 μM.
CSN22496 RH1 221635-42-3 RH1 is a potent bioreductive agent with profound anti-cancer activity in vitro and in vivo.
CSN22509 SNT-207707 1064662-40-3 SNT-207707 is a selective, potent and orally active melanocortin MC-4 receptor antagonist with an IC50 of 8 nM (binding) and 5 nM (function) on the MC-4 receptor.
CSN22521 TNF-α-IN-1 444287-49-4 TNF-α-IN-1 is a TNF-α inhibitor extracted from patent US20030096841A1, compound example I-7.
CSN22476 OSW-1 145075-81-6 OSW-1, isolated from Ornithogalum caudatum, is a specific antagonist of osterol-binding protein (OSBP) and OSBP-related protein 4 (ORP4) with GI50s in the nanomolar range in human cancer lines.
CSN22499 Ropidoxuridine 93265-81-7 Ropidoxuridine is an orally available, halogenated thymidine analog and is a potential radiosensitizer for use in human tumors.
CSN22534 WIT 002 240427-90-1 WIT 002 is an antagonist of 20-hydroxyeicosatetraenoic acid (20-HETE).
CSN22501 Rpn11-IN-1 2084867-65-0 Rpn11-IN-1 is a potent and selective inhibitor of proteasome subunit Rpn11 with an IC50 of 390 nM.
CSN22480 Parsaclisib 1426698-88-5 Parsaclisib is a potent and selective PI3Kδ inhibitor, with an IC50 of 1 nM at 1 mM ATP, and shows appr 20,000-fold selectivity for PI3Kα, PI3Kβ, PI3Kγ and 57 other kinases.
CSN22466 ML132 1230628-71-3 ML132 is a potent and selective caspase 1 inhibitor with an IC50 of 0.316 nM.
CSN22502 RR-11a 1361390-56-8 RR-11a is a synthetic enzyme inhibitor of Legumain, an asparaginyl endopeptidase.
CSN22515 Target Protein-binding Moiety 13 1092369-24-8 PROTAC FKBP12-binding moiety 1 is a synthetic ligand for FKBP, used as a warhead ligand for conjugation reactions of PROTAC targeting on FKBP12.
CSN22516 Target Protein-binding Moiety 6 2097512-23-5 PROTAC BRD9-binding moiety 1 is a I-BRD9-based warhead ligand for conjugation reactions of PROTAC targeting on BRD9.
CSN22531 Valemetostat 1809336-39-7 Valemetostat is an antineoplastic agent.
CSN22473 OBE022 2005486-31-5 OBE022 is an oral and selective prostaglandin F2α (PGF2α) receptor antagonist, with Kis of 1 nM, 26 nM for human and rat FP receptors, respectively.
CSN22517 Target Protein-binding Moiety 8 910297-51-7 PROTAC Bcr-Abl-binding moiety 1 is a Dasatinib-based warhead ligand for conjugation reactions of PROTAC targeting on Bcr-Abl.
CSN23328 GDC-0575 1196541-47-5 GDC-0575 is a potent and selective CHK1 inhibitor.
CSN23752 Elemicin 487-11-6 Elemicin is a phenylpropene with anticancer and antifungal activities, it exhibits anticholinergic-like effects in humans.
CSN23754 NFAT Inhibitor 249537-73-3 NFAT Inhibitor is a high-affinity calcineurin-binding peptide that inhibits NFAT (Nuclear Factor of Activated T cells) activation and NFAT-dependent expression of endogenous cytokine genes in T cells.
CSN23770 Aurora Kinase Inhibitor III 879127-16-9
CSN23772 E3 Ligase Ligand-Linker Conjugates 20 1950635-15-0 Thalidomide-O-amido-C8-Amine is a PROTAC block consist of Thalidomide linked to alkyl with Amine functional group for conjugation reactions.
CSN23775 VTX-27 1321924-70-2
CSN23768 E3 ligase Ligand 5 1264754-13-3
CSN22491 PRI-724 1422253-38-0 PRI-724 is a selective inhibitor of the CBP/β-catenin interaction.
CSN24156 E260 1241537-79-0 E260 is an inhibitor of the Fer/FerT kinase with Kd of 0.85 μM, selectively evokes metabolic stress and necrotic death in cancer cells.
CSN24157 666-15 1433286-70-4 666-15 is a potent and cell-permeable inhibitor of cAMP-response element binding protein (CREB) with efficacious anti-cancer activity both in vitro and in vivo.
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