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5-HT Receptor
货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
CSN23092 | SB 204070A | 148688-01-1 | SB 204070A is a highly selective 5-HT4 receptor antagonist. |
CSN23091 | SB-203186 HCl | 207572-69-8 | SB 203186 HCl is potent 5-HT4 receptor antagonist with high affinity for human atrial 5-HT4 receptors. |
CSN23066 | Ro 04-6790 | 202466-68-0 | Ro 04-6790 is a potent and selective 5-HT6 receptor antagonist (pKi values are 7.26 and 7.35 at rat and human 5-HT6 receptors respectively). Ro 04-6790 displays no affinity at a range of other receptors (IC50 > 10 μM). |
CSN23059 | Quipazine dimaleate | 150323-78-7 | Quipazine Dimaleate is a selective 5-HT3 receptor agonist. |
CSN23048 | PNU-142633 | 187665-65-2 | PNU 142633 is a very selective, high affinity 5-HT1D receptor agonist with Ki of 6 nM at human 5-HT1D. |
CSN23019 | Org37684 | 213007-95-5 | Org 37684 is an agonist of 5-HT2 receptors. |
CSN23017 | Org-12962 HCl | 210821-63-9 | Org 12962 HCl is a selective 5-HT2C receptor agonist with pEC50 of 7.01. |
CSN23008 | NPS ALX Compound 4a | 299433-10-6 | NPS ALX Compound 4a is a potent and competitive 5-HT6 antagonist with IC50 of 7.2 nM and Ki of 0.2 nM. |
CSN22997 | NAS-181 dimesylate | 1217474-40-2 | NAS-181 is a potent, selective antagonist at the rat 5-HT1B receptor with Ki of 47 nM. |
CSN22996 | Robalzotan hydrochloride | 184674-99-5 | NAD 299 HCl is a selective, high affinity 5-HT1A receptor antagonist with Ki of 0.6 nM in vitro. |
CSN23003 | N-Methylquipazine dimaleate | 171205-17-7 | N-Methylquipazine Dimaleate is a 5-HT3 agonist. |
CSN22975 | ML 10302 HCl | 186826-17-5 | ML 10302 HCl is a potent 5-HT4 partial agonist with EC50 of 4 nM. |
CSN22973 | MK-212 HCl | 61655-58-1 | MK 212 HCl is a 5-HT receptor agonist with IC50 of 0.028 μM. |
CSN22967 | MDL 73005EF hydrochloride | 102908-60-1 | MDL 73005EF HCl is a potent and selective 5-HT1A receptor antagonist. |
CSN22966 | MDL 72832 HCl | 113777-40-5 | MDL 72832 HCl is a potent ligand at 5-HT1A receptors. |
CSN22965 | Bemesetron | 40796-97-2 | MDL 72222 is a 5-HT3 antagonist. |
CSN22963 | Volinanserin | 139290-65-6 | MDL 100907 is a potent and selective 5-HT2A receptor antagonist with Ki of 0.36 nM. |
CSN22962 | m-CPBG hydrochloride | 2113-05-5 | m-Chlorophenylbiguanide HCl is a prototypical potent and selective 5-HT3 receptor agonist. |
CSN22955 | LY 334370 hydrochloride | 199673-74-0 | LY 334370 HCl is a selective 5-HT1F receptor agonist with Ki of 1.87 nM. |
CSN22948 | LP44 HCl | 824958-12-5 | LP 44 is a high affinity 5-HT7 receptor agonist with Ki of 0.22 nM. |
CSN22946 | LP 12 HCl | 1185136-22-4 | LP 12 HCl is a 5-HT7 receptor agonist with Ki of 0.22 nM. |
CSN22876 | L-694,247 | 137403-12-4 | L-694,247 is a selective and extremely potent 5-HT1D receptor agonist. |
CSN22861 | Isamoltane hemifumarate | 874882-92-5 | Isamoltane Hemifumarate is a 5-HT1B antagonist. |
CSN22857 | Ipsapirone | 95847-70-4 | Ipsapirone is a selective 5-HT1A receptor agonist with Ki of 10 nM. |
CSN22856 | Indatraline HCl | 96850-13-4 | Indatraline HCl is a potent 5-HT uptake inhibitor, and also inhibits dopamine and noradrenalin uptake with Ki of 0.42, 1.7 and 5.8 nM, respectively. |
CSN22837 | GR 55562 dihydrochloride | 159533-25-2 | GR 55562 2HCl is a selective competitive 5-HT1B silent antagonist with pKB of 7.3 for human cloned 5-HT1B. |
CSN22835 | GR127935 HCl | 148642-42-6 | GR 127935 HCl is a potent and selective 5-HT1B/1D receptor antagonist with pKi of 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptors. |
CSN22834 | GR125487 sulfamate | 859502-43-5 | GR 125487 Sulfamate is a potent and selective 5-HT4 receptor antagonist with Ki of 0.19 nM for porcine 5-HT4. |
CSN22833 | GR 113808 | 144625-51-4 | GR 113808 is a potent, selective 5-HT4 receptor antagonist with Kd of 0.15 nM for binding to cloned human 5-HT4 receptors. |
CSN22814 | Fananserin | 127625-29-0 | Fananserin is a 5-HT2A receptor antagonist that also displays high affinity at D4 receptors with Ki of 0.26 and 2.93 nM for 5-HT2A and D4, respectively. |
CSN22809 | Eplivanserin hemifumarate | 130580-02-8 | Eplivanserin Hemifumarate is a potent and selective 5-HT2A antagonist with IC50 of 5.8 nM. |
CSN22806 | EMD386088 | 1171123-46-8 | EMD 386088 HCl is a potent 5-HT6 receptor agonist with EC50 of 1.0 nM. |
CSN22795 | DV-7028 hydrochloride | 133364-62-2 | DV 7028 HCl is a selective 5-HT2A receptor antagonist with Ki of 22 nM for at 5-HT2 receptors. |
CSN22793 | DR4485 HCl | 402942-53-4 | DR 4485 HCl is a high affinity and selective 5-HT7 antagonist with pKi of 8.14. |
CSN22776 | CP94253 HCl | 845861-39-4 | CP 94253 HCl is a potent, selective 5-HT1B agonist with Ki of 2 nM. |
CSN22775 | CP 93129 2HCl | 879089-64-2 | CP 93129 2HCl is a potent and highly selective 5-HT1B agonist with Ki of 8.1 nM. |
CSN22769 | CP-135807 | 151272-90-1 | CP 135807 is a selective 5-HT1D receptor agonist. |
CSN22763 | CJ033466 | 519148-48-2 | CJ 033466 is a potent and selective 5-HT4 partial agonist with EC50 of 0.927 nM. |
CSN22761 | Cinanserin HCl | 54-84-2 | Cinanserin HCl is a selective 5-HT2 antagonist. |
CSN22749 | CGS 12066 dimaleate | 109028-10-6 | CGS 12066B Dimaleate is a 5-HT1B full agonist. |