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Apelin Receptor

货号 产品名 CAS号 信息
CSN23653 [Pyr1]-Apelin-13 217082-60-5 [Pyr1]-Apelin-13 is a potent peptide apelin agonist with EC50 of 0.37 nM.
CSN24633 MM 54 1313027-43-8 MM 54 is a potent apelin receptor antagonist with Ki of 82 nM and IC50 of 93 nM.
CSN26194 MM 07 1876450-21-3 MM 07 is a biased apelin receptor agonist, with a KD of 300 nM in CHO-K1 cells and a KD of 172 nM in human heart. It stimulates endothelial NOS phosphorylation and expression, promotes proliferation, and attenuates apoptosis of human pulmonary arterial endothelial cells in vitro.
CSN21287 4-Oxo-6-((pyrimidin-2-ylthio)methyl)-4H-pyran-3-yl 4-nitrobenzoate 877636-42-5 ML221 is a potent apelin receptor (APJ) antagonist with IC50s of 0.70 μM and 1.75 μM in cAMP and β-arrestin assay respectively.
CSN23651 Apelin-13 217082-58-1 Apelin-13 is the endogenous ligand of the orphan G protein-coupled receptor APJ, activates APJ receptor with an EC50 value of 0.37 nM in CHO cells[1][2].
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